JP2013532651A - シロドシンと塩基性コポリマーとの混合物を含む経口投与用医薬品 - Google Patents
シロドシンと塩基性コポリマーとの混合物を含む経口投与用医薬品 Download PDFInfo
- Publication number
- JP2013532651A JP2013532651A JP2013520157A JP2013520157A JP2013532651A JP 2013532651 A JP2013532651 A JP 2013532651A JP 2013520157 A JP2013520157 A JP 2013520157A JP 2013520157 A JP2013520157 A JP 2013520157A JP 2013532651 A JP2013532651 A JP 2013532651A
- Authority
- JP
- Japan
- Prior art keywords
- silodosin
- pharmaceutically acceptable
- copolymer
- pharmaceutical product
- present
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1682—Processes
- A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Urology & Nephrology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10170649.7 | 2010-07-23 | ||
EP10170649 | 2010-07-23 | ||
PCT/EP2011/062566 WO2012010669A2 (de) | 2010-07-23 | 2011-07-21 | Arzneimittel zur oralen verabreichung umfassend ein gemisch aus silodosin und einem basischen copolymer |
Publications (1)
Publication Number | Publication Date |
---|---|
JP2013532651A true JP2013532651A (ja) | 2013-08-19 |
Family
ID=44628851
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2013520157A Withdrawn JP2013532651A (ja) | 2010-07-23 | 2011-07-21 | シロドシンと塩基性コポリマーとの混合物を含む経口投与用医薬品 |
Country Status (3)
Country | Link |
---|---|
EP (1) | EP2595607A2 (de) |
JP (1) | JP2013532651A (de) |
WO (1) | WO2012010669A2 (de) |
Cited By (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2016051782A1 (ja) * | 2014-09-30 | 2016-04-07 | キッセイ薬品工業株式会社 | 苦味を有する薬剤の苦味をマスキングした経口投与製剤 |
JP2016138073A (ja) * | 2015-01-29 | 2016-08-04 | 大原薬品工業株式会社 | 安定性を改善した、シロドシンを含有する錠剤 |
JP2017014119A (ja) * | 2015-06-26 | 2017-01-19 | 東和薬品株式会社 | 経口医薬組成物 |
JP2018065752A (ja) * | 2016-10-17 | 2018-04-26 | 東和薬品株式会社 | シロドシン含有医薬組成物とその製造方法 |
JP2018199699A (ja) * | 2013-03-26 | 2018-12-20 | キッセイ薬品工業株式会社 | シロドシンの苦味をマスキングした経口投与製剤 |
JP2019070045A (ja) * | 2019-02-06 | 2019-05-09 | 大原薬品工業株式会社 | 安定性を改善した、シロドシンを含有する錠剤 |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013061338A1 (en) * | 2011-08-24 | 2013-05-02 | Cadila Healthcare Limited | Pharmaceutical compositions of silodosin |
EP2866793A4 (de) * | 2012-07-02 | 2016-07-27 | Hetero Research Foundation | Feste orale zusammensetzungen aus silodosin |
KR102206104B1 (ko) * | 2014-04-03 | 2021-01-22 | 한미약품 주식회사 | 실로도신을 포함하는 과립물, 및 이를 포함하는 약학적 조성물 및 제형 |
EP3354283B1 (de) | 2017-06-20 | 2019-08-07 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Pharmazeutische kapselzusammensetzung mit silodosin |
CN112933084A (zh) * | 2019-12-10 | 2021-06-11 | 广东东阳光药业有限公司 | 一种赛洛多辛组合物 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0600675B1 (de) | 1992-12-02 | 1998-07-08 | Kissei Pharmaceutical Co., Ltd. | Indolin Verbindungen zur Behandlung von Dysurien |
DE19653605C2 (de) | 1996-12-20 | 2002-11-28 | Roehm Gmbh | Haft- und Bindemittel für dermale oder transdermale Therapiesysteme und dessen Verwendung zur Herstellung eines transdermalen Therapiesystems |
JP4324266B2 (ja) * | 1999-02-26 | 2009-09-02 | キッセイ薬品工業株式会社 | α1Aアドレナリン受容体の変異体、当該変異体を用いた測定方法及び前立腺肥大に伴う排尿困難症治療剤 |
UA78854C2 (en) | 2002-09-06 | 2007-04-25 | Kissei Pharmaceutical | Crystal for an oral solid drug and oral solid drug for dysuria treatment containing the same |
JP4523265B2 (ja) | 2002-11-13 | 2010-08-11 | 旭化成ファーマ株式会社 | 排尿障害治療用口腔内崩壊製剤 |
