JP2018514523A5 - - Google Patents
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- Publication number
- JP2018514523A5 JP2018514523A5 JP2017553915A JP2017553915A JP2018514523A5 JP 2018514523 A5 JP2018514523 A5 JP 2018514523A5 JP 2017553915 A JP2017553915 A JP 2017553915A JP 2017553915 A JP2017553915 A JP 2017553915A JP 2018514523 A5 JP2018514523 A5 JP 2018514523A5
- Authority
- JP
- Japan
- Prior art keywords
- tablet
- ribocyclic
- rib
- ribocyclib
- succinate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- KDYFGRWQOYBRFD-UHFFFAOYSA-L succinate(2-) Chemical compound [O-]C(=O)CCC([O-])=O KDYFGRWQOYBRFD-UHFFFAOYSA-L 0.000 claims 7
- 150000003839 salts Chemical class 0.000 claims 6
- 239000012156 elution solvent Substances 0.000 claims 4
- 239000011248 coating agent Substances 0.000 claims 2
- 238000000576 coating method Methods 0.000 claims 2
- 239000012458 free base Substances 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562148240P | 2015-04-16 | 2015-04-16 | |
| US62/148,240 | 2015-04-16 | ||
| PCT/IB2016/052136 WO2016166703A1 (en) | 2015-04-16 | 2016-04-14 | Ribociclib tablet |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2018514523A JP2018514523A (ja) | 2018-06-07 |
| JP2018514523A5 true JP2018514523A5 (enExample) | 2019-05-23 |
Family
ID=55806565
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017553915A Pending JP2018514523A (ja) | 2015-04-16 | 2016-04-14 | リボシクリブ錠剤 |
Country Status (29)
| Country | Link |
|---|---|
| US (6) | US10799506B2 (enExample) |
| EP (3) | EP4620458A3 (enExample) |
| JP (1) | JP2018514523A (enExample) |
| KR (2) | KR102750931B1 (enExample) |
| CN (2) | CN115554257A (enExample) |
| AR (1) | AR104257A1 (enExample) |
| AU (5) | AU2016248017A1 (enExample) |
| BR (1) | BR112017021283A2 (enExample) |
| CA (1) | CA2982425C (enExample) |
| CL (1) | CL2017002593A1 (enExample) |
| CO (1) | CO2017010510A2 (enExample) |
| DK (1) | DK3283058T3 (enExample) |
| EA (1) | EA201792290A1 (enExample) |
| EC (1) | ECSP17075052A (enExample) |
| ES (1) | ES2938261T3 (enExample) |
| FI (1) | FI3283058T3 (enExample) |
| HR (1) | HRP20230053T1 (enExample) |
| HU (1) | HUE061213T2 (enExample) |
| IL (1) | IL254818A0 (enExample) |
| MX (1) | MX2017013350A (enExample) |
| PE (1) | PE20180035A1 (enExample) |
| PH (1) | PH12017501820A1 (enExample) |
| PL (1) | PL3283058T3 (enExample) |
| PT (1) | PT3283058T (enExample) |
| SG (1) | SG11201708084PA (enExample) |
| SI (1) | SI3283058T1 (enExample) |
| TN (1) | TN2017000422A1 (enExample) |
| TW (1) | TW201642864A (enExample) |
| WO (1) | WO2016166703A1 (enExample) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018514523A (ja) * | 2015-04-16 | 2018-06-07 | ノバルティス アーゲー | リボシクリブ錠剤 |
| CA3048036A1 (en) | 2018-07-02 | 2020-01-02 | Apotex Inc | Novel crystalline form of ribociclib succinate |
| EP4021450B1 (en) | 2019-08-26 | 2025-11-05 | Arvinas Operations, Inc. | Methods of treating breast cancer with tetrahydronaphthalene derivatives as estrogen receptor degraders |
| IL293940A (en) | 2019-12-16 | 2022-08-01 | Lunella Biotech Inc | Selective cancer drugs cdk4/6 inhibitors |
