JP2016518369A5 - - Google Patents
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- Publication number
- JP2016518369A5 JP2016518369A5 JP2016508974A JP2016508974A JP2016518369A5 JP 2016518369 A5 JP2016518369 A5 JP 2016518369A5 JP 2016508974 A JP2016508974 A JP 2016508974A JP 2016508974 A JP2016508974 A JP 2016508974A JP 2016518369 A5 JP2016518369 A5 JP 2016518369A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- haloalkyl
- halogen
- independently
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- 229910052736 halogen Inorganic materials 0.000 claims description 35
- 150000002367 halogens Chemical class 0.000 claims description 35
- 125000001188 haloalkyl group Chemical group 0.000 claims description 22
- 125000000217 alkyl group Chemical group 0.000 claims description 21
- 125000004432 carbon atom Chemical group C* 0.000 claims description 20
- 125000001424 substituent group Chemical group 0.000 claims description 18
- 150000001875 compounds Chemical class 0.000 claims description 12
- 125000004433 nitrogen atom Chemical group N* 0.000 claims description 10
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 10
- 229910052799 carbon Inorganic materials 0.000 claims description 8
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 8
- 125000003545 alkoxy group Chemical group 0.000 claims description 6
- 230000000844 anti-bacterial effect Effects 0.000 claims description 6
- 230000000855 fungicidal effect Effects 0.000 claims description 6
- 125000004430 oxygen atom Chemical group O* 0.000 claims description 6
- 125000004434 sulfur atom Chemical group 0.000 claims description 6
- 125000004076 pyridyl group Chemical group 0.000 claims description 5
- 125000000623 heterocyclic group Chemical group 0.000 claims description 4
- 229910052739 hydrogen Inorganic materials 0.000 claims description 4
- 125000004438 haloalkoxy group Chemical group 0.000 claims description 3
- 125000006677 (C1-C3) haloalkoxy group Chemical group 0.000 claims description 2
- 125000001054 5 membered carbocyclic group Chemical group 0.000 claims description 2
- 125000004008 6 membered carbocyclic group Chemical group 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- 125000003118 aryl group Chemical group 0.000 claims description 2
- 201000010099 disease Diseases 0.000 claims description 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims description 2
- 244000000004 fungal plant pathogen Species 0.000 claims description 2
- 239000000417 fungicide Substances 0.000 claims description 2
- 125000005842 heteroatom Chemical group 0.000 claims description 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims description 2
- 229910052760 oxygen Inorganic materials 0.000 claims description 2
- 125000003373 pyrazinyl group Chemical group 0.000 claims description 2
- 125000002098 pyridazinyl group Chemical group 0.000 claims description 2
- 150000003839 salts Chemical class 0.000 claims description 2
- 229910052717 sulfur Inorganic materials 0.000 claims description 2
- 125000004665 trialkylsilyl group Chemical group 0.000 claims description 2
- 239000003899 bactericide agent Substances 0.000 claims 1
- 229910052801 chlorine Inorganic materials 0.000 description 12
- 229910052731 fluorine Inorganic materials 0.000 description 12
- 229910052794 bromium Inorganic materials 0.000 description 11
- 125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 description 6
- -1 3-oxetanyl Chemical group 0.000 description 2
- 239000003085 diluting agent Substances 0.000 description 2