EP1574215B1 (de) * | 2002-12-16 | 2015-07-15 | Kissei Pharmaceutical Co., Ltd. | Feste arznei zur oralen verabreichung |
US20060013880A1 (en) * | 2004-07-19 | 2006-01-19 | Robert Femia | Formulation stabilizer for proton pump inhibitors |
-
2011
- 2011-07-21 WO PCT/EP2011/062566 patent/WO2012010669A2/de active Application Filing
- 2011-07-21 JP JP2013520157A patent/JP2013532651A/ja not_active Withdrawn
- 2011-07-21 EP EP11735435.7A patent/EP2595607A2/de not_active Withdrawn
Cited By (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2018199699A (ja) * | 2013-03-26 | 2018-12-20 | キッセイ薬品工業株式会社 | シロドシンの苦味をマスキングした経口投与製剤 |
WO2016051782A1 (ja) * | 2014-09-30 | 2016-04-07 | キッセイ薬品工業株式会社 | 苦味を有する薬剤の苦味をマスキングした経口投与製剤 |
JPWO2016051782A1 (ja) * | 2014-09-30 | 2017-07-13 | キッセイ薬品工業株式会社 | 苦味を有する薬剤の苦味をマスキングした経口投与製剤 |
JP2016138073A (ja) * | 2015-01-29 | 2016-08-04 | 大原薬品工業株式会社 | 安定性を改善した、シロドシンを含有する錠剤 |
JP2017014119A (ja) * | 2015-06-26 | 2017-01-19 | 東和薬品株式会社 | 経口医薬組成物 |
JP2018065752A (ja) * | 2016-10-17 | 2018-04-26 | 東和薬品株式会社 | シロドシン含有医薬組成物とその製造方法 |
JP7023600B2 (ja) | 2016-10-17 | 2022-02-22 | 東和薬品株式会社 | シロドシン含有医薬組成物とその製造方法 |
JP2019070045A (ja) * | 2019-02-06 | 2019-05-09 | 大原薬品工業株式会社 | 安定性を改善した、シロドシンを含有する錠剤 |
Also Published As
Publication number | Publication date |
---|---|
WO2012010669A3 (de) | 2012-07-26 |
WO2012010669A2 (de) | 2012-01-26 |
EP2595607A2 (de) | 2013-05-29 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
JP2013532651A (ja) | シロドシンと塩基性コポリマーとの混合物を含む経口投与用医薬品 | |
RU2404775C2 (ru) | Фармацевтические композиции, содержащие иматиниб и замедлитель высвобождения | |
TWI478712B (zh) | 釋控性醫藥組成物 | |
TW201904565A (zh) | 控釋藥物組合物及其製備方法 | |
JP2005517690A (ja) | 固体薬物分散物を含有する即時放出剤形 | |
CA2729979A1 (en) | Pharmaceutical compositions comprising 5-chloro-n-({(5s)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid | |
CN106232144B (zh) | 固体分散体 | |
TW200848056A (en) | Solid dispersion of a neurokinin antagonist | |
JP5714562B2 (ja) | 経口用徐放性固形製剤 | |
JP2010519200A (ja) | シロスタゾールを含む制御放出製剤及びその製造方法 | |
JP2023513444A (ja) | ダサチニブの非晶質固体分散体及びその使用 | |
US20140319720A1 (en) | Pharmaceutical compositions comprising rivaroxaban | |
JP2016117738A (ja) | シロドシン−シクロデキストリン包接化合物 | |
EP2701689B1 (de) | Pharmazeutische zusammensetzungen aus raltegravir sowie verfahren zu ihrer herstellung und verwendung | |
JPWO2008114859A1 (ja) | ピラゾール誘導体を含有する医薬組成物 | |
TW201609195A (zh) | 固體抗病毒劑型 | |
JP6680297B2 (ja) | 経口投与用医薬組成物 | |
CA2934586A1 (en) | Pharmaceutical composition | |
US20230147712A1 (en) | Oleyl phosphocholine containing granulates | |
JP5669751B2 (ja) | 低い経口生物学的利用能を有する化合物のプレ圧縮崩壊性製剤 | |
JP2022113667A (ja) | エドキサバン含有医薬組成物 | |
WO2019004980A2 (en) | SOLID ORAL PHARMACEUTICAL COMPOSITIONS OF DABIGATRAN DEXILATE | |
WO2022177983A1 (en) | Pharmaceutical compositions of cabozantinib | |
EP4279075A1 (de) | Pharmazeutische zusammensetzung enthaltend elagolix | |
RU2696870C2 (ru) | Пероральный препарат с замедленным высвобождением |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
A521 | Written amendment |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20130517 |
|
A300 | Withdrawal of application because of no request for examination |
Free format text: JAPANESE INTERMEDIATE CODE: A300 Effective date: 20141007 |