WO2012010669A3 - Arzneimittel zur oralen verabreichung umfassend ein gemisch aus silodosin und einem basischen copolymer - Google Patents
Arzneimittel zur oralen verabreichung umfassend ein gemisch aus silodosin und einem basischen copolymer Download PDFInfo
- Publication number
- WO2012010669A3 WO2012010669A3 PCT/EP2011/062566 EP2011062566W WO2012010669A3 WO 2012010669 A3 WO2012010669 A3 WO 2012010669A3 EP 2011062566 W EP2011062566 W EP 2011062566W WO 2012010669 A3 WO2012010669 A3 WO 2012010669A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- silodosin
- mixture
- oral administration
- medicinal drug
- basic copolymer
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1682—Processes
- A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Die Erfindung betrifft ein Arzneimittel zur oralen Verabreichung umfassend ein Gemisch aus Silodosin bzw. einem pharmazeutisch verträglichen Salz davon und einem basischen Copolymer. Des Weiteren betrifft die vorliegende Erfindung ein Verfahren zur Herstellung dieses Arzneimittels.
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP11735435.7A EP2595607A2 (de) | 2010-07-23 | 2011-07-21 | Arzneimittel zur oralen verabreichung umfassend ein gemisch aus silodosin und einem basischen copolymer |
JP2013520157A JP2013532651A (ja) | 2010-07-23 | 2011-07-21 | シロドシンと塩基性コポリマーとの混合物を含む経口投与用医薬品 |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10170649.7 | 2010-07-23 | ||
EP10170649 | 2010-07-23 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2012010669A2 WO2012010669A2 (de) | 2012-01-26 |
WO2012010669A3 true WO2012010669A3 (de) | 2012-07-26 |
Family
ID=44628851
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/EP2011/062566 WO2012010669A2 (de) | 2010-07-23 | 2011-07-21 | Arzneimittel zur oralen verabreichung umfassend ein gemisch aus silodosin und einem basischen copolymer |
Country Status (3)
Country | Link |
---|---|
EP (1) | EP2595607A2 (de) |
JP (1) | JP2013532651A (de) |
WO (1) | WO2012010669A2 (de) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013061338A1 (en) * | 2011-08-24 | 2013-05-02 | Cadila Healthcare Limited | Pharmaceutical compositions of silodosin |
WO2014006635A2 (en) * | 2012-07-02 | 2014-01-09 | Hetero Research Foundation | Solid oral compositions of silodosin |
CN105142633A (zh) * | 2013-03-26 | 2015-12-09 | 橘生药品工业株式会社 | 西洛多辛苦味被掩蔽的口服给药制剂 |
KR102206104B1 (ko) * | 2014-04-03 | 2021-01-22 | 한미약품 주식회사 | 실로도신을 포함하는 과립물, 및 이를 포함하는 약학적 조성물 및 제형 |
WO2016051782A1 (ja) * | 2014-09-30 | 2016-04-07 | キッセイ薬品工業株式会社 | 苦味を有する薬剤の苦味をマスキングした経口投与製剤 |
JP2016138073A (ja) * | 2015-01-29 | 2016-08-04 | 大原薬品工業株式会社 | 安定性を改善した、シロドシンを含有する錠剤 |
JP2017014119A (ja) * | 2015-06-26 | 2017-01-19 | 東和薬品株式会社 | 経口医薬組成物 |
JP7023600B2 (ja) * | 2016-10-17 | 2022-02-22 | 東和薬品株式会社 | シロドシン含有医薬組成物とその製造方法 |
EP3354283B1 (de) | 2017-06-20 | 2019-08-07 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Pharmazeutische kapselzusammensetzung mit silodosin |
JP2019070045A (ja) * | 2019-02-06 | 2019-05-09 | 大原薬品工業株式会社 | 安定性を改善した、シロドシンを含有する錠剤 |
CN112933084A (zh) * | 2019-12-10 | 2021-06-11 | 广东东阳光药业有限公司 | 一种赛洛多辛组合物 |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1574215A1 (de) * | 2002-12-16 | 2005-09-14 | Kissei Pharmaceutical Co., Ltd. | Feste arznei zur oralen verabreichung |
WO2006020111A1 (en) * | 2004-07-19 | 2006-02-23 | Par Pharmaceutical, Inc. | Formulation stabilizer for proton pump inhibitors |
JP4324266B2 (ja) * | 1999-02-26 | 2009-09-02 | キッセイ薬品工業株式会社 | α1Aアドレナリン受容体の変異体、当該変異体を用いた測定方法及び前立腺肥大に伴う排尿困難症治療剤 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69319551T2 (de) | 1992-12-02 | 1998-10-29 | Kissei Pharmaceutical | Indolin Verbindungen zur Behandlung von Dysurien |
DE19653605C2 (de) | 1996-12-20 | 2002-11-28 | Roehm Gmbh | Haft- und Bindemittel für dermale oder transdermale Therapiesysteme und dessen Verwendung zur Herstellung eines transdermalen Therapiesystems |
UA78854C2 (en) | 2002-09-06 | 2007-04-25 | Kissei Pharmaceutical | Crystal for an oral solid drug and oral solid drug for dysuria treatment containing the same |
JP4523265B2 (ja) | 2002-11-13 | 2010-08-11 | 旭化成ファーマ株式会社 | 排尿障害治療用口腔内崩壊製剤 |
-
2011
- 2011-07-21 JP JP2013520157A patent/JP2013532651A/ja not_active Withdrawn
- 2011-07-21 WO PCT/EP2011/062566 patent/WO2012010669A2/de active Application Filing
- 2011-07-21 EP EP11735435.7A patent/EP2595607A2/de not_active Withdrawn
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP4324266B2 (ja) * | 1999-02-26 | 2009-09-02 | キッセイ薬品工業株式会社 | α1Aアドレナリン受容体の変異体、当該変異体を用いた測定方法及び前立腺肥大に伴う排尿困難症治療剤 |
EP1574215A1 (de) * | 2002-12-16 | 2005-09-14 | Kissei Pharmaceutical Co., Ltd. | Feste arznei zur oralen verabreichung |
WO2006020111A1 (en) * | 2004-07-19 | 2006-02-23 | Par Pharmaceutical, Inc. | Formulation stabilizer for proton pump inhibitors |
Also Published As
Publication number | Publication date |
---|---|
JP2013532651A (ja) | 2013-08-19 |
EP2595607A2 (de) | 2013-05-29 |
WO2012010669A2 (de) | 2012-01-26 |
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