JP2018514523A5 - - Google Patents
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- Publication number
- JP2018514523A5 JP2018514523A5 JP2017553915A JP2017553915A JP2018514523A5 JP 2018514523 A5 JP2018514523 A5 JP 2018514523A5 JP 2017553915 A JP2017553915 A JP 2017553915A JP 2017553915 A JP2017553915 A JP 2017553915A JP 2018514523 A5 JP2018514523 A5 JP 2018514523A5
- Authority
- JP
- Japan
- Prior art keywords
- tablet
- ribocyclic
- rib
- ribocyclib
- succinate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- KDYFGRWQOYBRFD-UHFFFAOYSA-L succinate(2-) Chemical compound [O-]C(=O)CCC([O-])=O KDYFGRWQOYBRFD-UHFFFAOYSA-L 0.000 claims 7
- 150000003839 salts Chemical class 0.000 claims 6
- 239000012156 elution solvent Substances 0.000 claims 4
- 239000011248 coating agent Substances 0.000 claims 2
- 238000000576 coating method Methods 0.000 claims 2
- 239000012458 free base Substances 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562148240P | 2015-04-16 | 2015-04-16 | |
| US62/148,240 | 2015-04-16 | ||
| PCT/IB2016/052136 WO2016166703A1 (en) | 2015-04-16 | 2016-04-14 | Ribociclib tablet |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2018514523A JP2018514523A (ja) | 2018-06-07 |
| JP2018514523A5 true JP2018514523A5 (enExample) | 2019-05-23 |
Family
ID=55806565
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017553915A Pending JP2018514523A (ja) | 2015-04-16 | 2016-04-14 | リボシクリブ錠剤 |
Country Status (29)
| Country | Link |
|---|---|
| US (6) | US10799506B2 (enExample) |
| EP (3) | EP4197530B1 (enExample) |
| JP (1) | JP2018514523A (enExample) |
| KR (2) | KR102750931B1 (enExample) |
| CN (2) | CN107530292B (enExample) |
| AR (1) | AR104257A1 (enExample) |
| AU (5) | AU2016248017A1 (enExample) |
| BR (1) | BR112017021283A2 (enExample) |
| CA (1) | CA2982425C (enExample) |
| CL (1) | CL2017002593A1 (enExample) |
| CO (1) | CO2017010510A2 (enExample) |
| DK (1) | DK3283058T3 (enExample) |
| EA (1) | EA201792290A1 (enExample) |
| EC (1) | ECSP17075052A (enExample) |
| ES (1) | ES2938261T3 (enExample) |
| FI (1) | FI3283058T3 (enExample) |
| HR (1) | HRP20230053T1 (enExample) |
| HU (1) | HUE061213T2 (enExample) |
| IL (1) | IL254818A0 (enExample) |
| MX (1) | MX2017013350A (enExample) |
| PE (1) | PE20180035A1 (enExample) |
| PH (1) | PH12017501820A1 (enExample) |
| PL (1) | PL3283058T3 (enExample) |
| PT (1) | PT3283058T (enExample) |
| SG (1) | SG11201708084PA (enExample) |
| SI (1) | SI3283058T1 (enExample) |
| TN (1) | TN2017000422A1 (enExample) |
| TW (1) | TW201642864A (enExample) |
| WO (1) | WO2016166703A1 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102750931B1 (ko) * | 2015-04-16 | 2025-01-09 | 노파르티스 아게 | 리보시클립 정제 |
| CA3048036A1 (en) | 2018-07-02 | 2020-01-02 | Apotex Inc | Novel crystalline form of ribociclib succinate |
| CN118986983A (zh) | 2019-08-26 | 2024-11-22 | 阿尔维纳斯运营股份有限公司 | 用四氢萘衍生物作为雌激素受体降解剂的治疗乳腺癌的方法 |
| EP4077331A4 (en) | 2019-12-16 | 2023-12-27 | Lunella Biotech, Inc. | SELECTIVE CDK4/6 INHIBITOR CANCER THERAPEUTICS |
| BR112022011851A2 (pt) | 2019-12-16 | 2022-09-06 | Lunella Biotech Inc | Terapêutica de câncer inibidor de cdk4/6 seletivo |
