MX2022007315A - Formulaciones de olanzapina de liberacion sostenida. - Google Patents
Formulaciones de olanzapina de liberacion sostenida.Info
- Publication number
- MX2022007315A MX2022007315A MX2022007315A MX2022007315A MX2022007315A MX 2022007315 A MX2022007315 A MX 2022007315A MX 2022007315 A MX2022007315 A MX 2022007315A MX 2022007315 A MX2022007315 A MX 2022007315A MX 2022007315 A MX2022007315 A MX 2022007315A
- Authority
- MX
- Mexico
- Prior art keywords
- sustained release
- olanzapine formulations
- release olanzapine
- olanzapine
- methods
- Prior art date
Links
- KVWDHTXUZHCGIO-UHFFFAOYSA-N olanzapine Chemical compound C1CN(C)CCN1C1=NC2=CC=CC=C2NC2=C1C=C(C)S2 KVWDHTXUZHCGIO-UHFFFAOYSA-N 0.000 title abstract 3
- 229960005017 olanzapine Drugs 0.000 title abstract 3
- 238000013268 sustained release Methods 0.000 title abstract 2
- 239000012730 sustained-release form Substances 0.000 title abstract 2
- 238000009472 formulation Methods 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 238000000034 method Methods 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 208000020925 Bipolar disease Diseases 0.000 abstract 1
- 239000002552 dosage form Substances 0.000 abstract 1
- 201000000980 schizophrenia Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0021—Intradermal administration, e.g. through microneedle arrays, needleless injectors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Inorganic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Biological Depolymerization Polymers (AREA)
Abstract
La presente invención está dirigida a métodos para tratar la esquizofrenia o el trastorno bipolar, administrando por vía subcutánea una forma de dosificación de liberación sostenida de olanzapina, o una sal farmacéuticamente aceptable de la misma. También se describen los métodos para administrar subcutáneamente olanzapina, o una sal farmacéuticamente aceptable de la misma.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201562221290P | 2015-09-21 | 2015-09-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2022007315A true MX2022007315A (es) | 2022-07-13 |
Family
ID=57047342
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2018003380A MX2018003380A (es) | 2015-09-21 | 2016-09-21 | Formulaciones de olanzapina de liberacion sostenida. |
MX2022007315A MX2022007315A (es) | 2015-09-21 | 2018-03-16 | Formulaciones de olanzapina de liberacion sostenida. |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2018003380A MX2018003380A (es) | 2015-09-21 | 2016-09-21 | Formulaciones de olanzapina de liberacion sostenida. |
Country Status (22)
Country | Link |
---|---|
US (4) | US20170079985A1 (es) |
EP (2) | EP3352735B1 (es) |
JP (2) | JP2018527397A (es) |
KR (1) | KR20180054627A (es) |
CN (2) | CN108289834A (es) |
AR (1) | AR106085A1 (es) |
AU (2) | AU2016328958B2 (es) |
CA (1) | CA2998504C (es) |
CL (1) | CL2018000727A1 (es) |
DK (1) | DK3352735T3 (es) |
EA (1) | EA201890788A1 (es) |
ES (1) | ES2960753T3 (es) |
FI (1) | FI3352735T3 (es) |
HK (1) | HK1255946A1 (es) |
HU (1) | HUE063850T2 (es) |
IL (3) | IL295161A (es) |
MX (2) | MX2018003380A (es) |
NZ (1) | NZ740665A (es) |
PL (1) | PL3352735T3 (es) |
PT (1) | PT3352735T (es) |
TW (1) | TWI798161B (es) |
WO (1) | WO2017053346A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA3057438A1 (en) | 2017-03-20 | 2018-09-27 | Teva Pharmaceuticals International Gmbh | Sustained release olanzapine formulaitons |
EP3735223A4 (en) | 2018-01-05 | 2021-10-13 | Impel Neuropharma Inc. | INTRANASAL ADMINISTRATION OF OLANZAPINE BY A PRECISION OLFACTORY DEVICE |
CN112587505A (zh) * | 2020-10-16 | 2021-04-02 | 长春斯菲尔生物科技有限公司 | 一种奥氮平双羟萘酸盐缓释微粒制剂及其制备方法 |
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AU752552C (en) * | 1997-09-30 | 2003-09-11 | Eli Lilly And Company | 2-methyl-thieno-benzodiazepine formulation |
US6495164B1 (en) | 2000-05-25 | 2002-12-17 | Alkermes Controlled Therapeutics, Inc. I | Preparation of injectable suspensions having improved injectability |
US7731947B2 (en) | 2003-11-17 | 2010-06-08 | Intarcia Therapeutics, Inc. | Composition and dosage form comprising an interferon particle formulation and suspending vehicle |
CN1863557B (zh) | 2003-06-26 | 2010-06-16 | 普西维达公司 | 原位胶凝的药物递送系统 |
KR101242486B1 (ko) | 2004-01-12 | 2013-03-13 | 더 트러스티스 오브 더 유니버시티 오브 펜실베니아 | 장기 전달을 위한 제형 및 그의 이용 방법 |
