JP2015516959A5 - - Google Patents

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Publication number
JP2015516959A5
JP2015516959A5 JP2015503828A JP2015503828A JP2015516959A5 JP 2015516959 A5 JP2015516959 A5 JP 2015516959A5 JP 2015503828 A JP2015503828 A JP 2015503828A JP 2015503828 A JP2015503828 A JP 2015503828A JP 2015516959 A5 JP2015516959 A5 JP 2015516959A5
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Japan
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formula
carried out
process according
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compound
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JP2015503828A
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English (en)
Japanese (ja)
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JP2015516959A (ja
JP6255550B2 (ja
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Priority claimed from PCT/EP2013/056638 external-priority patent/WO2013149926A1/en
Publication of JP2015516959A publication Critical patent/JP2015516959A/ja
Publication of JP2015516959A5 publication Critical patent/JP2015516959A5/ja
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Publication of JP6255550B2 publication Critical patent/JP6255550B2/ja
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JP2015503828A 2012-04-02 2013-03-28 Ccr3阻害薬の製造方法 Active JP6255550B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP12162852.3 2012-04-02
EP12162852 2012-04-02
PCT/EP2013/056638 WO2013149926A1 (en) 2012-04-02 2013-03-28 Process for the manufacturing of ccr3 inhibitors

Publications (3)

Publication Number Publication Date
JP2015516959A JP2015516959A (ja) 2015-06-18
JP2015516959A5 true JP2015516959A5 (https=) 2016-05-26
JP6255550B2 JP6255550B2 (ja) 2018-01-10

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ID=47998462

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015503828A Active JP6255550B2 (ja) 2012-04-02 2013-03-28 Ccr3阻害薬の製造方法

Country Status (9)

Country Link
US (1) US8680280B2 (https=)
EP (1) EP2834229B1 (https=)
JP (1) JP6255550B2 (https=)
AR (1) AR090566A1 (https=)
DK (1) DK2834229T3 (https=)
ES (1) ES2641862T3 (https=)
TW (1) TW201400474A (https=)
UY (1) UY34719A (https=)
WO (1) WO2013149926A1 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
AR090566A1 (es) 2012-04-02 2014-11-19 Boehringer Ingelheim Int Proceso para la produccion de inhibidores de crr
US10213421B2 (en) 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
MY199462A (en) 2017-04-05 2023-10-30 Alkahest Inc Methods and compositions for treating retina-associated disease using ccr3-inhibitors
SG11201909245PA (en) 2017-04-05 2019-11-28 Alkahest Inc Methods and compositions for treating aging-associated impairments using ccr3-inhibitors
MY198220A (en) 2018-05-15 2023-08-14 Alkahest Inc Treatment Of Aging-Associated Disease With Modulators Of Leukotriene A4 Hydrolase
AU2021287906B2 (en) 2020-06-11 2025-09-11 Alkahest Inc. Methods of improving retina-associated disease outcome using CCR3-inhibitors
AU2022376563A1 (en) 2021-11-01 2023-12-07 Alkahest, Inc. Benzodioxane modulators of leukotriene a4 hydrolase (lta4h) for prevention and treatment of aging-associated diseases

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE7907121L (sv) 1979-08-27 1981-02-28 Astra Laekemedel Ab Ftalimidinderivat
JP2807577B2 (ja) 1990-06-15 1998-10-08 エーザイ株式会社 環状アミド誘導体
JPH08134041A (ja) * 1994-11-10 1996-05-28 Fuji Photo Film Co Ltd ピラゾールアミド類の製造方法
US6433165B1 (en) 1998-01-21 2002-08-13 Millennium Pharmaceuticals, Inc. Chemokine receptor antagonists and methods of use therefor
WO1999038514A1 (en) 1998-02-02 1999-08-05 Merck & Co., Inc. Cyclic amine modulators of chemokine receptor activity
US6140349A (en) 1998-02-02 2000-10-31 Merck & Co., Inc. Cyclic amine modulators of chemokine receptor activity
EP1725235B1 (en) 2004-02-05 2009-04-15 Schering Corporation Piperidine derivatives useful as ccr3 antagonists
JP2006137718A (ja) 2004-11-12 2006-06-01 Astellas Pharma Inc インドール若しくはインダゾール誘導体
US8030003B2 (en) 2004-12-07 2011-10-04 Children's Hospital Medical Center Diagnosis of eosinophilic esophagitis based on presence of an elevated level of eotaxin-3
DOP2006000051A (es) 2005-02-24 2006-08-31 Lilly Co Eli Inhibidores de vegf-r2 y métodos
US20090124636A1 (en) 2006-04-12 2009-05-14 Pfizer Inc. Chemical compounds
GB0701992D0 (en) 2007-02-02 2007-03-14 7Tm Pharma As Grehlin Receptor Modulators
US8008092B2 (en) 2007-10-09 2011-08-30 University Of Kentucky Research Foundation CCR3 inhibition for ocular angiogenesis and macular degeneration
TW201000446A (en) 2008-05-30 2010-01-01 Astrazeneca Ab New compounds useful in pain therapy
US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
AR090566A1 (es) 2012-04-02 2014-11-19 Boehringer Ingelheim Int Proceso para la produccion de inhibidores de crr
US20130261153A1 (en) 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists

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