| CA3164619A1 (en) | 2019-12-16 | 2021-06-24 | Lunella Biotech, Inc. | Selective cdk4/6 inhibitor cancer therapeutics |
| US20230310327A1 (en) * | 2020-08-03 | 2023-10-05 | Natco Pharma Limited | Pharmaceutical compositions comprising ribociclib |
| KR20230079187A (ko) * | 2020-09-29 | 2023-06-05 | 라보라토리오스 실레인즈, 에스.에이. 드 씨.브이. | 고지혈증 및 심혈관 질환의 치료 및 예방을 위한 스타틴 및 피브레이트의 약학적 병용 |
| WO2022162122A1 (en) | 2021-01-29 | 2022-08-04 | Biotx.Ai Gmbh | Genetically verified netosis inhibitor for use in the treatment of a sars-cov2 infection |
| TWI848533B (zh) | 2022-01-25 | 2024-07-11 | 瑞士商諾華公司 | 瑞博西尼藥物組成物 |
| TWI866427B (zh) | 2022-08-31 | 2024-12-11 | 美商亞文納營運公司 | 雌激素受體降解劑之給藥方案 |
| EP4626890A1 (en) | 2022-12-01 | 2025-10-08 | KRKA, d.d., Novo mesto | Ribociclib salts and formulations thereof |
| AU2024244511A1 (en) | 2023-03-27 | 2025-09-25 | Novartis Ag | Method of treating early breast cancer with ribociclib in combination with an aromatase inhibitor |
| WO2025219830A1 (en) | 2024-04-15 | 2025-10-23 | Novartis Ag | Pharmaceutical compositions of ribociclib |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5428812A (en) * | 1977-08-09 | 1979-03-03 | Yoshitomi Pharmaceut Ind Ltd | Preparation of coated tablet |
| GB9414045D0 (en) | 1994-07-12 | 1994-08-31 | Berwind Pharma Service | Moisture barrier film coating composition, method, and coated form |
| EP0771339B1 (en) * | 1994-07-12 | 2003-10-15 | BPSI Holdings, Inc. | Dry moisture barrier film coating composition, method of coating substrates using the same and pharmaceutical tablets coated therewith |
| US6448323B1 (en) * | 1999-07-09 | 2002-09-10 | Bpsi Holdings, Inc. | Film coatings and film coating compositions based on polyvinyl alcohol |
| ES2522346T3 (es) | 2008-08-22 | 2014-11-14 | Novartis Ag | Compuestos de pirrolopirimidina como inhibidores de CDK |
| US8343533B2 (en) * | 2009-09-24 | 2013-01-01 | Mcneil-Ppc, Inc. | Manufacture of lozenge product with radiofrequency |
| US20120115878A1 (en) | 2010-11-10 | 2012-05-10 | John Vincent Calienni | Salt(s) of 7-cyclopentyl-2-(5-piperazin-1-yl-pyridin-2-ylamino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid dimethylamide and processes of making thereof |
| EA025033B1 (ru) * | 2011-02-11 | 2016-11-30 | Уиста Лэборэтэриз Лтд. | Диаминиевые соли фенотиазина и их применение |
| IN2015DN01046A (enExample) * | 2012-07-13 | 2015-06-26 | Gtx Inc | |
| EP3251673A1 (en) * | 2012-12-13 | 2017-12-06 | IP Gesellschaft für Management mbH | Combination therapy comprising a cdk4/6 inhibitor and a pi3k inhibitor for use in the treatment of cancer |
| WO2014097125A1 (en) * | 2012-12-20 | 2014-06-26 | Novartis Ag | Pharmaceutical combination comprising binimetinib |
| PT2976106T (pt) * | 2013-03-21 | 2021-05-26 | Array Biopharma Inc | Terapia de combinação que compreende um inibidor de b-raf e um segundo inibidor |
| EP2810644A1 (en) * | 2013-06-06 | 2014-12-10 | Ferrer Internacional, S.A. | Oral formulation for the treatment of cardiovascular diseases |
| JP2018514523A (ja) * | 2015-04-16 | 2018-06-07 | ノバルティス アーゲー | リボシクリブ錠剤 |
