JP2017503760A5 - - Google Patents

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Publication number
JP2017503760A5
JP2017503760A5 JP2016534901A JP2016534901A JP2017503760A5 JP 2017503760 A5 JP2017503760 A5 JP 2017503760A5 JP 2016534901 A JP2016534901 A JP 2016534901A JP 2016534901 A JP2016534901 A JP 2016534901A JP 2017503760 A5 JP2017503760 A5 JP 2017503760A5
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JP
Japan
Prior art keywords
alkyl
group
cycloalkyl
atoms
membered aromatic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2016534901A
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English (en)
Japanese (ja)
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JP2017503760A (ja
JP6441928B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2014/075358 external-priority patent/WO2015078802A1/en
Publication of JP2017503760A publication Critical patent/JP2017503760A/ja
Publication of JP2017503760A5 publication Critical patent/JP2017503760A5/ja
Application granted granted Critical
Publication of JP6441928B2 publication Critical patent/JP6441928B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2016534901A 2013-11-28 2014-11-24 新規インダニルオキシフェニルシクロプロパンカルボン酸 Expired - Fee Related JP6441928B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13194945 2013-11-28
EP13194945.5 2013-11-28
PCT/EP2014/075358 WO2015078802A1 (en) 2013-11-28 2014-11-24 New indanyloxyphenylcyclopropanecarboxylic acids

Publications (3)

Publication Number Publication Date
JP2017503760A JP2017503760A (ja) 2017-02-02
JP2017503760A5 true JP2017503760A5 (enExample) 2018-01-11
JP6441928B2 JP6441928B2 (ja) 2018-12-19

Family

ID=49726512

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016534901A Expired - Fee Related JP6441928B2 (ja) 2013-11-28 2014-11-24 新規インダニルオキシフェニルシクロプロパンカルボン酸

Country Status (4)

Country Link
US (1) US9308194B2 (enExample)
EP (1) EP3074375B1 (enExample)
JP (1) JP6441928B2 (enExample)
WO (1) WO2015078802A1 (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018095877A1 (en) * 2016-11-28 2018-05-31 Boehringer Ingelheim International Gmbh Indanylaminopyridylcyclopropanecarboxylic acids, pharmaceutical compositions and uses thereof
US10253004B2 (en) * 2017-01-26 2019-04-09 Boehringer Ingelheim International Gmbh Indanylaminopyrazinylcyclopropanecarboxylic acids, pharmaceutical compositions and uses thereof
EP3580222B1 (en) * 2017-02-08 2021-04-07 Boehringer Ingelheim International GmbH Indanylaminoazadihydrobenzofuranylacetic acids, pharmaceutical compositions for the treatment of diabetes
BR102018007822A2 (pt) 2017-04-20 2018-11-06 Gilead Sciences, Inc. composto, métodos para inibir pd-1, pd-l1 e/ou interação de pd-1/pd-l1 e para tratamento de câncer, composição farmacêutica, e, kit para tratamento de ou prevenção de câncer ou uma doença ou condição
KR102708681B1 (ko) 2018-02-13 2024-09-26 길리애드 사이언시즈, 인코포레이티드 Pd-1/pd-l1 억제제
EP4600247A3 (en) 2018-04-19 2025-11-19 Gilead Sciences, Inc. Pd-1/pd-l1 inhibitors
UA126421C2 (uk) 2018-07-13 2022-09-28 Гіліад Сайєнсіз, Інк. Інгібітори pd-1/pd-l1
US11236085B2 (en) 2018-10-24 2022-02-01 Gilead Sciences, Inc. PD-1/PD-L1 inhibitors
JP7135931B2 (ja) 2019-02-22 2022-09-13 スズキ株式会社 車両の走行制御装置
BR112022006546A2 (pt) 2019-10-07 2022-08-30 Kallyope Inc Agonistas de gpr119
CA3173731A1 (en) 2020-02-28 2021-09-02 Kallyope, Inc. Gpr40 agonists
CN116323608A (zh) 2020-05-19 2023-06-23 卡尔优普公司 Ampk活化剂
EP4172162A4 (en) 2020-06-26 2024-08-07 Kallyope, Inc. AMPK ACTIVATORS

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20030701A1 (es) * 2001-12-20 2003-08-21 Schering Corp Compuestos para el tratamiento de trastornos inflamatorios
CA2727340A1 (en) * 2008-06-25 2009-12-30 Daiichi Sankyo Company, Limited Carboxylic acid compound
EP2646425B1 (en) * 2010-12-01 2015-06-10 Boehringer Ingelheim International Gmbh Indanyloxydihydrobenzofuranylacetic acids useful for the treatment of metabolic syndrome

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