JP2014506582A5 - - Google Patents
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- Publication number
- JP2014506582A5 JP2014506582A5 JP2013554644A JP2013554644A JP2014506582A5 JP 2014506582 A5 JP2014506582 A5 JP 2014506582A5 JP 2013554644 A JP2013554644 A JP 2013554644A JP 2013554644 A JP2013554644 A JP 2013554644A JP 2014506582 A5 JP2014506582 A5 JP 2014506582A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- alkyl
- cycloalkyl
- alkynyl
- alkenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 Cc1ccc(**C2=NC(****3)=C3**2)cc1 Chemical compound Cc1ccc(**C2=NC(****3)=C3**2)cc1 0.000 description 8
- FTTWNYREDCBOSI-UHFFFAOYSA-N CC(Cc1nnc(C(C)=C(C)C)[nH]1)C#CC Chemical compound CC(Cc1nnc(C(C)=C(C)C)[nH]1)C#CC FTTWNYREDCBOSI-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161444602P | 2011-02-18 | 2011-02-18 | |
| US201161444587P | 2011-02-18 | 2011-02-18 | |
| US61/444,602 | 2011-02-18 | ||
| US61/444,587 | 2011-02-18 | ||
| US201161482097P | 2011-05-03 | 2011-05-03 | |
| US201161482106P | 2011-05-03 | 2011-05-03 | |
| US61/482,097 | 2011-05-03 | ||
| US61/482,106 | 2011-05-03 | ||
| PCT/US2012/025685 WO2012112918A1 (en) | 2011-02-18 | 2012-02-17 | Methods for treating diseases of the retina |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2014506582A JP2014506582A (ja) | 2014-03-17 |
| JP2014506582A5 true JP2014506582A5 (enExample) | 2015-04-16 |
| JP6038051B2 JP6038051B2 (ja) | 2016-12-07 |
Family
ID=45787351
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013554644A Expired - Fee Related JP6038051B2 (ja) | 2011-02-18 | 2012-02-17 | 網膜の疾患を治療するための方法 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20120214842A1 (enExample) |
| EP (1) | EP2675456A1 (enExample) |
| JP (1) | JP6038051B2 (enExample) |
| AR (1) | AR085285A1 (enExample) |
| AU (1) | AU2012219288A1 (enExample) |
| CA (1) | CA2827509A1 (enExample) |
| WO (1) | WO2012112918A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9790203B2 (en) | 2012-11-26 | 2017-10-17 | Abbvie Inc. | Inhibitor compounds of phosphodiesterase type 10A |
| FR3008618A1 (fr) * | 2013-07-19 | 2015-01-23 | Univ Paris Curie | Utilisation de composes pour restaurer la reponse a la lumiere des cellules de la retine |
| EP3886854A4 (en) | 2018-11-30 | 2022-07-06 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
| WO2021257863A1 (en) | 2020-06-19 | 2021-12-23 | Incyte Corporation | Pyrrolotriazine compounds as jak2 v617f inhibitors |
| US11691971B2 (en) | 2020-06-19 | 2023-07-04 | Incyte Corporation | Naphthyridinone compounds as JAK2 V617F inhibitors |
| BR112023000047A2 (pt) | 2020-07-02 | 2023-03-14 | Incyte Corp | Compostos de ureia tricíclicos como inibidores da v617f da jak2 |
| WO2022006456A1 (en) | 2020-07-02 | 2022-01-06 | Incyte Corporation | Tricyclic pyridone compounds as jak2 v617f inhibitors |
| US11661422B2 (en) | 2020-08-27 | 2023-05-30 | Incyte Corporation | Tricyclic urea compounds as JAK2 V617F inhibitors |
| WO2022140231A1 (en) | 2020-12-21 | 2022-06-30 | Incyte Corporation | Deazaguaine compounds as jak2 v617f inhibitors |
| AR125273A1 (es) | 2021-02-25 | 2023-07-05 | Incyte Corp | Lactamas espirocíclicas como inhibidores de jak2 v617f |
| KR20240163688A (ko) | 2022-03-17 | 2024-11-19 | 인사이트 코포레이션 | Jak2 v617f 억제제로서의 삼환계 우레아 화합물 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EA012211B1 (ru) | 2005-01-07 | 2009-08-28 | Пфайзер Продактс Инк. | Гетероароматические соединения хинолинов и их применение в качестве ингибиторов pde10 |
| EP1954128A4 (en) * | 2005-11-04 | 2010-09-22 | Merck Sharp & Dohme | DIPHENYLMETHANE DERIVATIVES AS AN INHIBITORS OF THE LEUKOTRIEN BIOSYNTHESIS |
| JP2009535394A (ja) * | 2006-05-02 | 2009-10-01 | ファイザー・プロダクツ・インク | Ｐｄｅ１０阻害剤としての二環式ヘテロアリール化合物 |
| KR100816670B1 (ko) * | 2006-08-18 | 2008-03-27 | 국방과학연구소 | 망막 손상 치료 및 망막 보호하기 위한 메틸렌블루의 용도 |
| PT2125786E (pt) | 2006-12-21 | 2011-04-21 | Pfizer Prod Inc | Sal succinato de 2-((4-(1-metil-4-(piridin-4-il)-1hpirazol- 3-il)fenoxi)metil)quinolina |
| US8349830B2 (en) * | 2009-10-30 | 2013-01-08 | Merck Sharp & Dohme | Aryl aminopyridine PDE10 inhibitors |
-
2012
- 2012-02-16 US US13/398,213 patent/US20120214842A1/en not_active Abandoned
- 2012-02-17 AR ARP120100553A patent/AR085285A1/es not_active Application Discontinuation
- 2012-02-17 AU AU2012219288A patent/AU2012219288A1/en not_active Abandoned
- 2012-02-17 JP JP2013554644A patent/JP6038051B2/ja not_active Expired - Fee Related
- 2012-02-17 EP EP12706981.3A patent/EP2675456A1/en not_active Withdrawn
- 2012-02-17 WO PCT/US2012/025685 patent/WO2012112918A1/en not_active Ceased
- 2012-02-17 CA CA2827509A patent/CA2827509A1/en not_active Abandoned
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