JP2013501733A5 - - Google Patents

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Publication number
JP2013501733A5
JP2013501733A5 JP2012524066A JP2012524066A JP2013501733A5 JP 2013501733 A5 JP2013501733 A5 JP 2013501733A5 JP 2012524066 A JP2012524066 A JP 2012524066A JP 2012524066 A JP2012524066 A JP 2012524066A JP 2013501733 A5 JP2013501733 A5 JP 2013501733A5
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JP
Japan
Prior art keywords
alkyl
heteroaryl
compound
formula
cycloalkyl
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
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JP2012524066A
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English (en)
Japanese (ja)
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JP2013501733A (ja
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Priority claimed from PCT/CA2010/001229 external-priority patent/WO2011017800A1/en
Publication of JP2013501733A publication Critical patent/JP2013501733A/ja
Publication of JP2013501733A5 publication Critical patent/JP2013501733A5/ja
Ceased legal-status Critical Current

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JP2012524066A 2009-08-10 2010-08-06 1,3−プロパンジスルホン酸を送達するための方法、化合物、および組成物 Ceased JP2013501733A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23259709P 2009-08-10 2009-08-10
US61/232,597 2009-08-10
PCT/CA2010/001229 WO2011017800A1 (en) 2009-08-10 2010-08-06 Methods, compounds, and compositions for delivering 1,3-propan ed isulfonic acid

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015179480A Division JP2016034960A (ja) 2009-08-10 2015-09-11 1,3−プロパンジスルホン酸を送達するための方法、化合物、および組成物

Publications (2)

Publication Number Publication Date
JP2013501733A JP2013501733A (ja) 2013-01-17
JP2013501733A5 true JP2013501733A5 (https=) 2013-08-29

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ID=43585812

Family Applications (2)

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JP2012524066A Ceased JP2013501733A (ja) 2009-08-10 2010-08-06 1,3−プロパンジスルホン酸を送達するための方法、化合物、および組成物
JP2015179480A Pending JP2016034960A (ja) 2009-08-10 2015-09-11 1,3−プロパンジスルホン酸を送達するための方法、化合物、および組成物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2015179480A Pending JP2016034960A (ja) 2009-08-10 2015-09-11 1,3−プロパンジスルホン酸を送達するための方法、化合物、および組成物

Country Status (15)

Country Link
US (2) US9051248B2 (https=)
EP (1) EP2464626A4 (https=)
JP (2) JP2013501733A (https=)
KR (1) KR20120087878A (https=)
CN (1) CN102471248B (https=)
AU (1) AU2010282170B2 (https=)
BR (1) BR112012002780A2 (https=)
CA (1) CA2768877A1 (https=)
EA (1) EA201290007A1 (https=)
IL (1) IL217572A (https=)
MX (1) MX2012001671A (https=)
NZ (1) NZ598085A (https=)
SG (2) SG10201600910YA (https=)
WO (1) WO2011017800A1 (https=)
ZA (1) ZA201201352B (https=)

