JP2018203733A5 - - Google Patents

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Publication number
JP2018203733A5
JP2018203733A5 JP2018103970A JP2018103970A JP2018203733A5 JP 2018203733 A5 JP2018203733 A5 JP 2018203733A5 JP 2018103970 A JP2018103970 A JP 2018103970A JP 2018103970 A JP2018103970 A JP 2018103970A JP 2018203733 A5 JP2018203733 A5 JP 2018203733A5
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JP
Japan
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group
formula
optionally substituted
compound represented
alkoxy
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JP2018103970A
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English (en)
Japanese (ja)
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JP2018203733A (ja
JP7102233B2 (ja
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Priority claimed from PCT/IB2018/053822 external-priority patent/WO2018220533A2/ja
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Priority to JP2022078462A priority Critical patent/JP7420865B2/ja
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Publication of JP7102233B2 publication Critical patent/JP7102233B2/ja
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JP2018103970A 2017-05-30 2018-05-30 光学活性化合物の製造法 Active JP7102233B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2022078462A JP7420865B2 (ja) 2017-05-30 2022-05-11 光学活性化合物の製造法

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2017106280 2017-05-30
JP2017106280 2017-05-30
PCT/IB2018/053822 WO2018220533A2 (ja) 2017-05-30 2018-05-29 光学活性化合物の製造法
WOPCT/IB2018/053822 2018-05-29

Related Child Applications (1)

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JP2022078462A Division JP7420865B2 (ja) 2017-05-30 2022-05-11 光学活性化合物の製造法

Publications (3)

Publication Number Publication Date
JP2018203733A JP2018203733A (ja) 2018-12-27
JP2018203733A5 true JP2018203733A5 (https=) 2021-07-26
JP7102233B2 JP7102233B2 (ja) 2022-07-19

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ID=64454503

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JP2018103970A Active JP7102233B2 (ja) 2017-05-30 2018-05-30 光学活性化合物の製造法
JP2022078462A Active JP7420865B2 (ja) 2017-05-30 2022-05-11 光学活性化合物の製造法

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JP2022078462A Active JP7420865B2 (ja) 2017-05-30 2022-05-11 光学活性化合物の製造法

Country Status (12)

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US (2) US10988469B2 (https=)
EP (2) EP3632441B1 (https=)
JP (2) JP7102233B2 (https=)
KR (1) KR102754527B1 (https=)
CN (2) CN111032047B (https=)
AU (1) AU2018276192B2 (https=)
CA (1) CA3065683A1 (https=)
EA (1) EA039880B1 (https=)
ES (1) ES2986461T3 (https=)
IL (1) IL270983B (https=)
MX (1) MX391164B (https=)
WO (1) WO2018220533A2 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX391164B (es) 2017-05-30 2025-03-21 Dot Therapeutics 1 Inc Metodo para producir compuesto opticamente activo
CN113557227A (zh) * 2019-03-27 2021-10-26 协和医药化工股份有限公司 前列腺素的制造方法
AU2021376286A1 (en) * 2020-11-06 2023-06-22 Dana-Farber Cancer Institute, Inc. Raf inhibitor for treating low grade glioma
CN114685564B (zh) * 2020-12-27 2023-09-22 西北大学 新型亚磷酰胺配体及其合成方法和应用
EP4377296A1 (en) 2021-07-26 2024-06-05 Arvinas Operations, Inc. Methods of manufacturing a bifunctional compound
CN117567388B (zh) * 2023-11-14 2024-04-16 济南悟通生物科技有限公司 一种2-乙酰基-5-噻唑甲酸的合成方法
WO2026028053A2 (en) 2024-07-27 2026-02-05 Assia Chemical Industries Ltd. Process for the preparation of tovorafenib
CN119241530B (zh) * 2024-09-20 2026-04-10 武汉九州钰民医药科技有限公司 一种Tovorafenib的药物合成工艺
CN119241529B (zh) * 2024-09-20 2026-04-10 武汉九州钰民医药科技有限公司 一种Tovorafenib的制备方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6764842B2 (en) * 2001-03-28 2004-07-20 Merck & Co., Inc. Enantioselective bioreduction for the preparation of integrin receptor antagonist intermediates
TW200303304A (en) * 2002-02-18 2003-09-01 Astrazeneca Ab Chemical compounds
US7754889B2 (en) * 2004-03-29 2010-07-13 Takasago International Corporation Optically active transition metal-diamine compound and process for producing optically active alcohol with the same
TWI345568B (en) * 2004-04-02 2011-07-21 Mitsubishi Tanabe Pharma Corp Tetrahydronaphthyridine derivatives and a process for preparing the same
AR067354A1 (es) * 2007-06-29 2009-10-07 Sunesis Pharmaceuticals Inc Compuestos utiles como inhibidores de la raf quinasa
EP2167497A2 (en) * 2007-06-29 2010-03-31 Sunesis Pharmaceuticals, Inc. Heterocyclic compounds useful as raf kinase inhibitors
MX351657B (es) * 2012-03-14 2017-10-23 Merck Sharp & Dohme Sales de alcaloide de cinchona bis-cuaternarias como catalizadores de transferencia de fase asimétrica.
CN107880075A (zh) 2012-03-28 2018-04-06 武田药品工业株式会社 铑催化剂和制备胺化合物的方法
TWI602803B (zh) * 2013-03-29 2017-10-21 第一三共股份有限公司 光學活性二胺衍生物之製造方法
WO2015178846A1 (en) * 2014-05-20 2015-11-26 Sp Process Development Ab Process for the preparation of chiral amines from prochiral ketones
JP6638363B2 (ja) 2015-12-11 2020-01-29 株式会社大林組 掘削装置および杭孔の拡径方法
CN105524111B (zh) * 2016-01-25 2017-10-27 西北农林科技大学 手性亚磷酰胺单齿配体及其合成方法与应用
MX391164B (es) 2017-05-30 2025-03-21 Dot Therapeutics 1 Inc Metodo para producir compuesto opticamente activo

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