JP2017528519A5 - - Google Patents
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- Publication number
- JP2017528519A5 JP2017528519A5 JP2017530971A JP2017530971A JP2017528519A5 JP 2017528519 A5 JP2017528519 A5 JP 2017528519A5 JP 2017530971 A JP2017530971 A JP 2017530971A JP 2017530971 A JP2017530971 A JP 2017530971A JP 2017528519 A5 JP2017528519 A5 JP 2017528519A5
- Authority
- JP
- Japan
- Prior art keywords
- pyridin
- methoxy
- benzoxazol
- methyl
- methoxypyridin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462043603P | 2014-08-29 | 2014-08-29 | |
| US62/043,603 | 2014-08-29 | ||
| PCT/US2015/047407 WO2016033445A1 (en) | 2014-08-29 | 2015-08-28 | Probes for imaging huntingtin protein |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020214504A Division JP7126541B2 (ja) | 2014-08-29 | 2020-12-24 | ハンチントンタンパク質のイメージング用プローブ |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017528519A JP2017528519A (ja) | 2017-09-28 |
| JP2017528519A5 true JP2017528519A5 (https=) | 2018-10-04 |
| JP6817207B2 JP6817207B2 (ja) | 2021-01-20 |
Family
ID=55400648
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017530971A Active JP6817207B2 (ja) | 2014-08-29 | 2015-08-28 | ハンチントンタンパク質のイメージング用プローブ |
| JP2020214504A Active JP7126541B2 (ja) | 2014-08-29 | 2020-12-24 | ハンチントンタンパク質のイメージング用プローブ |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020214504A Active JP7126541B2 (ja) | 2014-08-29 | 2020-12-24 | ハンチントンタンパク質のイメージング用プローブ |
Country Status (20)
| Country | Link |
|---|---|
| US (3) | US10479802B2 (https=) |
| EP (2) | EP3186233B8 (https=) |
| JP (2) | JP6817207B2 (https=) |
| KR (2) | KR102456946B1 (https=) |
| CN (2) | CN116655618B (https=) |
| AU (1) | AU2015308774B2 (https=) |
| BR (1) | BR112017004141B8 (https=) |
| CA (1) | CA2959501C (https=) |
| DK (1) | DK3186233T3 (https=) |
| EA (1) | EA035646B1 (https=) |
| ES (1) | ES2898965T3 (https=) |
| HR (1) | HRP20211778T1 (https=) |
| HU (1) | HUE056957T2 (https=) |
| IL (1) | IL250803B (https=) |
| MX (2) | MX380810B (https=) |
| PL (1) | PL3186233T3 (https=) |
| PT (1) | PT3186233T (https=) |
| SG (1) | SG11201701600QA (https=) |
| SI (1) | SI3186233T1 (https=) |
| WO (1) | WO2016033445A1 (https=) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3186241B1 (en) | 2014-08-29 | 2020-10-07 | CHDI Foundation, Inc. | Probes for imaging huntington protein |
| DK3197277T3 (da) | 2014-08-29 | 2022-01-31 | Chdi Foundation Inc | Prober til billeddannelse af huntingtin-protein |
| AU2015308709B2 (en) | 2014-08-29 | 2020-01-02 | Chdi Foundation, Inc. | Probes for imaging huntingtin protein |
| HUE056957T2 (hu) * | 2014-08-29 | 2022-04-28 | Chdi Foundation Inc | Próbák huntingtin fehérjét megjelenítõ képalkotásra |
| PT3340796T (pt) | 2015-08-28 | 2021-07-28 | Chdi Foundation Inc | Sondas para imagens da proteína huntingtina |
| NZ746901A (en) | 2016-03-11 | 2023-06-30 | Ac Immune Sa | Bicyclic compounds for diagnosis and therapy |
| CN107056723A (zh) * | 2017-04-21 | 2017-08-18 | 云南大学 | 一种具有抑制血管内皮生长因子受体信号传导的化合物 |
| CA3075892C (en) | 2017-09-14 | 2024-01-23 | Daiichi Sankyo Company, Limited | Heterocyclic compounds for the treatment and/or prevention of inflammatory diseases |
| AU2019254499A1 (en) | 2018-04-20 | 2020-12-03 | Bayer Aktiengesellschaft | Heterocyclene derivatives as pest control agents |
| IL279219B2 (en) | 2018-06-08 | 2024-08-01 | Ac Immune Sa | Novel compounds for diagnosis |
| ES2974634T3 (es) | 2018-12-21 | 2024-06-28 | Celgene Corp | Inhibidores de tienopiridinas de RIPK2 |
| JP7619952B2 (ja) | 2019-02-25 | 2025-01-22 | シーエイチディーアイ ファウンデーション，インコーポレーテッド | 変異型ハンチンチンタンパク質を標的とするための化合物及びその使用 |
| CN111635400A (zh) | 2019-03-02 | 2020-09-08 | 察略盛医药科技(上海)有限公司 | 吡唑并[1,5-a]吡啶类衍生物、及其制备方法和用途 |
| JP7720847B2 (ja) * | 2019-12-18 | 2025-08-08 | シーエイチディーアイ ファウンデーション，インコーポレーテッド | ハンチンチンタンパク質をイメージングするための化合物及びプローブ |
| KR20220140515A (ko) | 2020-01-13 | 2022-10-18 | 버지 애널리틱스, 인크. | 치환된 피라졸로-피리미딘 및 그의 용도 |
| EP4146653A1 (en) | 2020-05-07 | 2023-03-15 | AC Immune SA | Novel compounds for diagnosis |
| WO2022031946A1 (en) * | 2020-08-06 | 2022-02-10 | Chdi Foundation, Inc. | Heterobiaryl compounds and imaging agents for imaging huntingtin protein |
