JP2018527397A5 - - Google Patents
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- Publication number
- JP2018527397A5 JP2018527397A5 JP2018515050A JP2018515050A JP2018527397A5 JP 2018527397 A5 JP2018527397 A5 JP 2018527397A5 JP 2018515050 A JP2018515050 A JP 2018515050A JP 2018515050 A JP2018515050 A JP 2018515050A JP 2018527397 A5 JP2018527397 A5 JP 2018527397A5
- Authority
- JP
- Japan
- Prior art keywords
- poly
- less
- olanzapine
- dosage form
- pharmaceutical dosage
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- KVWDHTXUZHCGIO-UHFFFAOYSA-N olanzapine Chemical compound C1CN(C)CCN1C1=NC2=CC=CC=C2NC2=C1C=C(C)S2 KVWDHTXUZHCGIO-UHFFFAOYSA-N 0.000 claims 19
- 229960005017 olanzapine Drugs 0.000 claims 19
- 239000002552 dosage form Substances 0.000 claims 14
- 150000003839 salts Chemical class 0.000 claims 8
- 206010072851 Post-injection delirium sedation syndrome Diseases 0.000 claims 6
- 238000000034 method Methods 0.000 claims 5
- JVTAAEKCZFNVCJ-UWTATZPHSA-N D-lactic acid Chemical compound C[C@@H](O)C(O)=O JVTAAEKCZFNVCJ-UWTATZPHSA-N 0.000 claims 4
- 239000002202 Polyethylene glycol Substances 0.000 claims 4
- 229920001710 Polyorthoester Polymers 0.000 claims 4
- 229920002988 biodegradable polymer Polymers 0.000 claims 4
- 239000004621 biodegradable polymer Substances 0.000 claims 4
- 229920001577 copolymer Polymers 0.000 claims 4
- 239000002745 poly(ortho ester) Substances 0.000 claims 4
- 229920001223 polyethylene glycol Polymers 0.000 claims 4
- 238000013268 sustained release Methods 0.000 claims 3
- 239000012730 sustained-release form Substances 0.000 claims 3
- RKDVKSZUMVYZHH-UHFFFAOYSA-N 1,4-dioxane-2,5-dione Chemical compound O=C1COC(=O)CO1 RKDVKSZUMVYZHH-UHFFFAOYSA-N 0.000 claims 2
- GQLCSJBRVSWWDV-UHFFFAOYSA-N 2-hydroxyacetic acid oxepan-2-one Chemical compound OCC(O)=O.O=C1CCCCCO1 GQLCSJBRVSWWDV-UHFFFAOYSA-N 0.000 claims 2
- VSKXVGWORBZZDY-UHFFFAOYSA-N 2-hydroxypropanoic acid;oxepan-2-one Chemical compound CC(O)C(O)=O.O=C1CCCCCO1 VSKXVGWORBZZDY-UHFFFAOYSA-N 0.000 claims 2
- 102000009027 Albumins Human genes 0.000 claims 2
- 108010088751 Albumins Proteins 0.000 claims 2
- 229920001661 Chitosan Polymers 0.000 claims 2
- 229920002732 Polyanhydride Polymers 0.000 claims 2
- 229920000954 Polyglycolide Polymers 0.000 claims 2
- DHKHKXVYLBGOIT-UHFFFAOYSA-N acetaldehyde Diethyl Acetal Natural products CCOC(C)OCC DHKHKXVYLBGOIT-UHFFFAOYSA-N 0.000 claims 2
- 125000002777 acetyl group Chemical class [H]C([H])([H])C(*)=O 0.000 claims 2
- 239000002253 acid Substances 0.000 claims 2
- 150000007933 aliphatic carboxylic acids Chemical class 0.000 claims 2
- 125000002947 alkylene group Chemical group 0.000 claims 2
- 239000005018 casein Substances 0.000 claims 2
- BECPQYXYKAMYBN-UHFFFAOYSA-N casein, tech. Chemical compound NCCCCC(C(O)=O)N=C(O)C(CC(O)=O)N=C(O)C(CCC(O)=N)N=C(O)C(CC(C)C)N=C(O)C(CCC(O)=O)N=C(O)C(CC(O)=O)N=C(O)C(CCC(O)=O)N=C(O)C(C(C)O)N=C(O)C(CCC(O)=N)N=C(O)C(CCC(O)=N)N=C(O)C(CCC(O)=N)N=C(O)C(CCC(O)=O)N=C(O)C(CCC(O)=O)N=C(O)C(COP(O)(O)=O)N=C(O)C(CCC(O)=N)N=C(O)C(N)CC1=CC=CC=C1 BECPQYXYKAMYBN-UHFFFAOYSA-N 0.000 claims 2
- 235000021240 caseins Nutrition 0.000 claims 2