- 125000006729 (C2-C5) alkenyl group Chemical group 0.000 description 1
- 125000006645 (C3-C4) cycloalkyl group Chemical group 0.000 description 1
- 0 C*C(*)(*=C)N(C(N)=*)N Chemical compound C*C(*)(*=C)N(C(N)=*)N 0.000 description 1
- VGHAUGKHGKPTCM-UHFFFAOYSA-N N-[[2-chloro-4-[3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]-N-cyclopropyl-3-(difluoromethyl)-5-fluoro-1-methylpyrazole-4-carboxamide Chemical compound Cn1nc(C(F)F)c(C(=O)N(Cc2ccc(cc2Cl)-n2ccc(n2)C(F)(F)F)C2CC2)c1F VGHAUGKHGKPTCM-UHFFFAOYSA-N 0.000 description 1
- 239000007788 liquid Substances 0.000 description 1
- BNTPBQKHADWSSB-UHFFFAOYSA-N n-cyclopropyl-3-(difluoromethyl)-5-fluoro-1-methyl-n-[[3-[3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]pyrazole-4-carboxamide Chemical compound CN1N=C(C(F)F)C(C(=O)N(CC=2C=C(C=CC=2)N2N=C(C=C2)C(F)(F)F)C2CC2)=C1F BNTPBQKHADWSSB-UHFFFAOYSA-N 0.000 description 1
- 239000007787 solid Substances 0.000 description 1
- 239000004094 surface-active agent Substances 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361811919P | 2013-04-15 | 2013-04-15 | |
| US61/811,919 | 2013-04-15 | ||
| PCT/US2014/033766 WO2014172191A1 (en) | 2013-04-15 | 2014-04-11 | Fungicidal carboxamides |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2016518369A JP2016518369A (ja) | 2016-06-23 |
| JP2016518369A5 true JP2016518369A5 (https=) | 2017-04-13 |
Family
ID=50680209
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016508974A Ceased JP2016518369A (ja) | 2013-04-15 | 2014-04-11 | 殺菌・殺カビ性アミド |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US10098350B2 (https=) |
| EP (1) | EP2986601B1 (https=) |
| JP (1) | JP2016518369A (https=) |
| KR (1) | KR20150143650A (https=) |
| CN (1) | CN105263920B (https=) |
| AU (1) | AU2014254262B2 (https=) |
| BR (1) | BR112015025647A2 (https=) |
| CL (1) | CL2015003007A1 (https=) |
| MX (1) | MX2015014406A (https=) |
| PL (1) | PL2986601T3 (https=) |
| WO (1) | WO2014172191A1 (https=) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR112015025686B1 (pt) | 2013-04-15 | 2020-10-27 | Fmc Corporation | composto, composições fungicidas e método para o controle das doenças dos vegetais |
| WO2015082587A1 (en) * | 2013-12-05 | 2015-06-11 | Bayer Cropscience Ag | N-cycloalkyl-n-{[2-(1-substitutedcycloalkyl)phenyl]methylene}-(thio)carboxamide derivatives |
| WO2016094307A1 (en) | 2014-12-08 | 2016-06-16 | The Research Foundation For The State University Of New York | Anti-fungals targeting the synthesis of fungal shingolipids |
| CN105181873B (zh) * | 2015-10-10 | 2016-10-05 | 浙江中一检测研究院股份有限公司 | 一种土壤中硫双威的简便测定方法 |
| WO2018165520A1 (en) | 2017-03-10 | 2018-09-13 | Vps-3, Inc. | Metalloenzyme inhibitor compounds |
| WO2018232298A1 (en) | 2017-06-16 | 2018-12-20 | The Research Foundation For The State University Of New York | Anti-fungals compounds targeting the synthesis of fungal sphingolipids |
| CN107384884B (zh) * | 2017-08-22 | 2020-01-31 | 中国农业科学院蔬菜花卉研究所 | 一种多主棒孢菌琥珀酸脱氢酶B亚基基因sdhB的等位基因及应用 |
| US20210002232A1 (en) * | 2018-03-09 | 2021-01-07 | Pi Industries Ltd. | Heterocyclic compounds as fungicides |
| WO2020113094A1 (en) | 2018-11-30 | 2020-06-04 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
| CN110208405A (zh) * | 2019-05-30 | 2019-09-06 | 江苏恒生检测有限公司 | 一种检测水稻上呋虫胺残留的方法 |
| AU2020321955A1 (en) | 2019-07-30 | 2022-03-17 | Eikonizo Therapapeutics, Inc. | HDAC6 inhibitors and uses thereof |
| KR102614653B1 (ko) * | 2021-06-09 | 2023-12-20 | 한국과학기술연구원 | 신규한 헤테로사이클릴-페닐-메틸아민 유도체, 이의 제조방법 및 이의 다발성 경화증 예방, 개선, 또는 치료 용도 |
