JP2013525265A5 - - Google Patents
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- Publication number
- JP2013525265A5 JP2013525265A5 JP2012549044A JP2012549044A JP2013525265A5 JP 2013525265 A5 JP2013525265 A5 JP 2013525265A5 JP 2012549044 A JP2012549044 A JP 2012549044A JP 2012549044 A JP2012549044 A JP 2012549044A JP 2013525265 A5 JP2013525265 A5 JP 2013525265A5
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- JP
- Japan
- Prior art keywords
- group
- formula
- production method
- manufacturing
- compound represented
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 0 C1*CCNC1 Chemical compound C1*CCNC1 0.000 description 6
- KRDOFMHJLWKXIU-UHFFFAOYSA-N C(C1)NCCN1c1n[s]c2ccccc12 Chemical compound C(C1)NCCN1c1n[s]c2ccccc12 KRDOFMHJLWKXIU-UHFFFAOYSA-N 0.000 description 1
- YZDLKGSISFGIRU-UHFFFAOYSA-N C(C1C(C2)CCCC1)[N]2(CC1)CCN1c1n[s]c2ccccc12 Chemical compound C(C1C(C2)CCCC1)[N]2(CC1)CCN1c1n[s]c2ccccc12 YZDLKGSISFGIRU-UHFFFAOYSA-N 0.000 description 1
- RIVOBMOBWMOLDJ-UHFFFAOYSA-N O=C(C1C2C3CC1CC3)NC2=O Chemical compound O=C(C1C2C3CC1CC3)NC2=O RIVOBMOBWMOLDJ-UHFFFAOYSA-N 0.000 description 1
- RIVOBMOBWMOLDJ-RNGGSSJXSA-N O=C([C@H]1[C@@H]2[C@H]3C[C@@H]1CC3)NC2=O Chemical compound O=C([C@H]1[C@@H]2[C@H]3C[C@@H]1CC3)NC2=O RIVOBMOBWMOLDJ-RNGGSSJXSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US32780410P | 2010-04-26 | 2010-04-26 | |
| US61/327,804 | 2010-04-26 | ||
| PCT/JP2011/060571 WO2011136384A1 (en) | 2010-04-26 | 2011-04-25 | A process of a quaternary ammonium salt using phosphate |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013525265A JP2013525265A (ja) | 2013-06-20 |
| JP2013525265A5 true JP2013525265A5 (https=) | 2014-05-22 |
| JP5820822B2 JP5820822B2 (ja) | 2015-11-24 |
Family
ID=44816341
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012549044A Active JP5820822B2 (ja) | 2010-04-26 | 2011-04-25 | リン酸塩を用いる第四級アンモニウム塩の製造法 |
Country Status (5)
| Country | Link |
|---|---|
| US (2) | US8586737B2 (https=) |
| EP (1) | EP2563791B1 (https=) |
| JP (1) | JP5820822B2 (https=) |
| ES (1) | ES2527545T3 (https=) |
| WO (1) | WO2011136384A1 (https=) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2594709T3 (es) * | 2010-04-26 | 2016-12-22 | Sumitomo Dainippon Pharma Co., Ltd. | Un proceso de preparación de una sal de amonio cuaternario |
| JP5820822B2 (ja) * | 2010-04-26 | 2015-11-24 | 大日本住友製薬株式会社 | リン酸塩を用いる第四級アンモニウム塩の製造法 |
| US9409899B2 (en) | 2012-02-13 | 2016-08-09 | Cadila Healthcare Limited | Process for preparing benzisothiazol-3-yl-piperazin-1-yl-methyl-cyclo hexylmethanisoindol-1,3-dione and its intermediates |
| CN102746289B (zh) * | 2012-04-28 | 2016-06-08 | 上海医药工业研究院 | 一种盐酸卢拉西酮的制备方法 |
| CN103450172A (zh) * | 2012-05-30 | 2013-12-18 | 广州药源生物医药科技有限公司 | 一种抗精神病药物鲁拉西酮的制备方法 |
