JP2013515073A5 - - Google Patents

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Publication number
JP2013515073A5
JP2013515073A5 JP2012546129A JP2012546129A JP2013515073A5 JP 2013515073 A5 JP2013515073 A5 JP 2013515073A5 JP 2012546129 A JP2012546129 A JP 2012546129A JP 2012546129 A JP2012546129 A JP 2012546129A JP 2013515073 A5 JP2013515073 A5 JP 2013515073A5
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JP
Japan
Prior art keywords
compound
hydrogen
gluc
stereoisomer
solvate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2012546129A
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English (en)
Japanese (ja)
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JP5760008B2 (ja
JP2013515073A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2010/061420 external-priority patent/WO2011079091A1/en
Publication of JP2013515073A publication Critical patent/JP2013515073A/ja
Publication of JP2013515073A5 publication Critical patent/JP2013515073A5/ja
Application granted granted Critical
Publication of JP5760008B2 publication Critical patent/JP5760008B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2012546129A 2009-12-22 2010-12-21 (メチルスルホニル)エチルベンゼンイソインドリン誘導体及びその治療的使用 Expired - Fee Related JP5760008B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28935609P 2009-12-22 2009-12-22
US61/289,356 2009-12-22
PCT/US2010/061420 WO2011079091A1 (en) 2009-12-22 2010-12-21 (methylsulfonyl) ethyl benzene isoindoline derivatives and their therapeutical uses

Publications (3)

Publication Number Publication Date
JP2013515073A JP2013515073A (ja) 2013-05-02
JP2013515073A5 true JP2013515073A5 (enExample) 2014-02-13
JP5760008B2 JP5760008B2 (ja) 2015-08-05

Family

ID=43528318

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012546129A Expired - Fee Related JP5760008B2 (ja) 2009-12-22 2010-12-21 (メチルスルホニル)エチルベンゼンイソインドリン誘導体及びその治療的使用

Country Status (18)

Country Link
US (1) US8716252B2 (enExample)
EP (1) EP2516395A1 (enExample)
JP (1) JP5760008B2 (enExample)
KR (1) KR20120113219A (enExample)
CN (1) CN102770412A (enExample)
AU (1) AU2010333767A1 (enExample)
BR (1) BR112012015129A2 (enExample)
CA (1) CA2783616A1 (enExample)
CL (1) CL2012001671A1 (enExample)
CO (1) CO6640204A2 (enExample)
CR (1) CR20120335A (enExample)
EC (1) ECSP12011987A (enExample)
MX (1) MX2012007217A (enExample)
PH (1) PH12012501237A1 (enExample)
RU (1) RU2012131164A (enExample)
SG (1) SG181891A1 (enExample)
WO (1) WO2011079091A1 (enExample)
ZA (1) ZA201203944B (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2012236655B2 (en) 2011-03-28 2016-09-22 Deuterx, Llc, 2',6'-dioxo-3'-deutero-piperdin-3-yl-isoindoline compounds
CA2935495C (en) 2013-01-14 2021-04-20 Deuterx, Llc 3-(5-substituted-4-oxoquinazolin-3(4h)-yl)-3-deutero-piperidine-2,6-dione derivatives
US9290475B2 (en) 2013-03-14 2016-03-22 Deuterx, Llc 3-(substituted-4-oxoquinazolin-3(4H)-yl)-3-deutero-piperidine-2,6-dione derivatives and compositions comprising and methods of using the same
US9809603B1 (en) 2015-08-18 2017-11-07 Deuterx, Llc Deuterium-enriched isoindolinonyl-piperidinonyl conjugates and oxoquinazolin-3(4H)-yl-piperidinonyl conjugates and methods of treating medical disorders using same
MY195528A (en) 2016-03-17 2023-01-30 Hoffmann La Roche 5-Ethyl-4-Methyl-Pyrazole-3-Carboxamide Derivative Having Activity as Agonist of Taar
US20190008837A1 (en) * 2016-12-15 2019-01-10 University Of Utah Research Foundation Ophthalmic compositions and associated methods
EP3838898B1 (en) * 2018-08-16 2023-06-07 Korea Research Institute of Chemical Technology Isoindolin-1-one derivative, method for preparing the same, and pharmaceutical composition comprising the same as an effective component for preventing or treating cancer
AU2020353984B2 (en) 2019-09-27 2025-09-25 Takeda Pharmaceutical Company Limited 2-isoindol-1,3,4-oxadiazole derivatives useful as HDAC6 inhibitors

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