EP1576952A1 (en) | 2004-03-18 | 2005-09-21 | OctoPlus Technologies B.V. | Hydrogel microspheres with improved release profile |
NL1026261C2 (nl) | 2004-05-25 | 2005-11-28 | Nanomi B V | Sproei inrichting met een nozzleplaat voorzien van structuren ter bevordering van self-breakup, een nozzleplaat, alsmede werkwijzen ter vervaardiging en toepassing van een dergelijke nozzleplaat. |
KR101225257B1 (ko) | 2004-06-04 | 2013-01-22 | 카무러스 에이비 | 유동성 데포 제제 |
JP5324098B2 (ja) * | 2004-11-16 | 2013-10-23 | アルケルメス ファーマ アイルランド リミテッド | 注射可能なナノ粒子のオランザピン製剤 |
JP2009533314A (ja) * | 2005-04-13 | 2009-09-17 | ファイザー・プロダクツ・インク | ナノ粒子を含む貧溶性薬物を持続放出するための注射用デポ製剤および方法 |
MX2007012103A (es) * | 2005-04-13 | 2007-11-20 | Pfizer Prod Inc | Formulaciones deposito inyectables y metodos para proporcionar una liberacion sostenida de composiciones de nanoparticulas. |
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US20070254832A1 (en) * | 2006-02-17 | 2007-11-01 | Pressler Milton L | Methods for the treatment of macular degeneration and related eye conditions |
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MX2009000434A (es) | 2006-07-11 | 2009-01-29 | Qps Llc | Composiciones farmaceuticas para la distribucion de liberacion sostenida de peptidos. |
FI20070174A0 (fi) | 2007-02-28 | 2007-02-28 | Delsitech Oy | Menetelmä silikakoostumusten valmistamiseksi, silikakoostumukset ja niiden käytöt |
KR100805208B1 (ko) | 2007-03-27 | 2008-02-21 | 주식회사 펩트론 | 엑센딘 함유 서방성 제제 조성물, 엑센딘 함유 서방성미립구 및 이의 제조 방법 |
CA2683698C (en) | 2007-04-19 | 2013-09-10 | Hyun Hee Kwak | A biodegradable microsphere composition suitable for the controlled release of glucose controlling peptide and formulation thereof |
MX354603B (es) | 2007-05-25 | 2018-03-13 | Indivior Uk Ltd | Formulaciones de transferencia sostenida de compuestos de risperidona. |
ES2324009B1 (es) | 2007-11-23 | 2010-05-21 | Gp Pharm S.A. | Composicion farmaceutica de liberacion sostenida de somatostatina o un analogo suyo. |
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-
2016
- 2016-09-21 US US15/271,508 patent/US20170079985A1/en not_active Abandoned
- 2016-09-21 IL IL295161A patent/IL295161A/en unknown
- 2016-09-21 CN CN201680066464.XA patent/CN108289834A/zh active Pending
- 2016-09-21 EA EA201890788A patent/EA201890788A1/ru unknown
- 2016-09-21 MX MX2018003380A patent/MX2018003380A/es unknown
- 2016-09-21 EP EP16775424.1A patent/EP3352735B1/en active Active
- 2016-09-21 KR KR1020187007791A patent/KR20180054627A/ko not_active Application Discontinuation
- 2016-09-21 WO PCT/US2016/052757 patent/WO2017053346A1/en active Application Filing
- 2016-09-21 NZ NZ740665A patent/NZ740665A/en unknown
- 2016-09-21 EP EP23193256.7A patent/EP4331570A1/en active Pending
- 2016-09-21 DK DK16775424.1T patent/DK3352735T3/da active
- 2016-09-21 PL PL16775424.1T patent/PL3352735T3/pl unknown
- 2016-09-21 AR ARP160102864A patent/AR106085A1/es unknown
- 2016-09-21 CA CA2998504A patent/CA2998504C/en active Active
- 2016-09-21 FI FIEP16775424.1T patent/FI3352735T3/fi active
- 2016-09-21 HU HUE16775424A patent/HUE063850T2/hu unknown
- 2016-09-21 TW TW105130439A patent/TWI798161B/zh active
- 2016-09-21 CN CN202310947482.0A patent/CN116942677A/zh active Pending
- 2016-09-21 AU AU2016328958A patent/AU2016328958B2/en active Active
- 2016-09-21 ES ES16775424T patent/ES2960753T3/es active Active
- 2016-09-21 JP JP2018515050A patent/JP2018527397A/ja active Pending
- 2016-09-21 PT PT167754241T patent/PT3352735T/pt unknown
-
2018
- 2018-03-13 IL IL258086A patent/IL258086A/en unknown
- 2018-03-16 MX MX2022007315A patent/MX2022007315A/es unknown
- 2018-03-20 CL CL2018000727A patent/CL2018000727A1/es unknown
- 2018-05-17 US US15/982,449 patent/US20180264001A1/en not_active Abandoned
- 2018-11-23 HK HK18115019.5A patent/HK1255946A1/zh unknown
-
2020
- 2020-06-29 IL IL275735A patent/IL275735A/en unknown
-
2021
- 2021-07-01 JP JP2021110240A patent/JP2021167331A/ja active Pending
-
2022
- 2022-06-23 US US17/847,685 patent/US20220323458A1/en not_active Abandoned
- 2022-07-18 AU AU2022206695A patent/AU2022206695A1/en not_active Abandoned
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2024
- 2024-04-01 US US18/623,327 patent/US20240238307A1/en active Pending
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