| CA3187241A1 (en) * | 2020-08-03 | 2022-02-10 | Krishna Murthy Bhavanasi | Pharmaceutical compositions comprising ribociclib |
| CA3191478A1 (en) * | 2020-09-29 | 2022-04-07 | Paola Yazmin Ollervides Rubio | Pharmaceutical combinations of statins and fibrates for the treatment and prevention of hyperlipidemias and cardiovascular disease |
| WO2022162122A1 (en) | 2021-01-29 | 2022-08-04 | Biotx.Ai Gmbh | Genetically verified netosis inhibitor for use in the treatment of a sars-cov2 infection |
| CN117396208A (zh) | 2021-07-16 | 2024-01-12 | 达纳－法伯癌症研究所公司 | 细胞周期蛋白依赖性激酶4/6(cdk4/6)和ikzf2(helios)的小分子降解剂及其使用方法 |
| TWI848533B (zh) | 2022-01-25 | 2024-07-11 | 瑞士商諾華公司 | 瑞博西尼藥物組成物 |
| CN120112291A (zh) | 2022-08-31 | 2025-06-06 | 阿尔维纳斯运营股份有限公司 | 雌激素受体降解剂的给药方案 |
| EP4626890A1 (en) | 2022-12-01 | 2025-10-08 | KRKA, d.d., Novo mesto | Ribociclib salts and formulations thereof |
| TW202440113A (zh) | 2023-03-27 | 2024-10-16 | 瑞士商諾華公司 | 治療早期乳癌之方法 |
| WO2025219830A1 (en) | 2024-04-15 | 2025-10-23 | Novartis Ag | Pharmaceutical compositions of ribociclib |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5428812A (en) * | 1977-08-09 | 1979-03-03 | Yoshitomi Pharmaceut Ind Ltd | Preparation of coated tablet |
| JP3672314B2 (ja) * | 1994-07-12 | 2005-07-20 | バーウィンド・ファーマスーティカル・サーヴィスィーズ・インコーポレーテッド | 防湿性フィルム被覆材組成物、方法および被覆成形物 |
| GB9414045D0 (en) | 1994-07-12 | 1994-08-31 | Berwind Pharma Service | Moisture barrier film coating composition, method, and coated form |
| US6448323B1 (en) * | 1999-07-09 | 2002-09-10 | Bpsi Holdings, Inc. | Film coatings and film coating compositions based on polyvinyl alcohol |
| SI2331547T1 (sl) | 2008-08-22 | 2014-11-28 | Novartis Ag | Pirolopirimidinske spojine kot CDK inhibitorji |
| US8807979B2 (en) * | 2009-09-24 | 2014-08-19 | Mcneil-Ppc, Inc. | Machine for the manufacture of dosage forms utilizing radiofrequency energy |
| AR083797A1 (es) * | 2010-11-10 | 2013-03-20 | Novartis Ag | Succinato de dimetil-amida del acido 7-ciclopentil-2-(5-piperazin-1-il-piridin-2-il-amino)-7h-pirrolo-[2,3-d]pirimidin-6-carboxilico, proceso para prepararla, intermediarios de dicha sintesis y proceso de preparacion de los mismos |
| SI2673266T1 (sl) * | 2011-02-11 | 2016-11-30 | Wista Laboratories Ltd. | Fenotiazin diaminijeve soli in njihova uporaba |
| WO2014011220A2 (en) * | 2012-07-13 | 2014-01-16 | Gtx, Inc. | A method of treating androgen receptor (ar)-positive breast cancers with selective androgen receptor modulator (sarms) |
| EP3251673A1 (en) * | 2012-12-13 | 2017-12-06 | IP Gesellschaft für Management mbH | Combination therapy comprising a cdk4/6 inhibitor and a pi3k inhibitor for use in the treatment of cancer |
| WO2014097125A1 (en) * | 2012-12-20 | 2014-06-26 | Novartis Ag | Pharmaceutical combination comprising binimetinib |
| MY181085A (en) * | 2013-03-21 | 2020-12-17 | Novartis Ag | Combination therapy |
| EP2810644A1 (en) * | 2013-06-06 | 2014-12-10 | Ferrer Internacional, S.A. | Oral formulation for the treatment of cardiovascular diseases |
| KR102750931B1 (ko) * | 2015-04-16 | 2025-01-09 | 노파르티스 아게 | 리보시클립 정제 |