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WO2011017800A1 (en) * 2009-08-10 2011-02-17 Bellus Health (International) Limited Methods, compounds, and compositions for delivering 1,3-propan ed isulfonic acid
WO2011107870A2 (en) * 2010-03-05 2011-09-09 Mahesh Kandula Compounds and compositions and their use in the treatment of diseases related to copper retention
US9303038B2 (en) 2011-09-06 2016-04-05 Cellix Bio Private Limited Compositions and methods for the treatment of epilepsy and neurological diseases
WO2013168021A1 (en) 2012-05-07 2013-11-14 Mahesh Kandula Compositions and methods for treatment of neuromuscular disorders and neurodegenerative disorders
WO2013167985A1 (en) 2012-05-07 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of neurological disorders
WO2013167990A1 (en) 2012-05-07 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of depression
WO2013168023A1 (en) 2012-05-08 2013-11-14 Mahesh Kandula Compositions and methods for treatment of parkinson's disease
US9403826B2 (en) 2012-05-08 2016-08-02 Cellix Bio Private Limited Compositions and methods for the treatment of inflammatory disorders
US9434704B2 (en) 2012-05-08 2016-09-06 Cellix Bio Private Limited Compositions and methods for the treatment of neurological degenerative disorders
WO2013167991A1 (en) 2012-05-08 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of metabolic disorders
WO2013168025A1 (en) 2012-05-08 2013-11-14 Mahesh Kandula Compositions and methods for treatment of blood clotting disorders
WO2013167999A2 (en) 2012-05-10 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of neurologic diseases
US9273061B2 (en) 2012-05-10 2016-03-01 Cellix Bio Private Limited Compositions and methods for the treatment of chronic pain
WO2013168005A2 (en) 2012-05-10 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of restless leg syndrome and fibromyalgia
WO2013167997A2 (en) 2012-05-10 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of metabolic syndrome
WO2013168014A1 (en) 2012-05-10 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of familial amyloid polyneuropathy
WO2013168004A2 (en) 2012-05-10 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of fibromyalgia pain
WO2013168000A1 (en) 2012-05-10 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of severe pain
WO2013168012A1 (en) 2012-05-10 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of respiratory disorders
WO2013168001A1 (en) 2012-05-10 2013-11-14 Mahesh Kandula Compositions and methods for the treatment of moderate to severe pain
WO2013168033A1 (en) 2012-05-10 2013-11-14 Mahesh Kandula Compositions and methods for treatment of neurologic diseases
US9233161B2 (en) 2012-05-10 2016-01-12 Cellix Bio Private Limited Compositions and methods for the treatment of neurological conditions
US9403857B2 (en) 2012-05-10 2016-08-02 Cellix Bio Private Limited Compositions and methods for the treatment of metabolic syndrome
US9394288B2 (en) 2012-05-10 2016-07-19 Cellix Bio Private Limited Compositions and methods for the treatment of asthma and allergy
WO2013175344A2 (en) 2012-05-23 2013-11-28 Mahesh Kandula Compositions and methods for the treatment of periodontitis and rheumatoid arthritis
US9492409B2 (en) 2012-05-23 2016-11-15 Cellix Bio Private Limited Compositions and methods for the treatment of local pain
US9498461B2 (en) 2012-05-23 2016-11-22 Cellix Bio Private Limited Compositions and methods for the treatment of inflammatory bowel disease
EP2852569B1 (en) 2012-05-23 2020-10-14 Cellixbio Private Limited Compositions and methods for the treatment of multiple sclerosis
AU2013264820A1 (en) 2012-05-23 2014-11-27 Cellixbio Private Limited Compositions and methods for treatment of mucositis
US9227974B2 (en) 2012-05-23 2016-01-05 Cellex Bio Private Limited Compositions and methods for the treatment of respiratory disorders