| IL316201A (en) | 2022-04-08 | 2024-12-01 | Eikonizo Therapeutics Inc | Oxadiazole HDAC6 inhibitors and their uses |
| CN116082240B (zh) * | 2023-02-07 | 2025-04-01 | 华中农业大学 | 一种琥珀酸脱氢酶抑制剂及其合成方法与应用 |
Family Cites Families (49)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2891855A (en) | 1954-08-16 | 1959-06-23 | Geigy Ag J R | Compositions and methods for influencing the growth of plants |
| US3235361A (en) | 1962-10-29 | 1966-02-15 | Du Pont | Method for the control of undesirable vegetation |
| US3060084A (en) | 1961-06-09 | 1962-10-23 | Du Pont | Improved homogeneous, readily dispersed, pesticidal concentrate |
| US3299566A (en) | 1964-06-01 | 1967-01-24 | Olin Mathieson | Water soluble film containing agricultural chemicals |
| US3309192A (en) | 1964-12-02 | 1967-03-14 | Du Pont | Method of controlling seedling weed grasses |
| US4144050A (en) | 1969-02-05 | 1979-03-13 | Hoechst Aktiengesellschaft | Micro granules for pesticides and process for their manufacture |
| US3920442A (en) | 1972-09-18 | 1975-11-18 | Du Pont | Water-dispersible pesticide aggregates |
| US4172714A (en) | 1976-12-20 | 1979-10-30 | E. I. Du Pont De Nemours And Company | Dry compactible, swellable herbicidal compositions and pellets produced therefrom |
| GB2095558B (en) | 1981-03-30 | 1984-10-24 | Avon Packers Ltd | Formulation of agricultural chemicals |
| DE3246493A1 (de) | 1982-12-16 | 1984-06-20 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von wasserdispergierbaren granulaten |
| US5180587A (en) | 1988-06-28 | 1993-01-19 | E. I. Du Pont De Nemours And Company | Tablet formulations of pesticides |
| DE69033861T2 (de) | 1989-08-30 | 2002-06-06 | Kynoch Agrochemicals (Proprietary) Ltd., Sandton | Herstellung eines Dosierungsmittels |
| ES2065680T3 (es) | 1990-03-12 | 1995-02-16 | Du Pont | Granulos de plaguicida dispersables en agua o solubles en agua a partir de aglutinantes activados por calor. |
| EP0480679B1 (en) | 1990-10-11 | 1996-09-18 | Sumitomo Chemical Company Limited | Pesticidal composition |
| US6406690B1 (en) | 1995-04-17 | 2002-06-18 | Minrav Industries Ltd. | Bacillus firmus CNCM I-1582 or Bacillus cereus CNCM I-1562 for controlling nematodes |
| EP1054011B1 (en) | 1998-02-06 | 2006-09-13 | Meiji Seika Kaisha Ltd. | Novel antifungal compounds and process for producing the same |
| CN1237051C (zh) | 1999-08-20 | 2006-01-18 | 道农业科学公司 | 杀真菌的杂环芳族酰胺和它们的组合物、使用方法和制备 |
| TWI283164B (en) | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| AR037328A1 (es) | 2001-10-23 | 2004-11-03 | Dow Agrosciences Llc | Compuesto de [7-bencil-2,6-dioxo-1,5-dioxonan-3-il]-4-metoxipiridin-2-carboxamida, composicion que lo comprende y metodo que lo utiliza |
| GB0227555D0 (en) | 2002-11-26 | 2002-12-31 | Syngenta Ltd | Fungicides |
| GB0312863D0 (en) | 2003-06-04 | 2003-07-09 | Syngenta Ltd | Fungicides |
| US7224810B2 (en) | 2003-09-12 | 2007-05-29 | Spatializer Audio Laboratories, Inc. | Noise reduction system |
| GB0426372D0 (en) | 2004-12-01 | 2005-01-05 | Syngenta Ltd | Fungicides |
| GB0426373D0 (en) | 2004-12-01 | 2005-01-05 | Syngenta Ltd | Fungicides |
| BRPI0612945B1 (pt) | 2005-05-13 | 2018-11-06 | Bayer Cropscience Sa | composto e método para o combate de fungo fitopatogênico |
| BRPI0614141A2 (pt) | 2005-08-05 | 2016-11-22 | Basf Se | composto, composição fungicida, uso de compostos, método para controlar fungos nocivos fitopatogênicos, e, semente |
| GB0704906D0 (en) | 2007-03-14 | 2007-04-25 | Syngenta Participations Ag | Fungicides |
| WO2008124092A2 (en) | 2007-04-03 | 2008-10-16 | E. I. Du Pont De Nemours And Company | Substituted benzene fungicides |
