JP2013536251A - 薬学的組成物およびその投与 - Google Patents

薬学的組成物およびその投与 Download PDF

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JP2013536251A
JP2013536251A JP2013526195A JP2013526195A JP2013536251A JP 2013536251 A JP2013536251 A JP 2013536251A JP 2013526195 A JP2013526195 A JP 2013526195A JP 2013526195 A JP2013526195 A JP 2013526195A JP 2013536251 A JP2013536251 A JP 2013536251A
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pharmaceutical composition
weight
compound
composition
solid dispersion
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JP2013536251A5 (https=
Inventor
エレニ ドコウ，
シャーラ ジャムザッド，
ラウラ ダス，
メグナ ジャイ イスラニ，
ドラグティン ネジック，
アンドリュー ジー． クズミッション，
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Vertex Pharmaceuticals Inc
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Vertex Pharmaceuticals Inc
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Publication of JP2013536251A publication Critical patent/JP2013536251A/ja
Publication of JP2013536251A5 publication Critical patent/JP2013536251A5/ja
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  • Organic Chemistry (AREA)
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  • Diabetes (AREA)
  • Biomedical Technology (AREA)
  • Hematology (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Psychology (AREA)
  • Reproductive Health (AREA)
  • Inorganic Chemistry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Hospice & Palliative Care (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
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JP2013526195A 2010-08-27 2011-08-26 薬学的組成物およびその投与 Pending JP2013536251A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US37787310P 2010-08-27 2010-08-27
US61/377,873 2010-08-27
PCT/US2011/049467 WO2012027731A2 (en) 2010-08-27 2011-08-26 Pharmaceutical composition and administrations thereof

Publications (2)

Publication Number Publication Date
JP2013536251A true JP2013536251A (ja) 2013-09-19
JP2013536251A5 JP2013536251A5 (https=) 2014-10-16

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JP2013526195A Pending JP2013536251A (ja) 2010-08-27 2011-08-26 薬学的組成物およびその投与

Country Status (12)

Country Link
US (2) US20120064157A1 (https=)
EP (1) EP2608775A2 (https=)
JP (1) JP2013536251A (https=)
CN (1) CN103153286A (https=)
AU (1) AU2011293135A1 (https=)
BR (1) BR112013004130A2 (https=)
CA (1) CA2809263A1 (https=)
MX (1) MX2013002353A (https=)
NZ (1) NZ607494A (https=)
RU (1) RU2013113627A (https=)
WO (1) WO2012027731A2 (https=)
ZA (1) ZA201301419B (https=)

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2017190356A (ja) * 2012-02-27 2017-10-19 バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ 薬学的組成物およびその投与
JP2018516900A (ja) * 2015-06-09 2018-06-28 カプスゲル・ベルギウム・ナムローゼ・フェンノートシャップＣａｐｓｕｇｅｌ Ｂｅｌｇｉｕｍ ＮＶ カプセル中の薬剤の噴霧乾燥ディスパーションからの迅速な溶解を達成するための製剤
WO2020032227A1 (ja) * 2018-08-10 2020-02-13 キッセイ薬品工業株式会社 スクロオキシ水酸化鉄含有顆粒及び医薬組成物
US10894058B2 (en) 2014-08-29 2021-01-19 Kao Corporation Method for producing solid dispersion containing hardly soluble polyphenol
JP2021512117A (ja) * 2018-02-05 2021-05-13 バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ 嚢胞性線維症を処置するための医薬組成物
JP2024511188A (ja) * 2021-03-26 2024-03-12 上海瑛派▲薬▼▲業▼有限公司 Ｐａｒｐ阻害剤の経口カプセルおよびその調製方法
WO2025105451A1 (ja) * 2023-11-17 2025-05-22 第一三共ヘルスケア株式会社 固形製剤

Families Citing this family (103)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2006111093A (ru) 2003-09-06 2007-10-27 Вертекс Фармасьютикалз Инкорпорейтед (Us) Модуляторы атр-связывающих кассетных транспортеров
US7977322B2 (en) 2004-08-20 2011-07-12 Vertex Pharmaceuticals Incorporated Modulators of ATP-binding cassette transporters
RS56037B1 (sr) 2004-06-24 2017-09-29 Vertex Pharma Modulatori atp-vezujućih kasetnih transportera
US7999113B2 (en) 2005-08-11 2011-08-16 Vertex Pharmaceuticals Incorporated Modulators of cystic fibrosis transmembrane conductance regulator
CN102775396B (zh) * 2005-11-08 2014-10-08 沃泰克斯药物股份有限公司 Atp-结合弹夹转运蛋白的杂环调控剂
CA2856037C (en) 2005-12-28 2017-03-07 Vertex Pharmaceuticals Incorporated Modulators of atp-binding cassette transporters
EP3219705B1 (en) 2005-12-28 2020-03-11 Vertex Pharmaceuticals Incorporated Pharmaceutical compositions of the amorphous form of n-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide
EP2674428B1 (en) 2006-04-07 2016-04-06 Vertex Pharmaceuticals Incorporated Modulators of ATP-binding cassette transporters
US7645789B2 (en) 2006-04-07 2010-01-12 Vertex Pharmaceuticals Incorporated Indole derivatives as CFTR modulators
USRE50453E1 (en) 2006-04-07 2025-06-10 Vertex Pharmaceuticals Incorporated Indole derivatives as CFTR modulators
US10022352B2 (en) 2006-04-07 2018-07-17 Vertex Pharmaceuticals Incorporated Modulators of ATP-binding cassette transporters
US8563573B2 (en) 2007-11-02 2013-10-22 Vertex Pharmaceuticals Incorporated Azaindole derivatives as CFTR modulators
CN104447716A (zh) 2007-05-09 2015-03-25 沃泰克斯药物股份有限公司 Cftr调节剂
JP5389030B2 (ja) 2007-08-24 2014-01-15 バーテックス ファーマシューティカルズ インコーポレイテッド （特に）嚢胞性線維症の処置に有用なイソチアゾロピリジノン
SI2578571T1 (sl) 2007-11-16 2016-01-29 Vertex Pharmaceuticals Incorporated Izokinolinski modulatorji prenašalcev z atp-vezavno kaseto
EP3683218B1 (en) 2007-12-07 2024-09-18 Vertex Pharmaceuticals Incorporated Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl) benzoic acid
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