JP2017537882A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2017537882A5 JP2017537882A5 JP2017520319A JP2017520319A JP2017537882A5 JP 2017537882 A5 JP2017537882 A5 JP 2017537882A5 JP 2017520319 A JP2017520319 A JP 2017520319A JP 2017520319 A JP2017520319 A JP 2017520319A JP 2017537882 A5 JP2017537882 A5 JP 2017537882A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- haloalkyl
- formula
- group
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 32
- 150000001875 compounds Chemical class 0.000 claims description 29
- 125000000217 alkyl group Chemical group 0.000 claims description 24
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 22
- 229910052736 halogen Inorganic materials 0.000 claims description 22
- 150000002367 halogens Chemical group 0.000 claims description 22
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 14
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 14
- 125000004122 cyclic group Chemical group 0.000 claims description 14
- 125000001424 substituent group Chemical group 0.000 claims description 13
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 12
- 229910052739 hydrogen Inorganic materials 0.000 claims description 12
- 239000001257 hydrogen Substances 0.000 claims description 12
- 238000000034 method Methods 0.000 claims description 11
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 10
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims description 10
- -1 C 1 -C 4 alkyl Chemical group 0.000 claims description 9
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 claims description 9
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 8
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 8
- 241000607479 Yersinia pestis Species 0.000 claims description 8
- 125000000623 heterocyclic group Chemical group 0.000 claims description 8
- 229910052717 sulfur Chemical group 0.000 claims description 8
- 229910052760 oxygen Inorganic materials 0.000 claims description 7
- 125000001188 haloalkyl group Chemical group 0.000 claims description 6
- 229910052757 nitrogen Inorganic materials 0.000 claims description 6
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims description 5
- 239000001301 oxygen Chemical group 0.000 claims description 5
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 4
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 4
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 4
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims description 4
- 125000003118 aryl group Chemical group 0.000 claims description 4
- 125000004186 cyclopropylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C1([H])[H] 0.000 claims description 4
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 4
- 125000005842 heteroatom Chemical group 0.000 claims description 4
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims description 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 4
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims description 4
- IJGRMHOSHXDMSA-UHFFFAOYSA-N nitrogen Substances N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims description 4
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- 229920006395 saturated elastomer Polymers 0.000 claims description 4
- 239000011593 sulfur Chemical group 0.000 claims description 4
- 125000004430 oxygen atom Chemical group O* 0.000 claims description 3
- 125000004434 sulfur atom Chemical group 0.000 claims description 3
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- 239000004480 active ingredient Substances 0.000 claims description 2
- 125000002619 bicyclic group Chemical group 0.000 claims description 2
- 229910052799 carbon Inorganic materials 0.000 claims description 2
- 125000004432 carbon atom Chemical group C* 0.000 claims description 2
- 238000002405 diagnostic procedure Methods 0.000 claims description 2
- 125000004439 haloalkylsulfanyl group Chemical group 0.000 claims description 2
- 125000004440 haloalkylsulfinyl group Chemical group 0.000 claims description 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 2
- 239000000463 material Substances 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- 125000002950 monocyclic group Chemical group 0.000 claims description 2
