JP2015083565A5 - - Google Patents
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- Publication number
- JP2015083565A5 JP2015083565A5 JP2014190339A JP2014190339A JP2015083565A5 JP 2015083565 A5 JP2015083565 A5 JP 2015083565A5 JP 2014190339 A JP2014190339 A JP 2014190339A JP 2014190339 A JP2014190339 A JP 2014190339A JP 2015083565 A5 JP2015083565 A5 JP 2015083565A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutical composition
- treating
- preventing
- disease according
- eye disease
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000008194 pharmaceutical composition Substances 0.000 claims 14
- 208000030533 eye disease Diseases 0.000 claims 13
- 150000001875 compounds Chemical class 0.000 claims 6
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 claims 5
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 claims 5
- 239000002202 Polyethylene glycol Substances 0.000 claims 5
- 125000005843 halogen group Chemical group 0.000 claims 5
- 229920001223 polyethylene glycol Polymers 0.000 claims 5
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 4
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 claims 3
- 150000003839 salts Chemical class 0.000 claims 3
- 208000002158 Proliferative Vitreoretinopathy Diseases 0.000 claims 2
- 206010038934 Retinopathy proliferative Diseases 0.000 claims 2
- 201000010099 disease Diseases 0.000 claims 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims 2
- 125000000350 glycoloyl group Chemical group O=C([*])C([H])([H])O[H] 0.000 claims 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 2
- 208000021971 neovascular inflammatory vitreoretinopathy Diseases 0.000 claims 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 2
- IBBMAWULFFBRKK-UHFFFAOYSA-N picolinamide Chemical compound NC(=O)C1=CC=CC=N1 IBBMAWULFFBRKK-UHFFFAOYSA-N 0.000 claims 2
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims 2
- 230000006785 proliferative vitreoretinopathy Effects 0.000 claims 2
- 125000000446 sulfanediyl group Chemical group *S* 0.000 claims 2
- 125000000876 trifluoromethoxy group Chemical group FC(F)(F)O* 0.000 claims 2
- 206010060823 Choroidal neovascularisation Diseases 0.000 claims 1
- 206010012688 Diabetic retinal oedema Diseases 0.000 claims 1
- 206010012689 Diabetic retinopathy Diseases 0.000 claims 1
- 208000010412 Glaucoma Diseases 0.000 claims 1
- 229920002565 Polyethylene Glycol 400 Polymers 0.000 claims 1
- 206010063381 Polypoidal choroidal vasculopathy Diseases 0.000 claims 1
- 206010064714 Radiation retinopathy Diseases 0.000 claims 1
- 201000007527 Retinal artery occlusion Diseases 0.000 claims 1
- 206010038933 Retinopathy of prematurity Diseases 0.000 claims 1
- 206010064930 age-related macular degeneration Diseases 0.000 claims 1
- 201000011190 diabetic macular edema Diseases 0.000 claims 1
- 208000024519 eye neoplasm Diseases 0.000 claims 1
- 208000002780 macular degeneration Diseases 0.000 claims 1
- 239000000203 mixture Substances 0.000 claims 1
- 201000003142 neovascular glaucoma Diseases 0.000 claims 1
- JLFNLZLINWHATN-UHFFFAOYSA-N pentaethylene glycol Chemical compound OCCOCCOCCOCCOCCO JLFNLZLINWHATN-UHFFFAOYSA-N 0.000 claims 1
- 230000002207 retinal effect Effects 0.000 claims 1
- 208000004644 retinal vein occlusion Diseases 0.000 claims 1
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2014190339A JP5856264B2 (ja) | 2013-09-20 | 2014-09-18 | ポリエチレングリコール含有組成物 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2013195329 | 2013-09-20 | ||
| JP2013195329 | 2013-09-20 | ||
| JP2014190339A JP5856264B2 (ja) | 2013-09-20 | 2014-09-18 | ポリエチレングリコール含有組成物 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015240775A Division JP2016094442A (ja) | 2013-09-20 | 2015-12-10 | ポリエチレングリコール含有組成物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2015083565A JP2015083565A (ja) | 2015-04-30 |
| JP2015083565A5 true JP2015083565A5 (enExample) | 2015-08-20 |
| JP5856264B2 JP5856264B2 (ja) | 2016-02-09 |
Family
ID=52688941
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014190339A Expired - Fee Related JP5856264B2 (ja) | 2013-09-20 | 2014-09-18 | ポリエチレングリコール含有組成物 |
| JP2015240775A Pending JP2016094442A (ja) | 2013-09-20 | 2015-12-10 | ポリエチレングリコール含有組成物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015240775A Pending JP2016094442A (ja) | 2013-09-20 | 2015-12-10 | ポリエチレングリコール含有組成物 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US20160228420A1 (enExample) |
| EP (1) | EP3047850A4 (enExample) |
| JP (2) | JP5856264B2 (enExample) |
| KR (1) | KR20160060656A (enExample) |
