JP2012522007A5 - - Google Patents

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Publication number
JP2012522007A5
JP2012522007A5 JP2012502295A JP2012502295A JP2012522007A5 JP 2012522007 A5 JP2012522007 A5 JP 2012522007A5 JP 2012502295 A JP2012502295 A JP 2012502295A JP 2012502295 A JP2012502295 A JP 2012502295A JP 2012522007 A5 JP2012522007 A5 JP 2012522007A5
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JP
Japan
Prior art keywords
methyl
benzo
oxazin
oxo
dihydro
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JP2012502295A
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English (en)
Japanese (ja)
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JP5730281B2 (ja
JP2012522007A (ja
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Priority claimed from PCT/US2010/028878 external-priority patent/WO2010111626A2/en
Publication of JP2012522007A publication Critical patent/JP2012522007A/ja
Publication of JP2012522007A5 publication Critical patent/JP2012522007A5/ja
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Publication of JP5730281B2 publication Critical patent/JP5730281B2/ja
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JP2012502295A 2009-03-27 2010-03-26 ポリ（ａｄｐ−リボース）ポリメラーゼ（ｐａｒｐ）阻害剤 Active JP5730281B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US16413209P 2009-03-27 2009-03-27
US61/164,132 2009-03-27
PCT/US2010/028878 WO2010111626A2 (en) 2009-03-27 2010-03-26 Poly (adp-ribose) polymerase (parp) inhibitors

Publications (3)

Publication Number Publication Date
JP2012522007A JP2012522007A (ja) 2012-09-20
JP2012522007A5 true JP2012522007A5 (https=) 2013-05-16
JP5730281B2 JP5730281B2 (ja) 2015-06-10

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ID=42288484

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JP2012502295A Active JP5730281B2 (ja) 2009-03-27 2010-03-26 ポリ（ａｄｐ−リボース）ポリメラーゼ（ｐａｒｐ）阻害剤

Country Status (4)

Country Link
US (1) US8669249B2 (https=)
EP (1) EP2415767B1 (https=)
JP (1) JP5730281B2 (https=)
WO (1) WO2010111626A2 (https=)

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WO2023046149A1 (zh) * 2021-09-26 2023-03-30 张文燕 喹喔啉类化合物及其医药用途
WO2023051716A1 (zh) * 2021-09-30 2023-04-06 海思科医药集团股份有限公司 杂芳基衍生物parp抑制剂及其用途
EP4410791A4 (en) * 2021-09-30 2025-10-22 Xizang Haisco Pharmaceutical Co Ltd BICYCLIC DERIVATIVE PARP INHIBITOR AND ITS USE
US20250289800A1 (en) * 2021-11-19 2025-09-18 Kangbaida (Sichuan) Biotechnology Co., Ltd. Selective Parp1 Inhibitor And Application Thereof
AU2023235233A1 (en) 2022-03-14 2024-09-12 Slap Pharmaceuticals Llc Multicyclic compounds
CN119487027A (zh) * 2022-04-28 2025-02-18 宁波新湾科技发展有限公司 作为parp1抑制剂的化合物
TW202408509A (zh) * 2022-07-14 2024-03-01 大陸商西藏海思科製藥有限公司 雜芳基衍生物的藥物組合物及其在醫藥上的應用
WO2024041608A1 (zh) * 2022-08-24 2024-02-29 四川海思科制药有限公司 一种杂芳基衍生物parp抑制剂的晶体形式及其用途
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