- 125000004433 nitrogen atom Chemical group N* 0.000 claims description 2
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 2
- 238000001356 surgical procedure Methods 0.000 claims description 2
- 238000002560 therapeutic procedure Methods 0.000 claims description 2
- 239000012752 auxiliary agent Substances 0.000 claims 1
- 125000000262 haloalkenyl group Chemical group 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 description 7
- 0 Cc1ccc(*)cc1 Chemical compound Cc1ccc(*)cc1 0.000 description 5
- 125000004414 alkyl thio group Chemical group 0.000 description 5
- 241001465754 Metazoa Species 0.000 description 2
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 description 1
- 125000004644 alkyl sulfinyl group Chemical group 0.000 description 1
- 125000004429 atom Chemical group 0.000 description 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14189186.1 | 2014-10-16 | ||
| EP14189186 | 2014-10-16 | ||
| PCT/EP2015/073856 WO2016059145A1 (en) | 2014-10-16 | 2015-10-15 | Pesticidally active tetracyclic heterocyclic derivatives with sulphur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017537882A JP2017537882A (ja) | 2017-12-21 |
| JP2017537882A5 true JP2017537882A5 (index.php) | 2018-11-22 |
| JP6675390B2 JP6675390B2 (ja) | 2020-04-01 |
Family
ID=51844501
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017520319A Expired - Fee Related JP6675390B2 (ja) | 2014-10-16 | 2015-10-15 | 硫黄含有置換基を有する有害生物防除に活性な四環式複素環誘導体 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US10544148B2 (index.php) |
| EP (1) | EP3207044B1 (index.php) |
| JP (1) | JP6675390B2 (index.php) |
| CN (1) | CN106795167B (index.php) |
| BR (1) | BR112017007510A2 (index.php) |
| ES (1) | ES2690131T3 (index.php) |
| WO (1) | WO2016059145A1 (index.php) |
Families Citing this family (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA121319C2 (uk) * | 2014-11-07 | 2020-05-12 | Сінгента Партісіпейшнс Аг | Пестицидно активні поліциклічні похідні з сірковмісними замісниками |
| CO2018009129A2 (es) | 2016-02-26 | 2018-09-20 | Nihon Nohyaku Co Ltd | Compuesto heterocíclico condensado ligado a heterociclo o su sal, insecticida agrícola y hortícola que comprende el compuesto y método para usar el insecticida |
| KR102477315B1 (ko) | 2016-10-06 | 2022-12-13 | 바이엘 크롭사이언스 악티엔게젤샤프트 | 해충 방제제로서의 2-(헤트)아릴-치환된 융합 비사이클릭 헤테로사이클 유도체 |
| WO2018065288A1 (de) | 2016-10-07 | 2018-04-12 | Bayer Cropscience Aktiengesellschaft | 2-[2-phenyl-1-(sulfonylmethyl)vinyl]-imidazo[4,5-b]pyridin-derivate und verwandte verbindungen als schädlingsbekämpfungsmittel im pflanzenschutz |
| WO2018091389A1 (en) * | 2016-11-17 | 2018-05-24 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| CN117624038A (zh) | 2016-12-01 | 2024-03-01 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
| BR112019012127A2 (pt) | 2016-12-15 | 2019-11-05 | Syngenta Participations Ag | derivados heterocíclicos ativos em termos pesticidas com substituintes contendo enxofre |
| US11083199B2 (en) | 2017-01-10 | 2021-08-10 | Bayer Aktiengesellschaft | Heterocycle derivatives as pesticides |
| AU2018207776B2 (en) | 2017-01-10 | 2021-06-17 | Bayer Aktiengesellschaft | Heterocyclene derivatives as pest control agents |
| WO2018202540A1 (en) | 2017-05-02 | 2018-11-08 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| US11505553B2 (en) | 2017-05-02 | 2022-11-22 | Bayer Aktiengesellschaft | 2-(Het)aryl-substituted fused heterocycle derivatives as pesticides |
| BR112019022837A2 (pt) | 2017-05-02 | 2020-05-26 | Bayer Aktiengesellschaft | Derivados heterocíclicos bicíclicos condensados substituídos por 2-(het)arila como agentes de controle de praga |
| WO2018215304A1 (en) | 2017-05-22 | 2018-11-29 | Syngenta Participations Ag | Tetracyclic pyridazine sulphur containing compounds and their use as pesticides |
| BR112019028233B1 (pt) | 2017-07-05 | 2023-12-05 | Syngenta Participations Ag | Derivados heterocíclicos com substituintes contendo enxofre ativos em termos pesticidas, composição pesticida, método para combater e controlar pragas e método para proteção de material de propagação vegetal |
| WO2019065568A1 (ja) * | 2017-09-26 | 2019-04-04 | 住友化学株式会社 | 複素環化合物及びそれを含有する有害節足動物防除剤 |
