JP2014005265A5 - - Google Patents
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- Publication number
- JP2014005265A5 JP2014005265A5 JP2012195912A JP2012195912A JP2014005265A5 JP 2014005265 A5 JP2014005265 A5 JP 2014005265A5 JP 2012195912 A JP2012195912 A JP 2012195912A JP 2012195912 A JP2012195912 A JP 2012195912A JP 2014005265 A5 JP2014005265 A5 JP 2014005265A5
- Authority
- JP
- Japan
- Prior art keywords
- cancer
- deuterium
- hydrogen
- compound
- composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261663221P | 2012-06-22 | 2012-06-22 | |
| US61/663,221 | 2012-06-22 | ||
| US201261680885P | 2012-08-08 | 2012-08-08 | |
| US61/680,885 | 2012-08-08 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2014005265A JP2014005265A (ja) | 2014-01-16 |
| JP2014005265A5 true JP2014005265A5 (OSRAM) | 2015-10-01 |
Family
ID=49892488
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012195912A Pending JP2014005265A (ja) | 2012-06-22 | 2012-09-06 | ピラゾール置換アミノ−ヘテロアリール化合物の誘導体 |
Country Status (2)
| Country | Link |
|---|---|
| JP (1) | JP2014005265A (OSRAM) |
| CN (1) | CN103509008A (OSRAM) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103304552B (zh) * | 2012-03-09 | 2016-12-28 | 广东东阳光药业有限公司 | 取代的吡啶化合物及其使用方法和用途 |
| CN104650049B (zh) * | 2013-08-28 | 2018-06-08 | 广东东阳光药业有限公司 | 取代的吡啶化合物及其使用方法和用途 |
| WO2017088784A1 (zh) * | 2015-11-27 | 2017-06-01 | 正大天晴药业集团股份有限公司 | 氘修饰的Brigatinib衍生物、含有该化合物的药物组合物及其用途 |
| WO2017148325A1 (zh) | 2016-03-03 | 2017-09-08 | 深圳市塔吉瑞生物医药有限公司 | 一种大环化合物及包含该化合物的组合物 |
| CN114437058A (zh) * | 2020-10-30 | 2022-05-06 | 珠海宇繁生物科技有限责任公司 | 氘代hpk1激酶抑制剂及其制备方法和应用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AP2373A (en) * | 2004-08-26 | 2012-03-07 | Pfizer | Enantiomerically pure aminoheteroaryl compounds asprotein kinase inhibitors. |
| BRPI0619424B1 (pt) * | 2005-12-05 | 2022-02-08 | Pfizer Products Inc | Uso de inibidores c-met/hgfrs para a fabricação de medicamentos |
| CN101967140A (zh) * | 2010-09-14 | 2011-02-09 | 郑州泰基鸿诺药物科技有限公司 | 氘代克里唑蒂尼及其衍生物、制备方法和应用 |
-
2012
- 2012-09-05 CN CN201210326710.4A patent/CN103509008A/zh active Pending
- 2012-09-06 JP JP2012195912A patent/JP2014005265A/ja active Pending
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