| CN117412960A (zh) * | 2021-04-08 | 2024-01-16 | Chdi基金会股份有限公司 | 用于对亨廷顿蛋白成像的异吲哚啉酮化合物和显像剂 |
| AU2022264490A1 (en) * | 2021-04-27 | 2023-11-09 | Chdi Foundation, Inc. | Deuterated compounds and imaging agents for imaging huntingtin protein |
| KR20240035820A (ko) | 2021-07-09 | 2024-03-18 | 플렉시움 인코포레이티드 | Ikzf2를 조절하는 아릴 화합물 및 약학 조성물 |
| EP4430044A1 (en) | 2021-11-10 | 2024-09-18 | AC Immune SA | Dihydropyrrolo[3,4-c]pyrazole derivatives and their use in diagnosis |
| WO2023083998A1 (en) | 2021-11-10 | 2023-05-19 | Ac Immune Sa | Dihydropyrrolo[3,4c]-pyrazole derivatives and their use in diagnosis |
| JP2024544539A (ja) | 2021-11-10 | 2024-12-03 | エーシー・イミューン・エス・アー | 診断のための４ｈ－イミダゾ［１，５－ｂ］ピラゾール誘導体 |
| TW202425965A (zh) | 2022-09-30 | 2024-07-01 | 日商科研製藥股份有限公司 | 縮環化合物及含有其之醫藥 |
| EP4634191A1 (en) | 2022-12-16 | 2025-10-22 | AC Immune SA | Novel compounds for diagnosis |
| EP4634190A1 (en) | 2022-12-16 | 2025-10-22 | AC Immune SA | Novel compounds for diagnosis |
| WO2024239000A2 (en) * | 2023-05-18 | 2024-11-21 | Enveda Therapeutics, Inc. | G-protein coupled receptor antagonist |
| WO2025037013A1 (en) | 2023-08-16 | 2025-02-20 | Ac Immune Sa | Diagnostic compounds that bind to alpha-synuclein |
| WO2025106920A1 (en) * | 2023-11-15 | 2025-05-22 | Yale University | Parp pet imaging agents and methods of using the same |
| CN119264072B (zh) * | 2024-12-06 | 2025-05-02 | 国科大杭州高等研究院 | 对细胞成像的荧光探针及其合成方法和应用 |
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| AU2015308709B2 (en) | 2014-08-29 | 2020-01-02 | Chdi Foundation, Inc. | Probes for imaging huntingtin protein |
| HUE056957T2 (hu) * | 2014-08-29 | 2022-04-28 | Chdi Foundation Inc | Próbák huntingtin fehérjét megjelenítõ képalkotásra |
| DK3197277T3 (da) | 2014-08-29 | 2022-01-31 | Chdi Foundation Inc | Prober til billeddannelse af huntingtin-protein |
| EP3186241B1 (en) | 2014-08-29 | 2020-10-07 | CHDI Foundation, Inc. | Probes for imaging huntington protein |
| PT3340796T (pt) | 2015-08-28 | 2021-07-28 | Chdi Foundation Inc | Sondas para imagens da proteína huntingtina |
-
2015
- 2015-08-28 HU HUE15836321A patent/HUE056957T2/hu unknown
- 2015-08-28 AU AU2015308774A patent/AU2015308774B2/en active Active
- 2015-08-28 KR KR1020177008383A patent/KR102456946B1/ko active Active
- 2015-08-28 CA CA2959501A patent/CA2959501C/en active Active
- 2015-08-28 HR HRP20211778TT patent/HRP20211778T1/hr unknown
- 2015-08-28 CN CN202310475134.8A patent/CN116655618B/zh active Active
- 2015-08-28 PT PT158363218T patent/PT3186233T/pt unknown
- 2015-08-28 CN CN201580058282.3A patent/CN107108534B/zh active Active
- 2015-08-28 EP EP15836321.8A patent/EP3186233B8/en active Active
- 2015-08-28 BR BR112017004141A patent/BR112017004141B8/pt active IP Right Grant
- 2015-08-28 EP EP21192872.6A patent/EP4006016A3/en not_active Withdrawn
- 2015-08-28 DK DK15836321.8T patent/DK3186233T3/da active
- 2015-08-28 KR KR1020227035965A patent/KR102586736B1/ko active Active
- 2015-08-28 US US15/507,208 patent/US10479802B2/en active Active
- 2015-08-28 SG SG11201701600QA patent/SG11201701600QA/en unknown
- 2015-08-28 WO PCT/US2015/047407 patent/WO2016033445A1/en not_active Ceased
- 2015-08-28 MX MX2017002703A patent/MX380810B/es unknown
- 2015-08-28 SI SI201531751T patent/SI3186233T1/sl unknown
- 2015-08-28 JP JP2017530971A patent/JP6817207B2/ja active Active
- 2015-08-28 EA EA201790407A patent/EA035646B1/ru unknown
- 2015-08-28 PL PL15836321T patent/PL3186233T3/pl unknown
- 2015-08-28 ES ES15836321T patent/ES2898965T3/es active Active
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2017
- 2017-02-27 IL IL250803A patent/IL250803B/en active IP Right Grant
- 2017-02-28 MX MX2021003311A patent/MX2021003311A/es unknown
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2019
- 2019-08-02 US US16/530,594 patent/US11059836B2/en active Active
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2020
- 2020-12-24 JP JP2020214504A patent/JP7126541B2/ja active Active
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2022
- 2022-08-05 US US17/881,895 patent/US12258355B2/en active Active