|
JP5995728B2
(ja)
*
|
2010-03-04 |
2016-09-21 |
メルク・シャープ・エンド・ドーム・コーポレイション |
カテコールo−メチルトランスフェラーゼの阻害剤および精神障害の治療におけるその使用
|
|
GB201111704D0
(en)
|
2011-07-07 |
2011-08-24 |
Takeda Pharmaceutical |
Novel compounds
|
|
GB201111705D0
(en)
|
2011-07-07 |
2011-08-24 |
Takeda Pharmaceutical |
Compounds and their use
|
|
JO3115B1
(ar)
|
2011-08-22 |
2017-09-20 |
Takeda Pharmaceuticals Co |
مركبات بيريدازينون واستخدامها كمثبطات daao
|
|
UA111861C2
(uk)
|
2011-11-15 |
2016-06-24 |
Такеда Фармасьютікал Компані Лімітед |
Ароматична гетероциклічна сполука дигідрокси
|
|
TWI638802B
(zh)
*
|
2012-05-24 |
2018-10-21 |
芬蘭商奧利安公司 |
兒茶酚o-甲基轉移酶活性抑制化合物
|
|
CN103845317B
(zh)
*
|
2012-11-28 |
2018-05-08 |
北京生命科学研究所 |
恩他卡朋在预防或治疗肥胖等代谢综合征中的应用
|
|
GB201222711D0
(en)
|
2012-12-17 |
2013-01-30 |
Takeda Pharmaceutical |
Novel compounds
|
|
MX2015006437A
(es)
*
|
2012-12-27 |
2015-08-14 |
Hoffmann La Roche |
Inhibidores de la enzima catecol-o-metiltransferasa (comt).
|
|
WO2014151367A1
(en)
|
2013-03-15 |
2014-09-25 |
Janssen Pharmaceutica Nv |
1,2,5-substituted benzimidazoles as flap modulators
|
|
US9695149B2
(en)
|
2013-03-15 |
2017-07-04 |
Janssen Pharmaceutica Nv |
1,2,6-substituted benzimidazoles as flap modulators
|
|
CN103588702B
(zh)
*
|
2013-10-26 |
2016-01-06 |
浙江大学 |
N-取代苯基吡啶-4-酮衍生物及其制备和应用
|
|
WO2015099107A1
(ja)
|
2013-12-26 |
2015-07-02 |
塩野義製薬株式会社 |
含窒素6員環誘導体およびそれらを含有する医薬組成物
|
|
JP6858712B2
(ja)
|
2015-01-30 |
2021-04-14 |
リーバー インスティテュート フォー ブレイン ディベロップメントLieber Institute For Brain Development |
Comt阻害方法及び組成物
|
|
JP6358639B2
(ja)
|
2015-04-24 |
2018-07-18 |
塩野義製薬株式会社 |
6員複素環誘導体およびそれらを含有する医薬組成物
|
|
US20170107216A1
(en)
|
2015-10-19 |
2017-04-20 |
Incyte Corporation |
Heterocyclic compounds as immunomodulators
|
|
AU2016358100B2
(en)
|
2015-11-19 |
2021-05-27 |
Incyte Corporation |
Heterocyclic compounds as immunomodulators
|
|
PL3380471T3
(pl)
|
2015-11-25 |
2021-12-20 |
Lieber Institute Inc. Dba Lieber Institute For Brain Development |
Tetrahydro-8h-pirydo[1,2-a]pirazyn-8-ony jako inhibitory comt do leczenia chorób i zaburzeń neurodegeneracyjnych
|
|
CN105481812B
(zh)
*
|
2015-11-30 |
2020-04-21 |
重庆天奕恒化科技有限公司 |
一种5-苄氧基-4-氧代-4h-吡喃-2-羧酸的制备方法
|
|
TW201726623A
(zh)
|
2015-12-17 |
2017-08-01 |
英塞特公司 |
作為免疫調節劑之雜環化合物
|
|
TWI850624B
(zh)
|
2015-12-22 |
2024-08-01 |
美商英塞特公司 |
作為免疫調節劑之雜環化合物
|
|
TW201808950A
(zh)
|
2016-05-06 |
2018-03-16 |
英塞特公司 |
作為免疫調節劑之雜環化合物
|
|
US20170342060A1
(en)
|
2016-05-26 |
2017-11-30 |
Incyte Corporation |
Heterocyclic compounds as immunomodulators
|
|
DK3472167T3
(da)
|
2016-06-20 |
2022-09-05 |
Incyte Corp |
Heterocykliske forbindelser som immunomodulatorer
|
|
EP3484866B1
(en)
|
2016-07-14 |
2022-09-07 |
Incyte Corporation |
Heterocyclic compounds as immunomodulators
|
|
EP3504198B1
(en)
|
2016-08-29 |
2023-01-25 |
Incyte Corporation |
Heterocyclic compounds as immunomodulators
|
|
MX393004B
(es)
|
2016-10-17 |
2025-03-24 |
Shionogi & Co |
Derivado heterociclico nitrogenado biciclico y composicion farmaceutica que lo contiene.
