JP2013504594A - 薬学的に有用な複素環置換ラクタム - Google Patents
薬学的に有用な複素環置換ラクタム Download PDFInfo
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- JP2013504594A JP2013504594A JP2012528930A JP2012528930A JP2013504594A JP 2013504594 A JP2013504594 A JP 2013504594A JP 2012528930 A JP2012528930 A JP 2012528930A JP 2012528930 A JP2012528930 A JP 2012528930A JP 2013504594 A JP2013504594 A JP 2013504594A
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- pyrazolo
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- methylene
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Classifications
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
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| US24180609P | 2009-09-11 | 2009-09-11 | |
| US61/241,806 | 2009-09-11 | ||
| US37114710P | 2010-08-05 | 2010-08-05 | |
| US61/371,147 | 2010-08-05 | ||
| PCT/US2010/048441 WO2011031979A1 (en) | 2009-09-11 | 2010-09-10 | Pharmaceutically useful heterocycle-substituted lactams |
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| JP2013504594A true JP2013504594A (ja) | 2013-02-07 |
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| JP2012528930A Pending JP2013504594A (ja) | 2009-09-11 | 2010-09-10 | 薬学的に有用な複素環置換ラクタム |
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| EP (1) | EP2475652A1 (enExample) |
| JP (1) | JP2013504594A (enExample) |
| KR (1) | KR20120104521A (enExample) |
| CN (1) | CN102625803A (enExample) |
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| BR (1) | BR112012005550A2 (enExample) |
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| IN (1) | IN2012DN03112A (enExample) |
| MX (1) | MX2012002994A (enExample) |
| SG (1) | SG179083A1 (enExample) |
| WO (1) | WO2011031979A1 (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2024541979A (ja) * | 2021-10-29 | 2024-11-13 | ギリアード サイエンシーズ， インコーポレイテッド | Ｃｄ７３化合物 |
| JP7787991B2 (ja) | 2021-10-29 | 2025-12-17 | ギリアード サイエンシーズ， インコーポレイテッド | Ｃｄ７３化合物 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE554078T1 (de) | 2007-07-26 | 2012-05-15 | Vitae Pharmaceuticals Inc | Synthese von 11-beta-hydroxysteroid-dehydrogenase-1-hemmern |
| AR069207A1 (es) | 2007-11-07 | 2010-01-06 | Vitae Pharmaceuticals Inc | Ureas ciclicas como inhibidores de la 11 beta - hidroxi-esteroide deshidrogenasa 1 |
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- 2010-09-10 WO PCT/US2010/048441 patent/WO2011031979A1/en not_active Ceased
- 2010-09-10 EP EP10816161A patent/EP2475652A1/en not_active Withdrawn
- 2010-09-10 SG SG2012016929A patent/SG179083A1/en unknown
- 2010-09-10 BR BR112012005550A patent/BR112012005550A2/pt not_active IP Right Cessation
- 2010-09-10 AU AU2010292116A patent/AU2010292116A1/en not_active Abandoned
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- 2010-09-10 IN IN3112DEN2012 patent/IN2012DN03112A/en unknown
- 2010-09-10 CA CA2773854A patent/CA2773854A1/en not_active Abandoned
- 2010-09-10 KR KR1020127009217A patent/KR20120104521A/ko not_active Withdrawn
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2024541979A (ja) * | 2021-10-29 | 2024-11-13 | ギリアード サイエンシーズ， インコーポレイテッド | Ｃｄ７３化合物 |
| JP7787991B2 (ja) | 2021-10-29 | 2025-12-17 | ギリアード サイエンシーズ， インコーポレイテッド | Ｃｄ７３化合物 |
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| EP2475652A1 (en) | 2012-07-18 |
| KR20120104521A (ko) | 2012-09-21 |
| IN2012DN03112A (enExample) | 2015-09-18 |
| SG179083A1 (en) | 2012-04-27 |
| CN102625803A (zh) | 2012-08-01 |
| US20110071115A1 (en) | 2011-03-24 |
| MX2012002994A (es) | 2012-07-17 |
| WO2011031979A1 (en) | 2011-03-17 |
| IL218521A0 (en) | 2012-07-31 |
| BR112012005550A2 (pt) | 2015-09-08 |
| AU2010292116A1 (en) | 2012-05-03 |
| CA2773854A1 (en) | 2011-03-17 |
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