| CN102863437A (zh) * | 2012-09-04 | 2013-01-09 | 济南百诺医药科技开发有限公司 | 一种鲁拉西酮的制备方法 |
| CN103864774B (zh) * | 2012-12-14 | 2016-09-28 | 成都弘达药业有限公司 | 一种鲁拉西酮的制备方法 |
| ITMI20130262A1 (it) * | 2013-02-22 | 2014-08-23 | Edmond Pharma Srl | Procedimento per la preparazione di lurasidone cloridrato |
| ITMI20131245A1 (it) * | 2013-07-24 | 2015-01-25 | Olon Spa | Procedimento per la produzione di lurasidone ad elevata purezza |
| ITMI20131737A1 (it) | 2013-10-17 | 2015-04-18 | Procos Spa | Processo per la sintesi industriale di lurasidone |
| JP6594351B2 (ja) | 2014-06-16 | 2019-10-23 | ジョンソン、マッセイ、パブリック、リミテッド、カンパニー | 新規中間体を含むアルキル化アリールピペラジン及びアルキル化アリールピペリジン化合物の製造方法 |
| US10426770B2 (en) | 2014-10-14 | 2019-10-01 | Jubilant Generics Limited | Process for the preparation of Lurasidone hydrochloride |
| EP3242876A4 (en) * | 2015-01-08 | 2019-01-02 | Piramal Enterprises Limited | An improved process for the preparation of lurasidone and its intermediate |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4351939A (en) * | 1980-10-16 | 1982-09-28 | Mead Johnson & Company | Spiro-quaternary ammonium halides and N-(2-pyrimidinyl)piperazinylalkylazaspiroalkanedione process |
| JP2800953B2 (ja) * | 1990-07-06 | 1998-09-21 | 住友製薬株式会社 | 新規なイミド誘導体 |
| FR2665161B1 (fr) * | 1990-07-26 | 1992-11-27 | Esteve Labor Dr | Nouveaux derives de benzimidazole, leur preparation et leur application en tant que medicaments. |
| JP3775823B2 (ja) * | 1995-06-09 | 2006-05-17 | 大日本住友製薬株式会社 | 新規なイミド誘導体 |
| JP4175800B2 (ja) * | 2001-11-27 | 2008-11-05 | 住友化学株式会社 | イミド誘導体の製造方法 |
| JP2006169154A (ja) * | 2004-12-15 | 2006-06-29 | Sumitomo Chemical Co Ltd | 第四級アンモニウム塩の製造方法 |
| JP4708012B2 (ja) * | 2004-12-15 | 2011-06-22 | 大日本住友製薬株式会社 | 第四級アンモニウム塩の製造法 |
| EP1919922B1 (en) * | 2005-08-30 | 2011-04-20 | Honeywell International Inc. | Method for synthesizing spiro quaternary ammonium systems |
| US20110003994A1 (en) * | 2009-07-02 | 2011-01-06 | Dainippon Sumitomo Pharma Co., Ltd. | Cycloalkane derivative |
| JP5820822B2 (ja) * | 2010-04-26 | 2015-11-24 | 大日本住友製薬株式会社 | リン酸塩を用いる第四級アンモニウム塩の製造法 |
| ES2594709T3 (es) | 2010-04-26 | 2016-12-22 | Sumitomo Dainippon Pharma Co., Ltd. | Un proceso de preparación de una sal de amonio cuaternario |
-
2011
- 2011-04-25 JP JP2012549044A patent/JP5820822B2/ja active Active
- 2011-04-25 EP EP11775165.1A patent/EP2563791B1/en active Active
- 2011-04-25 WO PCT/JP2011/060571 patent/WO2011136384A1/en not_active Ceased
- 2011-04-25 ES ES11775165.1T patent/ES2527545T3/es active Active
- 2011-04-26 US US13/093,985 patent/US8586737B2/en active Active
-
2013
- 2013-09-30 US US14/041,657 patent/US20140031548A1/en not_active Abandoned
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