JP2012503026A5 - - Google Patents

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Publication number
JP2012503026A5
JP2012503026A5 JP2011528084A JP2011528084A JP2012503026A5 JP 2012503026 A5 JP2012503026 A5 JP 2012503026A5 JP 2011528084 A JP2011528084 A JP 2011528084A JP 2011528084 A JP2011528084 A JP 2011528084A JP 2012503026 A5 JP2012503026 A5 JP 2012503026A5
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JP
Japan
Prior art keywords
polypeptide
enhanced
helix
helical
amino acid
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JP2011528084A
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English (en)
Japanese (ja)
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JP5711128B2 (ja
JP2012503026A (ja
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Priority claimed from PCT/US2009/057934 external-priority patent/WO2010034034A1/en
Publication of JP2012503026A publication Critical patent/JP2012503026A/ja
Publication of JP2012503026A5 publication Critical patent/JP2012503026A5/ja
Application granted granted Critical
Publication of JP5711128B2 publication Critical patent/JP5711128B2/ja
Expired - Fee Related legal-status Critical Current
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JP2011528084A 2008-09-22 2009-09-22 ペプチド模倣大環状分子 Expired - Fee Related JP5711128B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US9906308P 2008-09-22 2008-09-22
US61/099,063 2008-09-22
PCT/US2009/057934 WO2010034034A1 (en) 2008-09-22 2009-09-22 Peptidomimetic macrocycles

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014142904A Division JP6067626B2 (ja) 2008-09-22 2014-07-11 ペプチド模倣大環状分子

Publications (3)

Publication Number Publication Date
JP2012503026A JP2012503026A (ja) 2012-02-02
JP2012503026A5 true JP2012503026A5 (https=) 2013-05-16
JP5711128B2 JP5711128B2 (ja) 2015-04-30

Family

ID=41611441

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2011528084A Expired - Fee Related JP5711128B2 (ja) 2008-09-22 2009-09-22 ペプチド模倣大環状分子
JP2014142904A Expired - Fee Related JP6067626B2 (ja) 2008-09-22 2014-07-11 ペプチド模倣大環状分子
JP2016159624A Pending JP2016190882A (ja) 2008-09-22 2016-08-16 ペプチド模倣大環状分子

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2014142904A Expired - Fee Related JP6067626B2 (ja) 2008-09-22 2014-07-11 ペプチド模倣大環状分子
JP2016159624A Pending JP2016190882A (ja) 2008-09-22 2016-08-16 ペプチド模倣大環状分子

Country Status (10)

Country Link
US (5) US8524653B2 (https=)
EP (1) EP2342222B1 (https=)
JP (3) JP5711128B2 (https=)
CN (1) CN102482336B (https=)
AU (1) AU2009294877C1 (https=)
BR (1) BRPI0918948A2 (https=)
CA (1) CA2737922A1 (https=)
ES (1) ES2666458T3 (https=)
IL (1) IL211836A0 (https=)
WO (1) WO2010034034A1 (https=)

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AR088392A1 (es) 2011-10-18 2014-05-28 Aileron Therapeutics Inc Macrociclos peptidomimeticos
HK1205454A1 (en) 2012-02-15 2015-12-18 Aileron Therapeutics, Inc. Triazole-crosslinked and thioether-crosslinked peptidomimetic macrocycles
CA2862038C (en) 2012-02-15 2021-05-25 Aileron Therapeutics, Inc. Peptidomimetic macrocycles
ES2874525T3 (es) 2012-09-26 2021-11-05 Harvard College Péptidos grapados bloqueados con prolina y usos de los mismos
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EP2352507A4 (en) 2008-11-24 2012-04-25 Aileron Therapeutics Inc PEPTIDOMIMETIC MACROCYCLES WITH IMPROVED PROPERTIES
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JP2012532929A (ja) 2009-07-13 2012-12-20 プレジデント アンド フェロウズ オブ ハーバード カレッジ 二機能性のステープリングされたポリペプチドおよびそれらの使用
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US20110223149A1 (en) 2009-10-14 2011-09-15 Aileron Therapeutics, Inc. Peptidomimetic macrocycles
KR20170058446A (ko) 2010-08-13 2017-05-26 에일러론 테라퓨틱스 인코포레이티드 펩티도미메틱 거대고리
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AR088392A1 (es) 2011-10-18 2014-05-28 Aileron Therapeutics Inc Macrociclos peptidomimeticos
WO2013059530A2 (en) 2011-10-18 2013-04-25 Aileron Therapeutics, Inc. Peptidomimetic macrocycles
CA2862038C (en) 2012-02-15 2021-05-25 Aileron Therapeutics, Inc. Peptidomimetic macrocycles
HK1205454A1 (en) 2012-02-15 2015-12-18 Aileron Therapeutics, Inc. Triazole-crosslinked and thioether-crosslinked peptidomimetic macrocycles
BR112015009470A2 (pt) 2012-11-01 2019-12-17 Aileron Therapeutics Inc aminoácidos dissubstituídos e seus métodos de preparação e uso
WO2014138429A2 (en) 2013-03-06 2014-09-12 Aileron Therapeutics, Inc. Peptidomimetic macrocycles and use thereof in regulating hif1alpha

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