JP2018503647A5 - - Google Patents
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- Publication number
- JP2018503647A5 JP2018503647A5 JP2017539234A JP2017539234A JP2018503647A5 JP 2018503647 A5 JP2018503647 A5 JP 2018503647A5 JP 2017539234 A JP2017539234 A JP 2017539234A JP 2017539234 A JP2017539234 A JP 2017539234A JP 2018503647 A5 JP2018503647 A5 JP 2018503647A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- compound
- group
- substituted
- independently selected
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562109890P | 2015-01-30 | 2015-01-30 | |
| US62/109,890 | 2015-01-30 | ||
| PCT/US2016/015251 WO2016123275A1 (en) | 2015-01-30 | 2016-01-28 | Aldosterone synthase inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018503647A JP2018503647A (ja) | 2018-02-08 |
| JP2018503647A5 true JP2018503647A5 (enExample) | 2019-03-07 |
| JP6615896B2 JP6615896B2 (ja) | 2019-12-04 |
Family
ID=55361967
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017539234A Active JP6615896B2 (ja) | 2015-01-30 | 2016-01-28 | アルドステロン合成酵素阻害剤 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US10131642B1 (enExample) |
| EP (1) | EP3250569B1 (enExample) |
| JP (1) | JP6615896B2 (enExample) |
| WO (1) | WO2016123275A1 (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP7225253B2 (ja) * | 2018-02-02 | 2023-02-20 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | グレリンｏ－アシルトランスフェラーゼ（ｇｏａｔ）阻害剤として使用するためのピラゾール置換及びインダゾール置換オキサジアゾロピリジン誘導体 |
| CA3087925A1 (en) | 2018-02-02 | 2019-08-08 | Boehringer Ingelheim International Gmbh | Triazolopyrimidine derivatives for use as ghrelin o-acyl transferase (goat) inhibitors |
| MX2020008053A (es) | 2018-02-02 | 2020-09-07 | Boehringer Ingelheim Int | Derivados de oxadiazolopiridina sustituidos con bencilo, (piridin-3-il)metilo o (piridin-4-il)metilo como inhibidores de ghrelin o-aciltransferasa (goat). |
| CN111655699B (zh) * | 2018-02-02 | 2023-07-14 | 勃林格殷格翰国际有限公司 | 用作饥饿素o-酰基转移酶(goat)抑制剂的杂环基取代的噁二唑并吡啶衍生物 |
| WO2021233884A1 (en) | 2020-05-22 | 2021-11-25 | Boehringer Ingelheim International Gmbh | Continuous process for manufacturing alkyl 7-amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridine-carboxylate |
| EP4153599B1 (en) | 2020-05-22 | 2024-03-13 | Boehringer Ingelheim International GmbH | Process for manufacturing alkyl 7-amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridine-carboxylate |
| WO2026093586A1 (en) | 2024-11-04 | 2026-05-07 | AstraZeneca Ireland Limited | Combination of a aldosterone synthase inhibitor (asi) and a sodium-glucose co-transporter 2 inhibitor (sglt2i) for use in methods of reducing the risk of cardiovascular and heart failure events in a subject |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4544864B2 (ja) * | 2002-03-08 | 2010-09-15 | 独立行政法人科学技術振興機構 | イソキサゾール誘導体及びその製造方法 |
| DE102004035322A1 (de) * | 2004-07-21 | 2006-02-16 | Universität des Saarlandes | Selektive Hemmstoffe humaner Corticoidsynthasen |
| BRPI0709678A2 (pt) * | 2006-03-29 | 2011-07-19 | Novartis Ag | compostos orgánicos |
| WO2007139992A2 (en) * | 2006-05-26 | 2007-12-06 | Novartis Ag | ALDOSTERONE SYNTHASE AND/OR 11β-HYDROXYLASE INHIBITORS |
| ITMI20062102A1 (it) * | 2006-11-02 | 2008-05-03 | Abiogen Pharma Spa | Nuovui sali di 3-benzil-2-metil-2,3,3a,4,5,6,7,7a-ottaidrobenzo-d-isossazol-4-one |
| AU2008345225A1 (en) * | 2007-12-21 | 2009-07-09 | University Of Rochester | Method for altering the lifespan of eukaryotic organisms |
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2016
- 2016-01-28 WO PCT/US2016/015251 patent/WO2016123275A1/en not_active Ceased
- 2016-01-28 US US15/545,331 patent/US10131642B1/en active Active
- 2016-01-28 EP EP16704980.8A patent/EP3250569B1/en active Active
- 2016-01-28 JP JP2017539234A patent/JP6615896B2/ja active Active