- 229940022769 d- lactic acid Drugs 0.000 claims 2
- 239000003814 drug Substances 0.000 claims 2
- 238000002347 injection Methods 0.000 claims 2
- 239000007924 injection Substances 0.000 claims 2
- 238000004519 manufacturing process Methods 0.000 claims 2
- 239000000203 mixture Substances 0.000 claims 2
- 229920001308 poly(aminoacid) Polymers 0.000 claims 2
- 229920000747 poly(lactic acid) Polymers 0.000 claims 2
- 229920001606 poly(lactic acid-co-glycolic acid) Polymers 0.000 claims 2
- 229940065514 poly(lactide) Drugs 0.000 claims 2
- 229920002463 poly(p-dioxanone) polymer Polymers 0.000 claims 2
- 229920001610 polycaprolactone Polymers 0.000 claims 2
- 239000004632 polycaprolactone Substances 0.000 claims 2
- 239000000622 polydioxanone Substances 0.000 claims 2
- 229920006149 polyester-amide block copolymer Polymers 0.000 claims 2
- 229920000642 polymer Polymers 0.000 claims 2
- 229920002635 polyurethane Polymers 0.000 claims 2
- 239000004814 polyurethane Substances 0.000 claims 2
- 229920000036 polyvinylpyrrolidone Polymers 0.000 claims 2
- 235000013855 polyvinylpyrrolidone Nutrition 0.000 claims 2
- 239000001267 polyvinylpyrrolidone Substances 0.000 claims 2
- 238000007920 subcutaneous administration Methods 0.000 claims 2
- 239000001993 wax Substances 0.000 claims 2
- 208000020925 Bipolar disease Diseases 0.000 claims 1
- 238000012544 monitoring process Methods 0.000 claims 1
- 201000000980 schizophrenia Diseases 0.000 claims 1
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021110240A JP2021167331A (ja) | 2015-09-21 | 2021-07-01 | 徐放性オランザピン製剤 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562221290P | 2015-09-21 | 2015-09-21 | |
| US62/221,290 | 2015-09-21 | ||
| PCT/US2016/052757 WO2017053346A1 (en) | 2015-09-21 | 2016-09-21 | Sustained release olanzapine formulations |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021110240A Division JP2021167331A (ja) | 2015-09-21 | 2021-07-01 | 徐放性オランザピン製剤 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2018527397A JP2018527397A (ja) | 2018-09-20 |
| JP2018527397A5 true JP2018527397A5 (cg-RX-API-DMAC7.html) | 2019-10-31 |
Family
ID=57047342
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018515050A Pending JP2018527397A (ja) | 2015-09-21 | 2016-09-21 | 徐放性オランザピン製剤 |
| JP2021110240A Pending JP2021167331A (ja) | 2015-09-21 | 2021-07-01 | 徐放性オランザピン製剤 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021110240A Pending JP2021167331A (ja) | 2015-09-21 | 2021-07-01 | 徐放性オランザピン製剤 |
Country Status (21)
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2018172850A1 (en) * | 2017-03-20 | 2018-09-27 | Teva Pharmaceuticals International Gmbh | Sustained release olanzapine formulaitons |
| CN111836615A (zh) * | 2018-01-05 | 2020-10-27 | 英倍尔药业股份有限公司 | 通过精密鼻装置的奥氮平的鼻内递送 |
| AU2020410549A1 (en) * | 2019-12-20 | 2022-04-14 | Alar Pharmaceuticals Inc. | Long-acting injectable formulations of ketamine pamoate salts |
| CN112587505A (zh) * | 2020-10-16 | 2021-04-02 | 长春斯菲尔生物科技有限公司 | 一种奥氮平双羟萘酸盐缓释微粒制剂及其制备方法 |
| WO2025188992A1 (en) * | 2024-03-06 | 2025-09-12 | Neurelis, Inc. | Oral film for rapid active delivery |