|
|
EP3558963B1
(en)
|
2016-12-22 |
2022-03-23 |
Incyte Corporation |
Bicyclic heteroaromatic compounds as immunomodulators
|
|
EP3558973B1
(en)
|
2016-12-22 |
2021-09-15 |
Incyte Corporation |
Pyridine derivatives as immunomodulators
|
|
IL295660A
(en)
|
2016-12-22 |
2022-10-01 |
Incyte Corp |
Benzooxazole derivatives as immunomodulators
|
|
ES2929193T3
(es)
|
2016-12-22 |
2022-11-25 |
Incyte Corp |
Derivados de tetrahidro imidazo[4,5-c]piridina como inductores de la internalización de PD-L1
|
|
ES2874756T3
(es)
|
2016-12-22 |
2021-11-05 |
Incyte Corp |
Derivados de triazolo[1,5-A]piridina como inmunomoduladores
|
|
EP3604301B1
(en)
*
|
2017-03-31 |
2021-09-22 |
FUJIFILM Corporation |
4-pyridone compound or salt thereof, and pharmaceutical composition and formulation including same
|
|
CN108191746B
(zh)
*
|
2018-02-02 |
2020-06-16 |
暨南大学 |
一种羟基吡啶酮类化合物及其制备方法与应用
|
|
RS64055B1
(sr)
|
2018-03-30 |
2023-04-28 |
Incyte Corp |
Heterociklična jedinjenja kao imunomodulatori
|
|
EP4219492B1
(en)
|
2018-05-11 |
2024-11-27 |
Incyte Corporation |
Heterocyclic compounds as immunomodulators
|
|
WO2020097400A1
(en)
|
2018-11-07 |
2020-05-14 |
Dana-Farber Cancer Institute, Inc. |
Imidazopyridine derivatives and aza-imidazopyridine derivatives as janus kinase 2 inhibitors and uses thereof
|
|
US12415816B2
(en)
|
2018-11-07 |
2025-09-16 |
Dana-Farber Cancer Institute, Inc. |
Benzothiazole derivatives and 7-aza-benzothiazole derivatives as janus kinase 2 inhibitors and uses thereof
|
|
US12522583B2
(en)
|
2018-11-07 |
2026-01-13 |
Dana-Farber Cancer Institute, Inc. |
Benzimidazole derivatives and aza-benzimidazole derivatives as Janus kinase 2 inhibitors and uses thereof
|
|
JP7665593B2
(ja)
|
2019-08-09 |
2025-04-21 |
インサイト・コーポレイション |
Pd-1/pd-l1阻害剤の塩
|
|
EP4037773A1
(en)
|
2019-09-30 |
2022-08-10 |
Incyte Corporation |
Pyrido[3,2-d]pyrimidine compounds as immunomodulators
|
|
BR112022009031A2
(pt)
|
2019-11-11 |
2022-10-11 |
Incyte Corp |
Sais e formas cristalinas de um inibidor de pd-1/pd-l1
|
|
CN111170936B
(zh)
|
2020-01-19 |
2021-01-01 |
杭州泽德医药科技有限公司 |
3,4-二羟基-n-(1’-苄基-2’-羟乙基)-2-甲基吡啶氯化物及制备和应用
|
|
TW202204350A
(zh)
|
2020-05-06 |
2022-02-01 |
美商雅捷可斯治療公司 |
作為jak2抑制劑之6-雜芳基氧基苯并咪唑及氮雜苯并咪唑
|
|
KR102377058B1
(ko)
|
2020-11-04 |
2022-03-22 |
경북대학교 산학협력단 |
니아스텔라 코리엔시스에서 유래한 카테콜 o-메틸 트렌스퍼라제 및 이의 변이체
|
|
WO2022099018A1
(en)
|
2020-11-06 |
2022-05-12 |
Incyte Corporation |
Process of preparing a pd-1/pd-l1 inhibitor
|
|
US11760756B2
(en)
|
2020-11-06 |
2023-09-19 |
Incyte Corporation |
Crystalline form of a PD-1/PD-L1 inhibitor
|
|
EP4240739A1
(en)
|
2020-11-06 |
2023-09-13 |
Incyte Corporation |
Process for making a pd-1/pd-l1 inhibitor and salts and crystalline forms thereof
|
|
US12043632B2
(en)
|
2020-12-23 |
2024-07-23 |
Ajax Therapeutics, Inc. |
6-heteroaryloxy benzimidazoles and azabenzimidazoles as JAK2 inhibitors
|
|
US20250276955A1
(en)
*
|
2021-07-19 |
2025-09-04 |
Baylor College Of Medicine |
Coronavirus main protease inhibitors and methods using same
|
|
CA3234638A1
(en)
|
2021-11-09 |
2023-05-19 |
Ajax Therapeutics, Inc. |
6-heteroaryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors
|
|
WO2023086320A1
(en)
|
2021-11-09 |
2023-05-19 |
Ajax Therapeutics, Inc. |
Forms and compositions of inhibitors of jak2
|
|
CN114716366B
(zh)
*
|
2022-04-13 |
2023-12-26 |
浙江大学 |
3-羟基吡啶-4-酮类衍生物及在抑制肾细胞铁死亡中的应用
|
|
CN116947812B
(zh)
*
|
2023-06-30 |
2025-09-02 |
南京红太阳医药研究院有限公司 |
一种艾司奥美拉唑镁降解杂质的制备方法
|
|
WO2025257687A1
(en)
*
|
2024-06-11 |
2025-12-18 |
Universidade Do Porto |
Hydroxypyridinone compounds as inhibitors of catechol-o-methyltransferase
|