JP2012509338A5 - - Google Patents

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Publication number
JP2012509338A5
JP2012509338A5 JP2011537582A JP2011537582A JP2012509338A5 JP 2012509338 A5 JP2012509338 A5 JP 2012509338A5 JP 2011537582 A JP2011537582 A JP 2011537582A JP 2011537582 A JP2011537582 A JP 2011537582A JP 2012509338 A5 JP2012509338 A5 JP 2012509338A5
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JP
Japan
Prior art keywords
group
independently
alkyl
haloalkyl
halogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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JP2011537582A
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English (en)
Japanese (ja)
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JP2012509338A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2009/064981 external-priority patent/WO2010059719A2/en
Publication of JP2012509338A publication Critical patent/JP2012509338A/ja
Publication of JP2012509338A5 publication Critical patent/JP2012509338A5/ja
Pending legal-status Critical Current

Links

JP2011537582A 2008-11-19 2009-11-18 二量体1−アリールピラゾール誘導体 Pending JP2012509338A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11602108P 2008-11-19 2008-11-19
US61/116,021 2008-11-19
PCT/US2009/064981 WO2010059719A2 (en) 2008-11-19 2009-11-18 Dimeric 1-arylpyrazole derivatives

Publications (2)

Publication Number Publication Date
JP2012509338A JP2012509338A (ja) 2012-04-19
JP2012509338A5 true JP2012509338A5 (enExample) 2013-01-17

Family

ID=42034586

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011537582A Pending JP2012509338A (ja) 2008-11-19 2009-11-18 二量体1−アリールピラゾール誘導体

Country Status (12)

Country Link
US (1) US8642636B2 (enExample)
EP (1) EP2364300B1 (enExample)
JP (1) JP2012509338A (enExample)
CN (1) CN102264706A (enExample)
AU (1) AU2009316710B2 (enExample)
BR (1) BRPI0922042B1 (enExample)
CA (2) CA2743553C (enExample)
EA (1) EA020923B1 (enExample)
ES (1) ES2605811T3 (enExample)
MX (1) MX2011005214A (enExample)
NZ (1) NZ592985A (enExample)
WO (1) WO2010059719A2 (enExample)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG194902A1 (en) 2011-05-13 2013-12-30 Array Biopharma Inc Pyrrolidinyl urea and pyrrolidinyl thiourea compounds as trka kinase inhibitors
WO2014078378A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
WO2014078322A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Thiazolyl and oxazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
WO2014078328A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-bicyclic aryl,n'-pyrazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
WO2014078408A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Bicyclic heteroaryl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
EP2922844B1 (en) 2012-11-13 2018-01-10 Array Biopharma, Inc. N-pyrrolidinyl, n'-pyrazolyl- urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
CA2891334C (en) 2012-11-13 2021-10-19 Array Biopharma Inc. Bicyclic urea, thiourea, guanidine and cyanoguanidine compounds useful for the treatment of pain
US9790210B2 (en) 2012-11-13 2017-10-17 Array Biopharma Inc. N-(monocyclic aryl),N'-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
US9809578B2 (en) 2012-11-13 2017-11-07 Array Biopharma Inc. Pyrazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trkA kinase inhibitors
US9969694B2 (en) 2012-11-13 2018-05-15 Array Biopharma Inc. N-(arylalkyl)-N′-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
WO2014078372A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
JP2016164125A (ja) * 2013-07-02 2016-09-08 国立大学法人帯広畜産大学 バベシア症の治療剤及び予防剤
US10835533B2 (en) 2014-05-15 2020-11-17 Array Biopharma Inc. 1 -((3S,4R)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1H-pyrazol-5-yl)urea as a TrkA kinase inhibitor
US11384032B2 (en) 2016-05-12 2022-07-12 Verdesian Life Sciences, U.S., Llc Compositions for controlling enzyme-induced urea decomposition
KR102480799B1 (ko) 2017-03-28 2022-12-22 베르데시안 라이프 사이언시스 유.에스., 엘엘씨 효소-유도된 우레아 분해를 조절하기 위한 트리아릴메탄 화합물
WO2020096831A1 (en) 2018-11-06 2020-05-14 Dow Agrosciences Llc Safened compositions comprising pyridine carboxylate herbicides and cloquintocet
DK3876726T3 (da) * 2018-11-06 2025-03-03 Corteva Agriscience Llc Sammensætninger, som omfatter pyridincarboxylat-herbicider og azolcarboxylat-safeners
AU2019377057B2 (en) 2018-11-07 2025-02-20 Corteva Agriscience Llc Compositions comprising pyridine carboxylate herbicides and 4-hydroxyphenyl-pyruvate dioxygenase (HPPD) inhibitor herbicides
AU2019377056B2 (en) 2018-11-07 2025-02-27 Corteva Agriscience Llc Compositions comprising pyridine carboxylate herbicides with acetolactate synthase (ALS) inhibitor herbicides
PL3876733T3 (pl) 2018-11-07 2025-11-03 Corteva Agriscience Llc Kompozycje zawierające herbicydy pirydynokarboksylanowe z herbicydami jako inhibitorami fotosystemu ii i opcjonalnie herbicydami jako inhibitorami hppd
WO2020096932A1 (en) 2018-11-07 2020-05-14 Dow Agrosciences Llc Compositions comprising a pyridine carboxylate herbicide and protoporphyrinogen oxidase (protox) inhibitor herbicides
AU2019387370A1 (en) 2018-11-30 2021-06-10 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
US20230257370A1 (en) 2020-07-24 2023-08-17 Elanco Us Inc. Process for making an isoxazoline compound and intermediate thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966900A (en) * 1969-03-12 1976-06-29 Airwick Industries, Inc. Evaporator system comprising a stabilized pesticidal phosphoric acid ester and method for stabilizing such ester enclosed in an evaporator
JP2003516941A (ja) * 1999-12-02 2003-05-20 アベンティス クロップサイエンス ソシエテ アノニム 動物における節足動物の制御
US7262214B2 (en) * 2003-02-26 2007-08-28 Merial Limited 1-N-arylpyrazole derivatives in prevention of arthropod-borne and mosquito-borne diseases
JP4958304B2 (ja) 2004-06-26 2012-06-20 メリアル リミテッド 殺虫剤としてのn−フェニルピラゾール誘導体

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