| CN109953966A (zh) * | 2017-12-26 | 2019-07-02 | 天津耀辰实业发展有限公司 | 一种含有瑞博西尼的药物组合物及其制备方法 |
| JP7347388B2 (ja) | 2020-09-25 | 2023-09-20 | 信越化学工業株式会社 | 紫外線硬化型有機変性シリコーン組成物および硬化物 |
-
2016
- 2016-04-14 JP JP2017553915A patent/JP2018514523A/ja active Pending
- 2016-04-14 PL PL16718020.7T patent/PL3283058T3/pl unknown
- 2016-04-14 ES ES16718020T patent/ES2938261T3/es active Active
- 2016-04-14 PE PE2017002096A patent/PE20180035A1/es unknown
- 2016-04-14 TN TNP/2017/000422A patent/TN2017000422A1/en unknown
- 2016-04-14 HR HRP20230053TT patent/HRP20230053T1/hr unknown
- 2016-04-14 DK DK16718020.7T patent/DK3283058T3/da active
- 2016-04-14 BR BR112017021283A patent/BR112017021283A2/pt not_active Application Discontinuation
- 2016-04-14 PT PT167180207T patent/PT3283058T/pt unknown
- 2016-04-14 SG SG11201708084PA patent/SG11201708084PA/en unknown
- 2016-04-14 EA EA201792290A patent/EA201792290A1/ru unknown
- 2016-04-14 FI FIEP16718020.7T patent/FI3283058T3/fi active
- 2016-04-14 MX MX2017013350A patent/MX2017013350A/es unknown
- 2016-04-14 KR KR1020177029433A patent/KR102750931B1/ko active Active
- 2016-04-14 EP EP25194967.3A patent/EP4620458A3/en active Pending
- 2016-04-14 CN CN202211237232.XA patent/CN115554257A/zh active Pending
- 2016-04-14 CA CA2982425A patent/CA2982425C/en active Active
- 2016-04-14 SI SI201631661T patent/SI3283058T1/sl unknown
- 2016-04-14 KR KR1020257000051A patent/KR20250009572A/ko active Pending
- 2016-04-14 US US15/564,534 patent/US10799506B2/en active Active
- 2016-04-14 CN CN201680022122.8A patent/CN107530292B/zh active Active
- 2016-04-14 EP EP16718020.7A patent/EP3283058B1/en active Active
- 2016-04-14 AU AU2016248017A patent/AU2016248017A1/en not_active Abandoned
- 2016-04-14 AR ARP160101012A patent/AR104257A1/es unknown
- 2016-04-14 HU HUE16718020A patent/HUE061213T2/hu unknown
- 2016-04-14 WO PCT/IB2016/052136 patent/WO2016166703A1/en not_active Ceased
- 2016-04-14 EP EP22203730.1A patent/EP4197530B1/en active Active
- 2016-04-15 TW TW105111921A patent/TW201642864A/zh unknown
-
2017
- 2017-10-01 IL IL254818A patent/IL254818A0/en unknown
- 2017-10-04 PH PH12017501820A patent/PH12017501820A1/en unknown
- 2017-10-13 CO CONC2017/0010510A patent/CO2017010510A2/es unknown
- 2017-10-13 CL CL2017002593A patent/CL2017002593A1/es unknown
- 2017-11-10 EC ECIEPI201775052A patent/ECSP17075052A/es unknown
-
2019
- 2019-03-20 AU AU2019201929A patent/AU2019201929B2/en active Active
-
2020
- 2020-08-26 US US17/003,771 patent/US20200390771A1/en not_active Abandoned
- 2020-10-06 AU AU2020250190A patent/AU2020250190A1/en not_active Abandoned
-
2022
- 2022-06-08 US US17/805,956 patent/US12064434B2/en active Active
- 2022-08-08 AU AU2022215155A patent/AU2022215155B2/en active Active
-
2024
- 2024-02-27 US US18/588,259 patent/US20250090531A1/en active Pending
- 2024-10-31 AU AU2024227794A patent/AU2024227794A1/en active Pending
- 2024-12-11 US US18/977,228 patent/US12419894B2/en active Active
- 2024-12-11 US US18/977,210 patent/US20250134893A1/en active Pending
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