JP2013541592A5 - - Google Patents

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Publication number
JP2013541592A5
JP2013541592A5 JP2013537864A JP2013537864A JP2013541592A5 JP 2013541592 A5 JP2013541592 A5 JP 2013541592A5 JP 2013537864 A JP2013537864 A JP 2013537864A JP 2013537864 A JP2013537864 A JP 2013537864A JP 2013541592 A5 JP2013541592 A5 JP 2013541592A5
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JP
Japan
Prior art keywords
compound
powder
free base
ray diffraction
single crystal
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Pending
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JP2013537864A
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English (en)
Japanese (ja)
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JP2013541592A (ja
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Priority claimed from PCT/US2010/055586 external-priority patent/WO2011057054A1/en
Application filed filed Critical
Priority claimed from PCT/US2011/059331 external-priority patent/WO2012061708A1/en
Publication of JP2013541592A publication Critical patent/JP2013541592A/ja
Publication of JP2013541592A5 publication Critical patent/JP2013541592A5/ja
Pending legal-status Critical Current

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JP2013537864A 2010-11-05 2011-11-04 ヘキサヒドロインデノピリジン及びオクタヒドロベンゾキノリンのアリール−及びヘテロアリールカルボニル誘導体 Pending JP2013541592A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
PCT/US2010/055586 WO2011057054A1 (en) 2009-11-06 2010-11-05 Aryl- and heteroarylcarbonyl derivatives of hexahydroindenopyridine and octahydrobenzoquinoline
USPCT/US2010/055586 2010-11-05
US201161484995P 2011-05-11 2011-05-11
US61/484,995 2011-05-11
PCT/US2011/059331 WO2012061708A1 (en) 2010-11-05 2011-11-04 Crystalline forms of hydrochloride salt of (4a-r,9a-s) -1- (1h - benzoimidazole- 5 -carbonyl) -2, 3, 4, 4a, 9, 9a - hexahydro -1h- indeno [2, 1 -b] pyridine- 6 -carbonitrile and their use as hsd 1 inhibitors

Publications (2)

Publication Number Publication Date
JP2013541592A JP2013541592A (ja) 2013-11-14
JP2013541592A5 true JP2013541592A5 (US07794700-20100914-C00152.png) 2014-11-27

Family

ID=44999935

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013537864A Pending JP2013541592A (ja) 2010-11-05 2011-11-04 ヘキサヒドロインデノピリジン及びオクタヒドロベンゾキノリンのアリール−及びヘテロアリールカルボニル誘導体

Country Status (36)

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US (2) US8686149B2 (US07794700-20100914-C00152.png)
EP (1) EP2635563B1 (US07794700-20100914-C00152.png)
JP (1) JP2013541592A (US07794700-20100914-C00152.png)
KR (1) KR20130119939A (US07794700-20100914-C00152.png)
CN (1) CN103228642B (US07794700-20100914-C00152.png)
AP (1) AP3521A (US07794700-20100914-C00152.png)
AR (1) AR083678A1 (US07794700-20100914-C00152.png)
AU (1) AU2011323164B2 (US07794700-20100914-C00152.png)
BR (1) BR112013011095A2 (US07794700-20100914-C00152.png)
CA (1) CA2816136A1 (US07794700-20100914-C00152.png)
CL (1) CL2013001221A1 (US07794700-20100914-C00152.png)
CO (1) CO6781480A2 (US07794700-20100914-C00152.png)
CY (1) CY1116043T1 (US07794700-20100914-C00152.png)
DK (1) DK2635563T3 (US07794700-20100914-C00152.png)
EA (1) EA022406B1 (US07794700-20100914-C00152.png)
EC (2) ECSP12011788A (US07794700-20100914-C00152.png)
ES (1) ES2533833T3 (US07794700-20100914-C00152.png)
GE (1) GEP20166481B (US07794700-20100914-C00152.png)
HK (1) HK1184144A1 (US07794700-20100914-C00152.png)
HR (1) HRP20150327T1 (US07794700-20100914-C00152.png)
IL (1) IL225647A0 (US07794700-20100914-C00152.png)
ME (1) ME02066B (US07794700-20100914-C00152.png)
MX (1) MX2013005069A (US07794700-20100914-C00152.png)
NZ (1) NZ609281A (US07794700-20100914-C00152.png)
PE (1) PE20140123A1 (US07794700-20100914-C00152.png)
PL (1) PL2635563T3 (US07794700-20100914-C00152.png)
PT (1) PT2635563E (US07794700-20100914-C00152.png)
RS (1) RS53900B1 (US07794700-20100914-C00152.png)
SG (1) SG189859A1 (US07794700-20100914-C00152.png)
SI (1) SI2635563T1 (US07794700-20100914-C00152.png)
SM (1) SMT201500095B (US07794700-20100914-C00152.png)
TN (1) TN2012000117A1 (US07794700-20100914-C00152.png)
TW (1) TWI537258B (US07794700-20100914-C00152.png)
UA (1) UA110807C2 (US07794700-20100914-C00152.png)
UY (1) UY33701A (US07794700-20100914-C00152.png)
WO (1) WO2012061708A1 (US07794700-20100914-C00152.png)

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EP3935050A4 (en) 2019-03-06 2023-01-04 C4 Therapeutics, Inc. HETEROCYCLIC COMPOUNDS FOR MEDICAL TREATMENT

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TWI531571B (zh) * 2009-11-06 2016-05-01 維它藥物公司 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜芳基羰基衍生物
TWI537258B (zh) 2010-11-05 2016-06-11 百靈佳殷格翰國際股份有限公司 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜環芳基羰基衍生物

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