US9108942B1 (en) 2014-11-05 2015-08-18 Mahesh Kandula Compositions and methods for the treatment of moderate to severe pain
WO2014020480A2 (en) 2012-08-03 2014-02-06 Mahesh Kandula Compositions and methods for the treatment migraine and neurologic diseases
WO2014037833A2 (en) 2012-09-06 2014-03-13 Mahesh Kandula Compositions and methods for the treatment inflammation and lipid disorders
CN104364231A (zh) 2012-09-08 2015-02-18 塞利克斯比奥私人有限公司 用于治疗炎症和脂质异常的组合物和方法
CN103012463B (zh) * 2013-01-17 2016-02-10 南京理工大学 (s)-3-甲基-2-(叔丁基二甲基硅氧基)-1-溴丁烷的合成方法
US9333187B1 (en) 2013-05-15 2016-05-10 Cellix Bio Private Limited Compositions and methods for the treatment of inflammatory bowel disease
EP3004049B1 (en) 2013-06-04 2018-09-05 Cellixbio Private Limited Compositions and methods for the treatment of diabetes and pre-diabetes
US9096537B1 (en) 2014-12-31 2015-08-04 Mahesh Kandula Compositions and methods for the treatment of mucositis
CN103755679A (zh) * 2014-02-14 2014-04-30 宁德新能源科技有限公司 一种亚烷基二磺酸酐的制备方法
SG11201608906SA (en) 2014-04-30 2016-11-29 Icahn School Med Mount Sinai Use of 1,3-propanedisulfonic acid or pharmaceutically acceptable salts thereof for the treatment of sarcoidosis
EP3240779B1 (en) 2014-09-26 2020-10-28 Cellixbio Private Limited Compositions and methods for the treatment of epilepsy and neurological disorders
JP6698643B2 (ja) 2014-09-29 2020-05-27 セリックス バイオ プライヴェート リミテッドCellix Bio Private Limited 多発性硬化症の治療のための組成物及び方法
AU2014414316B2 (en) 2014-10-27 2020-04-09 Cellix Bio Private Limited Three component salts of fumaric acid monomethyl ester with piperazine or ethylene diamine for the treatment of multiple sclerosis
US10208014B2 (en) 2014-11-05 2019-02-19 Cellix Bio Private Limited Compositions and methods for the treatment of neurological disorders
US9321716B1 (en) 2014-11-05 2016-04-26 Cellix Bio Private Limited Compositions and methods for the treatment of metabolic syndrome
US9284287B1 (en) 2014-11-05 2016-03-15 Cellix Bio Private Limited Compositions and methods for the suppression of carbonic anhydrase activity
US9150557B1 (en) 2014-11-05 2015-10-06 Cellix Bio Private Limited Compositions and methods for the treatment of hyperglycemia
US9175008B1 (en) 2014-11-05 2015-11-03 Cellix Bio Private Limited Prodrugs of anti-platelet agents
US9290486B1 (en) 2014-11-05 2016-03-22 Cellix Bio Private Limited Compositions and methods for the treatment of epilepsy
US9173877B1 (en) 2014-11-05 2015-11-03 Cellix Bio Private Limited Compositions and methods for the treatment of local pain
US9932294B2 (en) 2014-12-01 2018-04-03 Cellix Bio Private Limited Compositions and methods for the treatment of multiple sclerosis
US9206111B1 (en) 2014-12-17 2015-12-08 Cellix Bio Private Limited Compositions and methods for the treatment of neurological diseases
CA2973178C (en) 2015-01-06 2022-11-01 Cellix Bio Private Limited Bupivacaine derivatives and their use in the treatment of inflammation and pain
CN109988085B (zh) * 2017-12-29 2021-11-09 张家港市国泰华荣化工新材料有限公司 金属离子含量低的1,3-丙二烷基磺酸的制备方法
KR102568464B1 (ko) * 2018-07-06 2023-08-21 화이자 인코포레이티드 피롤로[2,3-d]피리미딘 화합물의 제조 방법, 이의 중간체, 및 이의 용도
CA3120658A1 (en) 2018-11-22 2020-05-28 Universite De Nantes Disulfonate stilbenes for use in the treatment of proliferative diseases
JP7324082B2 (ja) * 2019-08-07 2023-08-09 東ソー・ファインケム株式会社 カルボン酸無水物またはスルホン酸無水物の製造方法
CN110818673B (zh) * 2019-11-22 2022-08-16 湖南阿斯达新材料有限公司 一种环状二磺酸亚甲酯的合成方法
CN112574167B (zh) * 2020-12-07 2021-11-09 烟台海川化学制品有限公司 一种甲烷二磺酸亚甲酯的制备方法
KR20240001118A (ko) * 2021-05-31 2024-01-03 미쯔비시 가스 케미칼 컴파니, 인코포레이티드 신규 아미노 화합물 및 그의 제조방법, 그리고, 이것을 이용한 에폭시 수지용 경화제, 에폭시 수지 조성물 및 에폭시 수지 경화물
CN115124502B (zh) * 2022-08-03 2024-09-13 张家港市国泰华荣化工新材料有限公司 一种丙烯二磺酸酐的制备方法

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