| BR112020006659B1 (pt) | 2017-10-04 | 2022-01-25 | Bayer Aktiengesellschaft | Derivados de compostos heterocíclicos, formulação agroquímica, método para controlar uma ou mais pragas animais, e produto |
| US11555035B2 (en) | 2017-12-22 | 2023-01-17 | Sumitomo Chemical Company, Limited | Heterocyclic compound and harmful arthropod-controlling agent containing same |
| AU2019254499A1 (en) | 2018-04-20 | 2020-12-03 | Bayer Aktiengesellschaft | Heterocyclene derivatives as pest control agents |
| WO2019219689A1 (en) | 2018-05-18 | 2019-11-21 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfoximine containing substituents |
| WO2019229089A1 (en) | 2018-05-31 | 2019-12-05 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| CN112368280B (zh) | 2018-06-26 | 2023-01-20 | 拜耳公司 | 作为害虫防治剂的杂环衍生物 |
| TW202035404A (zh) | 2018-10-24 | 2020-10-01 | 瑞士商先正達農作物保護公司 | 具有含亞碸亞胺的取代基之殺有害生物活性雜環衍生物 |
| WO2021009311A1 (en) | 2019-07-17 | 2021-01-21 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| UA128104C2 (uk) | 2019-09-12 | 2024-04-03 | Ніхон Нохіяку Ко., Лтд. | Сільськогосподарський або садовий інсектицид або засіб для боротьби з ектопаразитами або ендопаразитами тварин, кожен з яких включає імідазопіридазинову сполуку, яка містить заміщену циклопропаноксадіазольну групу, або її сіль як активний інгредієнт, і спосіб застосування вказаного інсектициду або засобу для боротьби |
| TW202120479A (zh) | 2019-11-27 | 2021-06-01 | 瑞士商先正達農作物保護公司 | 用於製備具有3-含硫取代基的5-氯-吡啶-2-羧酸及羧酸酯之方法 |
| TW202134214A (zh) | 2020-03-04 | 2021-09-16 | 瑞士商先正達農作物保護公司 | 用於製備具有3-含硫取代基的5-氯-吡啶-2-甲酸醯胺以及甲酸鹽之方法 |
| WO2021219810A1 (en) | 2020-04-30 | 2021-11-04 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| EP4175961A1 (de) | 2020-07-02 | 2023-05-10 | Bayer Aktiengesellschaft | Heterocyclen-derivate als schädlingsbekämpfungsmittel |
| CN116917276A (zh) | 2021-03-01 | 2023-10-20 | 日本农药株式会社 | 具有磺酰胺基的缩合杂环化合物或其盐类及含有该化合物或其盐类的农业园艺用杀虫剂或者动物用的外部或内部寄生虫防除剂以及其使用方法 |
| KR20240088848A (ko) | 2021-09-13 | 2024-06-20 | 베링거잉겔하임베트메디카게엠베하 | 사이클로프로필-(헤테로)아릴-치환된 에틸설포닐-피리딘 유도체 |
| CN121001995A (zh) * | 2022-12-16 | 2025-11-21 | 腾维治疗公司 | 化合物、组合物和方法 |
| US20240300957A1 (en) | 2023-02-23 | 2024-09-12 | Boehringer Ingelheim Vetmedica Gmbh | Tetrazole-substituted ethyl-sulfone / sulfoximine-pyridine derivatives |
| CN120882309A (zh) | 2023-03-14 | 2025-10-31 | 先正达农作物保护股份公司 | 对杀昆虫剂具有抗性的有害生物的控制 |
| CN116585740A (zh) * | 2023-05-04 | 2023-08-15 | 中国科学院沈阳应用生态研究所 | 一种枸杞提取物及制备方法、应用 |
| WO2025026738A1 (en) | 2023-07-31 | 2025-02-06 | Bayer Aktiengesellschaft | 6-[5-(ethylsulfonyl)-1-methyl-1h-imidazol-4-yl]-7-methyl-3-(pentafluoroethyl)-7h-imidazo[4,5-c]pyridazine derivatives as pesticides |
| CN117534677B (zh) * | 2024-01-09 | 2024-03-12 | 广东省农业科学院农业质量标准与监测技术研究所 | 一类含亚胺的三环稠合杂环化合物及其应用 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW201234965A (en) | 2010-12-24 | 2012-09-01 | Sumitomo Chemical Co | Fused heterocyclic compound and use for pest control thereof |
| WO2013187424A1 (ja) * | 2012-06-15 | 2013-12-19 | 住友化学株式会社 | 有害節足動物防除組成物及び有害節足動物の防除方法 |
| EP2961275A4 (en) * | 2013-02-13 | 2016-07-27 | Sumitomo Chemical Co | PEST CONTROL COMPOSITION AND USE THEREOF |
| UY35421A (es) | 2013-03-15 | 2014-10-31 | Nihon Nohyaku Co Ltd | Compuesto heterocíclico condensado o su sal, insecticida agrícola u hortícola que comprende el comp uesto y método de uso del insecticida |
| WO2016039444A1 (ja) * | 2014-09-12 | 2016-03-17 | 日本農薬株式会社 | イミダゾピリダジン化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法 |
| TW201625522A (zh) * | 2014-09-12 | 2016-07-16 | Nihon Nohyaku Co Ltd | 咪唑嗒化合物或其鹽類及含有該化合物之農園藝用殺蟲劑及其使用方法 |
-
2015
- 2015-10-15 EP EP15780882.5A patent/EP3207044B1/en not_active Not-in-force
- 2015-10-15 ES ES15780882.5T patent/ES2690131T3/es active Active
- 2015-10-15 CN CN201580055740.8A patent/CN106795167B/zh not_active Expired - Fee Related
- 2015-10-15 WO PCT/EP2015/073856 patent/WO2016059145A1/en not_active Ceased
- 2015-10-15 US US15/518,833 patent/US10544148B2/en not_active Expired - Fee Related
- 2015-10-15 JP JP2017520319A patent/JP6675390B2/ja not_active Expired - Fee Related
- 2015-10-15 BR BR112017007510A patent/BR112017007510A2/pt active Search and Examination