JP6038051B2 - 網膜の疾患を治療するための方法 - Google Patents

網膜の疾患を治療するための方法 Download PDF

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Publication number
JP6038051B2
JP6038051B2 JP2013554644A JP2013554644A JP6038051B2 JP 6038051 B2 JP6038051 B2 JP 6038051B2 JP 2013554644 A JP2013554644 A JP 2013554644A JP 2013554644 A JP2013554644 A JP 2013554644A JP 6038051 B2 JP6038051 B2 JP 6038051B2
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Japan
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alkyl
group
cycloalkyl
hydrogen
alkenyl
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JP2013554644A
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Japanese (ja)
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JP2014506582A (ja
JP2014506582A5 (enExample
Inventor
ジョン イー ドネロ
ジョン イー ドネロ
ロン ヤン
ロン ヤン
ヴェーナ ヴィスワナス
ヴェーナ ヴィスワナス
ベルトラン ルブロン
ベルトラン ルブロン
エリック ボーソレイユ
エリック ボーソレイユ
マテュー ペ パンド
マテュー ペ パンド
ローラン ジ エール デジル
ローラン ジ エール デジル
アンヌ−ソフィー カサグランデ
アンヌ−ソフィー カサグランデ
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Allergan Inc
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Allergan Inc
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2013554644A 2011-02-18 2012-02-17 網膜の疾患を治療するための方法 Expired - Fee Related JP6038051B2 (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US201161444587P 2011-02-18 2011-02-18
US201161444602P 2011-02-18 2011-02-18
US61/444,587 2011-02-18
US61/444,602 2011-02-18
US201161482106P 2011-05-03 2011-05-03
US201161482097P 2011-05-03 2011-05-03
US61/482,106 2011-05-03
US61/482,097 2011-05-03
PCT/US2012/025685 WO2012112918A1 (en) 2011-02-18 2012-02-17 Methods for treating diseases of the retina

Publications (3)

Publication Number Publication Date
JP2014506582A JP2014506582A (ja) 2014-03-17
JP2014506582A5 JP2014506582A5 (enExample) 2015-04-16
JP6038051B2 true JP6038051B2 (ja) 2016-12-07

Family

ID=45787351

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013554644A Expired - Fee Related JP6038051B2 (ja) 2011-02-18 2012-02-17 網膜の疾患を治療するための方法

Country Status (7)

Country Link
US (1) US20120214842A1 (enExample)
EP (1) EP2675456A1 (enExample)
JP (1) JP6038051B2 (enExample)
AR (1) AR085285A1 (enExample)
AU (1) AU2012219288A1 (enExample)
CA (1) CA2827509A1 (enExample)
WO (1) WO2012112918A1 (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9790203B2 (en) 2012-11-26 2017-10-17 Abbvie Inc. Inhibitor compounds of phosphodiesterase type 10A
FR3008618A1 (fr) * 2013-07-19 2015-01-23 Univ Paris Curie Utilisation de composes pour restaurer la reponse a la lumiere des cellules de la retine
EP3886854A4 (en) 2018-11-30 2022-07-06 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
US11691971B2 (en) 2020-06-19 2023-07-04 Incyte Corporation Naphthyridinone compounds as JAK2 V617F inhibitors
WO2021257863A1 (en) 2020-06-19 2021-12-23 Incyte Corporation Pyrrolotriazine compounds as jak2 v617f inhibitors
US11767323B2 (en) 2020-07-02 2023-09-26 Incyte Corporation Tricyclic pyridone compounds as JAK2 V617F inhibitors
LT4175719T (lt) 2020-07-02 2025-08-25 Incyte Corporation Tricikliniai karbamido dariniai kaip jak2 v617f inhibitoriai
US11661422B2 (en) 2020-08-27 2023-05-30 Incyte Corporation Tricyclic urea compounds as JAK2 V617F inhibitors
WO2022140231A1 (en) 2020-12-21 2022-06-30 Incyte Corporation Deazaguaine compounds as jak2 v617f inhibitors
WO2022182839A1 (en) 2021-02-25 2022-09-01 Incyte Corporation Spirocyclic lactams as jak2 v617f inhibitors
UY40188A (es) 2022-03-17 2023-10-13 Incyte Corp Compuestos de urea tricíclica como inhibidores de jak2 v617f

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006072828A2 (en) * 2005-01-07 2006-07-13 Pfizer Products Inc. Heteroaromatic quinoline compounds and their use as pde10 inhibitors
WO2007056210A2 (en) * 2005-11-04 2007-05-18 Merck & Co., Inc. Diphenylmethane derivatives as inhibitors of leukotriene biosynthesis
WO2007129183A2 (en) * 2006-05-02 2007-11-15 Pfizer Products Inc. Bicyclic heteroaryl compounds as pde10 inhibitors
KR100816670B1 (ko) * 2006-08-18 2008-03-27 국방과학연구소 망막 손상 치료 및 망막 보호하기 위한 메틸렌블루의 용도
KR20120043775A (ko) * 2006-12-21 2012-05-04 화이자 프로덕츠 인크. 2-((4-(1-메틸-4-(피리딘-4-일)-1h-피라졸-3-일)페녹시)메틸)퀴놀린의 숙시네이트 염
US8349830B2 (en) * 2009-10-30 2013-01-08 Merck Sharp & Dohme Aryl aminopyridine PDE10 inhibitors

Also Published As

Publication number Publication date
JP2014506582A (ja) 2014-03-17
WO2012112918A1 (en) 2012-08-23
US20120214842A1 (en) 2012-08-23
EP2675456A1 (en) 2013-12-25
AU2012219288A1 (en) 2013-09-05
AR085285A1 (es) 2013-09-18
CA2827509A1 (en) 2012-08-23

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