JP2015517577A5 - - Google Patents

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Publication number
JP2015517577A5
JP2015517577A5 JP2015514140A JP2015514140A JP2015517577A5 JP 2015517577 A5 JP2015517577 A5 JP 2015517577A5 JP 2015514140 A JP2015514140 A JP 2015514140A JP 2015514140 A JP2015514140 A JP 2015514140A JP 2015517577 A5 JP2015517577 A5 JP 2015517577A5
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JP
Japan
Prior art keywords
aryl
het
nhr
cycloalkyl
independently
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JP2015514140A
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English (en)
Japanese (ja)
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JP2015517577A (ja
JP6653573B2 (ja
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Priority claimed from PCT/US2013/042148 external-priority patent/WO2013177241A1/en
Publication of JP2015517577A publication Critical patent/JP2015517577A/ja
Publication of JP2015517577A5 publication Critical patent/JP2015517577A5/ja
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Publication of JP6653573B2 publication Critical patent/JP6653573B2/ja
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JP2015514140A 2012-05-22 2013-05-22 シクロアルカニル［ｂ］インドール、シクロアルカニル［ｂ］ベンゾフラン、シクロアルカニル［ｂ］ベンゾチオフェンを合成するための方法、化合物および使用の方法 Active JP6653573B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261650039P 2012-05-22 2012-05-22
US61/650,039 2012-05-22
US201361757876P 2013-01-29 2013-01-29
US61/757,876 2013-01-29
PCT/US2013/042148 WO2013177241A1 (en) 2012-05-22 2013-05-22 Method for synthesizing cycloalkanyl(b}indoles, cycloalkanyl(b) benzofurans, cycloalkanyl(b)benzothiophenes, compounds and methods of use

Publications (3)

Publication Number Publication Date
JP2015517577A JP2015517577A (ja) 2015-06-22
JP2015517577A5 true JP2015517577A5 (enExample) 2016-07-07
JP6653573B2 JP6653573B2 (ja) 2020-02-26

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ID=49624309

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015514140A Active JP6653573B2 (ja) 2012-05-22 2013-05-22 シクロアルカニル［ｂ］インドール、シクロアルカニル［ｂ］ベンゾフラン、シクロアルカニル［ｂ］ベンゾチオフェンを合成するための方法、化合物および使用の方法

Country Status (4)

Country Link
US (1) US9598365B2 (enExample)
EP (1) EP2887804B1 (enExample)
JP (1) JP6653573B2 (enExample)
WO (1) WO2013177241A1 (enExample)

Families Citing this family (9)

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AU2015360416A1 (en) 2014-12-10 2017-06-08 Massachusetts Institute Of Technology Fused 1,3-azole derivatives useful for the treatment of proliferative diseases
EP3286172B1 (en) 2015-04-23 2019-06-12 Constellation Pharmaceuticals, Inc. Lsd1 inhibitors and uses thereof
KR102686073B1 (ko) 2015-10-14 2024-07-17 엑스-써마 인코포레이티드 얼음 결정 형성을 감소시키기 위한 조성물 및 방법
CN109071456A (zh) 2016-02-16 2018-12-21 麻省理工学院 作为myc调节剂的max结合剂及其用途
CN109863137B (zh) 2016-10-26 2022-12-16 星座制药公司 Lsd1抑制剂及其医学用途
US11633379B2 (en) * 2017-01-04 2023-04-25 Trustees Of Dartmouth College Methods of inhibiting PCSK9
CA3184282A1 (en) 2020-06-27 2021-12-30 Emre Koyuncu Composition of compounds that modulate cell metabolism and methods of use
US12138243B2 (en) 2021-12-31 2024-11-12 Crescenta Biosciences Antiviral use of FABP4 modulating compounds
CN120590310B (zh) * 2025-08-07 2025-10-28 昆明医科大学 一种吲哚-3-芳基酮衍生物及其制备方法和应用

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ES2230382T3 (es) * 2000-11-03 2005-05-01 Wyeth Ciclopental(b)(1,4)diazpino(6,7,1-hi)indoles como antagonistas de 5ht2c.
TW200307540A (en) 2002-04-25 2003-12-16 Wyeth Corp [1, 4]Diazocino[7, 8, 1-hi] indole derivatives as antipsychotic and antiobesity agents
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