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| US7833543B2 (en) | 1995-06-07 | 2010-11-16 | Durect Corporation | High viscosity liquid controlled delivery system and medical or surgical device |
| EA002825B1 (ru) * | 1997-09-30 | 2002-10-31 | Эли Лилли Энд Компани | Препарат 2-метилтиенобензодиазепина |
| US6495164B1 (en) | 2000-05-25 | 2002-12-17 | Alkermes Controlled Therapeutics, Inc. I | Preparation of injectable suspensions having improved injectability |
| US7731947B2 (en) | 2003-11-17 | 2010-06-08 | Intarcia Therapeutics, Inc. | Composition and dosage form comprising an interferon particle formulation and suspending vehicle |
| DK1635875T3 (da) | 2003-06-26 | 2009-01-12 | Psivida Inc | In-situ-geldannende lægemiddeladministrationssystem |
| KR101242486B1 (ko) | 2004-01-12 | 2013-03-13 | 더 트러스티스 오브 더 유니버시티 오브 펜실베니아 | 장기 전달을 위한 제형 및 그의 이용 방법 |
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| NL1026261C2 (nl) | 2004-05-25 | 2005-11-28 | Nanomi B V | Sproei inrichting met een nozzleplaat voorzien van structuren ter bevordering van self-breakup, een nozzleplaat, alsmede werkwijzen ter vervaardiging en toepassing van een dergelijke nozzleplaat. |
| NZ551990A (en) | 2004-06-04 | 2011-01-28 | Camurus Ab | Liquid depot formulations |
| AU2005307797B2 (en) * | 2004-11-16 | 2011-06-02 | Alkermes Pharma Ireland Limited | Injectable nanoparticulate olanzapine formulations |
| EP1874267A1 (en) * | 2005-04-13 | 2008-01-09 | Pfizer Products Inc. | Injectable depot formulations and methods for providing sustained release of poorly soluble drugs comprising nanoparticles |
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| ATE552032T1 (de) * | 2005-07-14 | 2012-04-15 | Lithera Inc | Verbesserte lipolytikum-formulierung mit hinhaltender wirkstofffreigabe für die arealbehandlung von fettgewebe |
| US8852638B2 (en) | 2005-09-30 | 2014-10-07 | Durect Corporation | Sustained release small molecule drug formulation |
| US20070254832A1 (en) * | 2006-02-17 | 2007-11-01 | Pressler Milton L | Methods for the treatment of macular degeneration and related eye conditions |
| WO2007139744A2 (en) | 2006-05-23 | 2007-12-06 | Titan Pharmaceuticals, Inc. | Implantable polymeric device for sustained release of buprenorphine with minimal initial burst |
| KR20140109509A (ko) | 2006-07-11 | 2014-09-15 | 큐피에스 엘엘씨 | 펩타이드의 지속 방출 전달을 위한 의약 조성물 |
| FI20070174A0 (fi) | 2007-02-28 | 2007-02-28 | Delsitech Oy | Menetelmä silikakoostumusten valmistamiseksi, silikakoostumukset ja niiden käytöt |
| KR100805208B1 (ko) | 2007-03-27 | 2008-02-21 | 주식회사 펩트론 | 엑센딘 함유 서방성 제제 조성물, 엑센딘 함유 서방성미립구 및 이의 제조 방법 |
| EP2139458A4 (en) | 2007-04-19 | 2013-01-23 | Dong A Pharm Co Ltd | COMPOSITION OF BIODEGRADABLE MICROSPHERES WITH CONTROLLED RELEASE OF A GLUCOSE REGULATING PEPTIDE AND RELATED FORMULA |
| US10010612B2 (en) | 2007-05-25 | 2018-07-03 | Indivior Uk Limited | Sustained delivery formulations of risperidone compounds |
| ES2324009B1 (es) | 2007-11-23 | 2010-05-21 | Gp Pharm S.A. | Composicion farmaceutica de liberacion sostenida de somatostatina o un analogo suyo. |
| JP5222550B2 (ja) * | 2007-12-27 | 2013-06-26 | 財團法人工業技術研究院 | 徐放性組成物およびその製造方法 |