| PE20090277A1 (es) | 2007-04-24 | 2009-04-06 | Takeda Pharmaceutical | Derivados de piperidina como antagonistas de taquiquininas |
| WO2009016220A1 (en) * | 2007-07-31 | 2009-02-05 | Bayer Cropscience Sa | Fungicidal n-cycloalkyl-benzyl-thiocarboxamides or n-cycloalkyl-benzyl-n' -substituted-amidine derivatives |
| GB0717260D0 (en) | 2007-09-05 | 2007-10-17 | Syngenta Participations Ag | Novel fungicides |
| GB0717258D0 (en) | 2007-09-05 | 2007-10-17 | Syngenta Participations Ag | Novel fungicides |
| GB0800407D0 (en) | 2008-01-10 | 2008-02-20 | Syngenta Participations Ag | Fungicides |
| BRPI0910837B1 (pt) | 2008-04-30 | 2017-03-07 | Bayer Cropscience Ag | ésteres e tioésteres tiazol-4-carboxílicos, seus usos, e método e composição para controlar fungos fitopatogênicos prejudiciais |
| KR101072284B1 (ko) * | 2008-08-01 | 2011-10-11 | 주식회사 케이엠더블유 | 고주파 필터의 유전체 공진기 및 그 조립 방법 |
| AR076839A1 (es) | 2009-05-15 | 2011-07-13 | Bayer Cropscience Ag | Derivados fungicidas de pirazol carboxamidas |
| TW201107329A (en) | 2009-07-30 | 2011-03-01 | Oncotherapy Science Inc | Fused imidazole derivative having ttk inhibitory action |
| PT3153020T (pt) | 2009-10-07 | 2019-02-26 | Dow Agrosciences Llc | Misturas fungicidas sinérgicas para o controlo de fungos em cereais |
| WO2011051243A1 (en) | 2009-10-29 | 2011-05-05 | Bayer Cropscience Ag | Active compound combinations |
| CA2784180C (en) | 2009-12-25 | 2014-03-11 | Daiichi Sankyo Company, Limited | Seven-membered ring compound and pharmaceutical use therefor |
| EP2606051B1 (en) | 2010-08-20 | 2016-10-05 | Hutchison Medipharma Limited | Pyrrolopyrimidine compounds and uses thereof |
| MX2013004278A (es) * | 2010-10-21 | 2013-06-05 | Bayer Ip Gmbh | N-bencil carboxamidas heterociclicas. |
| JP2013542967A (ja) | 2010-11-17 | 2013-11-28 | ノバルティス アーゲー | ３−（アミノアリール）−ピリジン化合物 |
| MX2013006768A (es) | 2010-12-23 | 2013-07-22 | Pfizer | Moduladores de receptor de glucagon. |
| WO2013009971A1 (en) | 2011-07-12 | 2013-01-17 | E. I. Du Pont De Nemours And Company | Detection and screening method and materials useful in performance thereof |
| UA115663C2 (uk) * | 2012-04-20 | 2017-12-11 | Байєр Кропсайнс Аг | (тіо)карбоксамідні похідні n-циклоалкіл-n-[(гетероциклілфеніл)метилену] |
| US8815772B2 (en) * | 2012-06-29 | 2014-08-26 | E I Du Pont De Nemours And Company | Fungicidal heterocyclic carboxamides |
| TWI654180B (zh) | 2012-06-29 | 2019-03-21 | 美商艾佛艾姆希公司 | 殺真菌之雜環羧醯胺 |
| BR112015025686B1 (pt) | 2013-04-15 | 2020-10-27 | Fmc Corporation | composto, composições fungicidas e método para o controle das doenças dos vegetais |
-
2014
- 2014-04-11 US US14/784,172 patent/US10098350B2/en not_active Expired - Fee Related
- 2014-04-11 CN CN201480021362.7A patent/CN105263920B/zh not_active Expired - Fee Related
- 2014-04-11 BR BR112015025647A patent/BR112015025647A2/pt not_active Application Discontinuation
- 2014-04-11 AU AU2014254262A patent/AU2014254262B2/en not_active Ceased
- 2014-04-11 KR KR1020157032286A patent/KR20150143650A/ko not_active Withdrawn
- 2014-04-11 EP EP14722507.2A patent/EP2986601B1/en not_active Not-in-force
- 2014-04-11 PL PL14722507T patent/PL2986601T3/pl unknown
- 2014-04-11 MX MX2015014406A patent/MX2015014406A/es unknown
- 2014-04-11 JP JP2016508974A patent/JP2016518369A/ja not_active Ceased
- 2014-04-11 WO PCT/US2014/033766 patent/WO2014172191A1/en not_active Ceased
-
2015
- 2015-10-09 CL CL2015003007A patent/CL2015003007A1/es unknown
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