| CN (1) | CN105555271A (enExample) |
| AU (1) | AU2014322111A1 (enExample) |
| BR (1) | BR112016006153A2 (enExample) |
| CA (1) | CA2924628A1 (enExample) |
| EA (1) | EA201690621A1 (enExample) |
| HK (2) | HK1221407A1 (enExample) |
| IL (1) | IL244648A0 (enExample) |
| MX (1) | MX2016003566A (enExample) |
| MY (1) | MY163236A (enExample) |
| PH (1) | PH12016500461A1 (enExample) |
| SG (1) | SG11201602020QA (enExample) |
| TW (1) | TW201518291A (enExample) |
| WO (1) | WO2015041294A1 (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102538806B1 (ko) * | 2015-03-17 | 2023-05-31 | 산텐 세이야꾸 가부시키가이샤 | 폴리펩티드를 함유하는 의약 조성물 |
| ES2969514T3 (es) | 2015-03-18 | 2024-05-21 | Santen Pharmaceutical Co Ltd | Composición farmacéutica de liberación sostenida |
| JP2017008047A (ja) * | 2015-06-25 | 2017-01-12 | 参天製薬株式会社 | 注射剤 |
| TWI755356B (zh) * | 2015-07-01 | 2022-02-21 | 日商參天製藥股份有限公司 | 含檸檬酸酯之緩釋劑之用途 |
| CN106902117A (zh) * | 2015-12-23 | 2017-06-30 | 瑞阳(苏州)生物科技有限公司 | 一种预防或治疗脉络膜新生血管形成的药物 |
| JP7018939B2 (ja) * | 2016-09-26 | 2022-02-14 | ルヤン (スーチョウ) バイオロジー サイエンス アンド テクノロジー カンパニー,リミテッド | 眼疾患の治療のための組成物ならびに使用および調製方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA833692B (en) * | 1982-05-28 | 1985-02-27 | Beecham Group Plc | Pharmaceutical formulations |
| JPS59101478A (ja) * | 1982-11-29 | 1984-06-12 | Sunstar Inc | リグスチライドを安定に配合した水系組成物 |
| JPH09110698A (ja) * | 1995-10-19 | 1997-04-28 | Taiho Yakuhin Kogyo Kk | 経口用医薬組成物の製造法 |
| JP4626353B2 (ja) * | 2004-02-17 | 2011-02-09 | 参天製薬株式会社 | 置換又は無置換アミノ基を導入した4−ピリジルアルキルチオ基を有する新規環式化合物 |
| ES2368153T3 (es) * | 2004-02-17 | 2011-11-14 | Santen Pharmaceutical Co., Ltd. | Nuevo compuesto cíclico que presenta un grupo 4-piridilalquiltio que presenta amino (no) sustituido introducido en el mismo. |
| EP1717229B1 (en) | 2004-02-17 | 2011-06-15 | Santen Pharmaceutical Co., Ltd. | Novel cyclic compound having 4-pyridylalkylthio group having (un)substituted amino introduced therein |
| US20060153920A1 (en) * | 2004-09-24 | 2006-07-13 | Ketan Amin | Lyophilized pharmaceutical compositions |
| BRPI0607606B1 (pt) * | 2005-02-09 | 2021-06-22 | Santen Pharmaceutical, Co., Ltd. | Formulação líquida |
| US20070149593A1 (en) | 2005-12-23 | 2007-06-28 | Alcon, Inc. | PHARMACEUTICAL FORMULATION FOR DELIVERY OF RECEPTOR TYROSINE KINASE INHIBITING (RTKi) COMPOUNDS TO THE EYE |
| CN101687042A (zh) | 2007-07-20 | 2010-03-31 | 爱尔康公司 | 用于递送作为受体酪氨酸激酶抑制剂(RTKi)的化合物至眼部的药物制剂 |
| MX2010005685A (es) * | 2007-11-26 | 2010-09-28 | Merial Ltd | Sistemas de solventes para formulaciones de vaciado determinado para combatir parasitos. |
| BRPI1008920A2 (pt) | 2009-03-03 | 2015-08-25 | Alcon Res Ltd | Composição farmacêutica para liberação de compostos inibidores de receptor de tirosina quinase (rtki) para o olho |
| EP2455368B1 (en) * | 2009-07-17 | 2015-09-16 | Santen Pharmaceutical Co., Ltd | 2-[[[2-[(hydroxyacetyl)amino]-4-pyridinyl]methyl]thio]-n-[4-(trifluoromethoxy)phenyl]-3-pyridinecarboxamide benzene- sulfonate, crystals of same, polymorphs thereof, and processes for production thereof |
| DK3158991T3 (da) * | 2010-01-28 | 2021-06-14 | Eagle Pharmaceuticals Inc | Formuleringer af bendamustin |
-
2014
- 2014-09-18 EA EA201690621A patent/EA201690621A1/ru unknown
- 2014-09-18 BR BR112016006153A patent/BR112016006153A2/pt not_active IP Right Cessation
- 2014-09-18 HK HK16109575.6A patent/HK1221407A1/en unknown
- 2014-09-18 WO PCT/JP2014/074698 patent/WO2015041294A1/ja not_active Ceased
- 2014-09-18 KR KR1020167008149A patent/KR20160060656A/ko not_active Withdrawn
- 2014-09-18 MX MX2016003566A patent/MX2016003566A/es unknown
- 2014-09-18 CN CN201480051151.8A patent/CN105555271A/zh active Pending
- 2014-09-18 SG SG11201602020QA patent/SG11201602020QA/en unknown
- 2014-09-18 AU AU2014322111A patent/AU2014322111A1/en not_active Abandoned
- 2014-09-18 HK HK16108793.4A patent/HK1220632A1/zh unknown
- 2014-09-18 US US15/023,207 patent/US20160228420A1/en not_active Abandoned
- 2014-09-18 JP JP2014190339A patent/JP5856264B2/ja not_active Expired - Fee Related
- 2014-09-18 MY MYPI2016000477A patent/MY163236A/en unknown
- 2014-09-18 EP EP14845745.0A patent/EP3047850A4/en active Pending
- 2014-09-18 CA CA2924628A patent/CA2924628A1/en not_active Abandoned
- 2014-09-18 TW TW103132199A patent/TW201518291A/zh unknown
-
2015
- 2015-12-10 JP JP2015240775A patent/JP2016094442A/ja active Pending
-
2016
- 2016-03-09 PH PH12016500461A patent/PH12016500461A1/en unknown
- 2016-03-17 IL IL244648A patent/IL244648A0/en unknown
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