| CN109953966A (zh) * | 2017-12-26 | 2019-07-02 | 天津耀辰实业发展有限公司 | 一种含有瑞博西尼的药物组合物及其制备方法 |
| JP7347388B2 (ja) | 2020-09-25 | 2023-09-20 | 信越化学工業株式会社 | 紫外線硬化型有機変性シリコーン組成物および硬化物 |
-
2016
- 2016-04-14 KR KR1020177029433A patent/KR102750931B1/ko active Active
- 2016-04-14 DK DK16718020.7T patent/DK3283058T3/da active
- 2016-04-14 EP EP22203730.1A patent/EP4197530B1/en active Active
- 2016-04-14 SI SI201631661T patent/SI3283058T1/sl unknown
- 2016-04-14 KR KR1020257000051A patent/KR20250009572A/ko active Pending
- 2016-04-14 AU AU2016248017A patent/AU2016248017A1/en not_active Abandoned
- 2016-04-14 HR HRP20230053TT patent/HRP20230053T1/hr unknown
- 2016-04-14 HU HUE16718020A patent/HUE061213T2/hu unknown
- 2016-04-14 MX MX2017013350A patent/MX2017013350A/es unknown
- 2016-04-14 CN CN201680022122.8A patent/CN107530292B/zh active Active
- 2016-04-14 AR ARP160101012A patent/AR104257A1/es unknown
- 2016-04-14 CN CN202211237232.XA patent/CN115554257A/zh active Pending
- 2016-04-14 PL PL16718020.7T patent/PL3283058T3/pl unknown
- 2016-04-14 TN TNP/2017/000422A patent/TN2017000422A1/en unknown
- 2016-04-14 FI FIEP16718020.7T patent/FI3283058T3/fi active
- 2016-04-14 EP EP25194967.3A patent/EP4620458A3/en active Pending
- 2016-04-14 PT PT167180207T patent/PT3283058T/pt unknown
- 2016-04-14 CA CA2982425A patent/CA2982425C/en active Active
- 2016-04-14 EA EA201792290A patent/EA201792290A1/ru unknown
- 2016-04-14 EP EP16718020.7A patent/EP3283058B1/en active Active
- 2016-04-14 PE PE2017002096A patent/PE20180035A1/es unknown
- 2016-04-14 US US15/564,534 patent/US10799506B2/en active Active
- 2016-04-14 JP JP2017553915A patent/JP2018514523A/ja active Pending
- 2016-04-14 SG SG11201708084PA patent/SG11201708084PA/en unknown
- 2016-04-14 ES ES16718020T patent/ES2938261T3/es active Active
- 2016-04-14 BR BR112017021283A patent/BR112017021283A2/pt not_active Application Discontinuation
- 2016-04-14 WO PCT/IB2016/052136 patent/WO2016166703A1/en not_active Ceased
- 2016-04-15 TW TW105111921A patent/TW201642864A/zh unknown
-
2017
- 2017-10-01 IL IL254818A patent/IL254818A0/en unknown
- 2017-10-04 PH PH12017501820A patent/PH12017501820A1/en unknown
- 2017-10-13 CL CL2017002593A patent/CL2017002593A1/es unknown
- 2017-10-13 CO CONC2017/0010510A patent/CO2017010510A2/es unknown
- 2017-11-10 EC ECIEPI201775052A patent/ECSP17075052A/es unknown
-
2019
- 2019-03-20 AU AU2019201929A patent/AU2019201929B2/en active Active
-
2020
- 2020-08-26 US US17/003,771 patent/US20200390771A1/en not_active Abandoned
- 2020-10-06 AU AU2020250190A patent/AU2020250190A1/en not_active Abandoned
-
2022
- 2022-06-08 US US17/805,956 patent/US12064434B2/en active Active
- 2022-08-08 AU AU2022215155A patent/AU2022215155B2/en active Active
-
2024
- 2024-02-27 US US18/588,259 patent/US20250090531A1/en active Pending
- 2024-10-31 AU AU2024227794A patent/AU2024227794A1/en active Pending
- 2024-12-11 US US18/977,210 patent/US20250134893A1/en active Pending
- 2024-12-11 US US18/977,228 patent/US12419894B2/en active Active
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