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| SI2717914T1 (sl) | 2011-06-10 | 2020-07-31 | Ramscor Inc. | Formulacije z zadržanim sproščanjem za dostavo proteinov v oko in postopki njihove priprave |
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| MX364864B (es) | 2012-01-23 | 2019-05-09 | Allergan Inc | Microesferas o microparticulas biodegradables o bioerosionables de liberacion progresiva suspendidas en una formulacion de farmaco inyectable de formacion de deposito solidificante. |
| CN103417492A (zh) * | 2012-05-25 | 2013-12-04 | 上海现代药物制剂工程研究中心有限公司 | 含有奥氮平的生物降解微球制剂及其制备方法 |
| US20140323517A1 (en) | 2013-04-30 | 2014-10-30 | Heron Therapeutics, Inc. | Compositions and methods for injection of a biodegradable polymer-based delivery system |
| WO2014202214A1 (en) | 2013-06-20 | 2014-12-24 | Pharmathen S.A. | Preparation of polylactide-polyglycolide microparticles having a sigmoidal release profile |
| CN103877005A (zh) * | 2014-03-26 | 2014-06-25 | 陈德香 | 一种复方奥氮平皮下埋植缓释剂 |
-
2016
- 2016-09-21 WO PCT/US2016/052757 patent/WO2017053346A1/en not_active Ceased
- 2016-09-21 HU HUE16775424A patent/HUE063850T2/hu unknown
- 2016-09-21 EP EP23193256.7A patent/EP4331570A1/en active Pending
- 2016-09-21 US US15/271,508 patent/US20170079985A1/en not_active Abandoned
- 2016-09-21 IL IL295161A patent/IL295161A/en unknown
- 2016-09-21 PT PT167754241T patent/PT3352735T/pt unknown
- 2016-09-21 CN CN202310947482.0A patent/CN116942677A/zh active Pending
- 2016-09-21 AU AU2016328958A patent/AU2016328958B2/en active Active
- 2016-09-21 PL PL16775424.1T patent/PL3352735T3/pl unknown
- 2016-09-21 MX MX2018003380A patent/MX2018003380A/es unknown
- 2016-09-21 JP JP2018515050A patent/JP2018527397A/ja active Pending
- 2016-09-21 EA EA201890788A patent/EA201890788A1/ru unknown
- 2016-09-21 EP EP16775424.1A patent/EP3352735B1/en active Active
- 2016-09-21 TW TW105130439A patent/TWI798161B/zh active
- 2016-09-21 ES ES16775424T patent/ES2960753T3/es active Active
- 2016-09-21 DK DK16775424.1T patent/DK3352735T3/da active
- 2016-09-21 CA CA2998504A patent/CA2998504C/en active Active
- 2016-09-21 NZ NZ740665A patent/NZ740665A/en unknown
- 2016-09-21 KR KR1020187007791A patent/KR20180054627A/ko not_active Ceased
- 2016-09-21 CN CN201680066464.XA patent/CN108289834A/zh active Pending
- 2016-09-21 AR ARP160102864A patent/AR106085A1/es not_active Application Discontinuation
- 2016-09-21 FI FIEP16775424.1T patent/FI3352735T3/fi active
-
2018
- 2018-03-13 IL IL258086A patent/IL258086A/en unknown
- 2018-03-16 MX MX2022007315A patent/MX2022007315A/es unknown
- 2018-03-20 CL CL2018000727A patent/CL2018000727A1/es unknown
- 2018-05-17 US US15/982,449 patent/US20180264001A1/en not_active Abandoned
-
2020
- 2020-06-29 IL IL275735A patent/IL275735A/en unknown
-
2021
- 2021-07-01 JP JP2021110240A patent/JP2021167331A/ja active Pending
-
2022
- 2022-06-23 US US17/847,685 patent/US20220323458A1/en not_active Abandoned
- 2022-07-18 AU AU2022206695A patent/AU2022206695A1/en not_active Abandoned
-
2024
- 2024-04-01 US US18/623,327 patent/US20240238307A1/en not_active Abandoned
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