JP2013505962A5 - - Google Patents

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Publication number
JP2013505962A5
JP2013505962A5 JP2012531109A JP2012531109A JP2013505962A5 JP 2013505962 A5 JP2013505962 A5 JP 2013505962A5 JP 2012531109 A JP2012531109 A JP 2012531109A JP 2012531109 A JP2012531109 A JP 2012531109A JP 2013505962 A5 JP2013505962 A5 JP 2013505962A5
Authority
JP
Japan
Prior art keywords
combination
day
pharmaceutically acceptable
solvate
acceptable salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012531109A
Other languages
English (en)
Japanese (ja)
Other versions
JP2013505962A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2010/050495 external-priority patent/WO2011038380A2/en
Publication of JP2013505962A publication Critical patent/JP2013505962A/ja
Publication of JP2013505962A5 publication Critical patent/JP2013505962A5/ja
Pending legal-status Critical Current

Links

JP2012531109A 2009-09-28 2010-09-28 組合せ Pending JP2013505962A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US24626509P 2009-09-28 2009-09-28
US61/246,265 2009-09-28
US38573810P 2010-09-23 2010-09-23
US61/385,738 2010-09-23
PCT/US2010/050495 WO2011038380A2 (en) 2009-09-28 2010-09-28 Combination

Publications (2)

Publication Number Publication Date
JP2013505962A JP2013505962A (ja) 2013-02-21
JP2013505962A5 true JP2013505962A5 (https=) 2013-11-14

Family

ID=43796526

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012531109A Pending JP2013505962A (ja) 2009-09-28 2010-09-28 組合せ

Country Status (13)

Country Link
US (1) US20120245180A1 (https=)
EP (1) EP2482819A4 (https=)
JP (1) JP2013505962A (https=)
KR (1) KR20120099217A (https=)
CN (1) CN102665719A (https=)
AU (1) AU2010298020B8 (https=)
BR (1) BR112012006968A2 (https=)
CA (1) CA2775874A1 (https=)
EA (1) EA201270475A1 (https=)
IL (1) IL218846A0 (https=)
MX (1) MX2012003779A (https=)
WO (1) WO2011038380A2 (https=)
ZA (1) ZA201202258B (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI505828B (zh) 2010-12-20 2015-11-01 葛蘭素史克智慧財產(第二)有限公司 新穎醫藥組成物
EP2943199A1 (en) * 2013-01-09 2015-11-18 Glaxosmithkline Intellectual Property (No. 2) Limited Combination
WO2014169843A1 (en) * 2013-04-18 2014-10-23 Shanghai Fochon Pharmaceutical Co Ltd Certain protein kinase inhibitors
WO2018126192A1 (en) * 2016-12-30 2018-07-05 Children's Medical Center Corporation Map2k1 (mek1) as a therapeutic target for arteriovenous malformations and associated disorders

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7378423B2 (en) 2004-06-11 2008-05-27 Japan Tobacco Inc. Pyrimidine compound and medical use thereof
AU2005252110B2 (en) * 2004-06-11 2008-09-04 Shionogi & Co., Ltd. 5-amino-2,4,7-trioxo-3,4,7,8-tetrahydro-2H-pyrido[2,3-D] pyrimidine derivatives and related compounds for the treatment of cancer
PE20060608A1 (es) * 2004-10-13 2006-08-22 Wyeth Corp Analogos de 17-hidroxiwortmanina como inhibidores de pi3k
TW200815429A (en) 2006-04-11 2008-04-01 Smithkline Beecham Corp Thiazolidinedione derivatives as PI3 kinase inhibitors
CN101528231A (zh) * 2006-08-16 2009-09-09 埃克塞利希斯股份有限公司 在癌症的治疗中使用pi3k和mek调控剂
PE20090717A1 (es) 2007-05-18 2009-07-18 Smithkline Beecham Corp Derivados de quinolina como inhibidores de la pi3 quinasa

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