JP2011530534A5 - - Google Patents

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Publication number
JP2011530534A5
JP2011530534A5 JP2011522274A JP2011522274A JP2011530534A5 JP 2011530534 A5 JP2011530534 A5 JP 2011530534A5 JP 2011522274 A JP2011522274 A JP 2011522274A JP 2011522274 A JP2011522274 A JP 2011522274A JP 2011530534 A5 JP2011530534 A5 JP 2011530534A5
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JP
Japan
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spp
use according
infection
pharmaceutically acceptable
acceptable salt
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JP2011522274A
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English (en)
Japanese (ja)
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JP5496202B2 (ja
JP2011530534A (ja
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Priority claimed from PCT/US2009/053142 external-priority patent/WO2010017470A1/en
Publication of JP2011530534A publication Critical patent/JP2011530534A/ja
Publication of JP2011530534A5 publication Critical patent/JP2011530534A5/ja
Application granted granted Critical
Publication of JP5496202B2 publication Critical patent/JP5496202B2/ja
Active legal-status Critical Current
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JP2011522274A 2008-08-08 2009-08-07 C7−フルオロ置換テトラサイクリン化合物 Active JP5496202B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18830708P 2008-08-08 2008-08-08
US61/188,307 2008-08-08
PCT/US2009/053142 WO2010017470A1 (en) 2008-08-08 2009-08-07 C7-fluoro substituted tetracycline compounds

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014041460A Division JP5690957B2 (ja) 2008-08-08 2014-03-04 C7−フルオロ置換テトラサイクリン化合物

Publications (3)

Publication Number Publication Date
JP2011530534A JP2011530534A (ja) 2011-12-22
JP2011530534A5 true JP2011530534A5 (OSRAM) 2012-09-20
JP5496202B2 JP5496202B2 (ja) 2014-05-21

Family

ID=41110902

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2011522274A Active JP5496202B2 (ja) 2008-08-08 2009-08-07 C7−フルオロ置換テトラサイクリン化合物
JP2014041460A Expired - Fee Related JP5690957B2 (ja) 2008-08-08 2014-03-04 C7−フルオロ置換テトラサイクリン化合物
JP2015018405A Expired - Fee Related JP6041911B2 (ja) 2008-08-08 2015-02-02 C7−フルオロ置換テトラサイクリン化合物

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2014041460A Expired - Fee Related JP5690957B2 (ja) 2008-08-08 2014-03-04 C7−フルオロ置換テトラサイクリン化合物
JP2015018405A Expired - Fee Related JP6041911B2 (ja) 2008-08-08 2015-02-02 C7−フルオロ置換テトラサイクリン化合物

Country Status (31)

Country Link
US (10) US8906887B2 (OSRAM)
EP (3) EP3000805B1 (OSRAM)
JP (3) JP5496202B2 (OSRAM)
KR (3) KR101679023B1 (OSRAM)
CN (3) CN103936645B (OSRAM)
AR (3) AR072990A1 (OSRAM)
AU (1) AU2009279473B2 (OSRAM)
BR (1) BRPI0916985B1 (OSRAM)
CA (1) CA2732883C (OSRAM)
CO (1) CO6351777A2 (OSRAM)
CY (3) CY1114689T1 (OSRAM)
DK (2) DK2682387T3 (OSRAM)
ES (3) ES2430254T3 (OSRAM)
FR (1) FR19C1012I2 (OSRAM)
HR (2) HRP20130928T1 (OSRAM)
HU (2) HUE026562T2 (OSRAM)
IL (3) IL211120A (OSRAM)
LT (1) LTC2323972I2 (OSRAM)
LU (1) LUC00107I2 (OSRAM)
MX (2) MX358961B (OSRAM)
NL (1) NL300971I2 (OSRAM)
NO (1) NO2019010I1 (OSRAM)
NZ (3) NZ591051A (OSRAM)
PL (3) PL3000805T3 (OSRAM)
PT (2) PT2323972E (OSRAM)
RS (2) RS53003B (OSRAM)
SG (1) SG10201806714PA (OSRAM)
SI (2) SI2323972T1 (OSRAM)
SM (1) SMT201600045B (OSRAM)
TW (3) TWI453183B (OSRAM)
WO (1) WO2010017470A1 (OSRAM)

Families Citing this family (18)

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SI2323972T1 (sl) 2008-08-08 2013-11-29 Tetraphase Pharmaceuticals, Inc. C7-fluoro substituirane tetraciklinske spojine
CN107021887A (zh) 2009-05-08 2017-08-08 四相制药公司 四环素类化合物
IN2012DN02502A (OSRAM) * 2009-08-28 2015-08-28 Tetraphase Pharmaceuticals Inc
WO2012021712A1 (en) * 2010-08-12 2012-02-16 Tetraphase Pharmaceuticals, Inc. Tetracycline analogs
WO2012021829A1 (en) * 2010-08-12 2012-02-16 Tetraphase Pharmaceuticals, Inc. Methods of treating bacterial infections
WO2012065028A2 (en) 2010-11-11 2012-05-18 Concert Pharmaceuticals Inc. Substituted tetracyclines
CN108276404A (zh) 2012-08-31 2018-07-13 四相制药公司 四环素化合物
CN104230960B (zh) * 2013-06-06 2017-02-15 山东轩竹医药科技有限公司 四并环类间变性淋巴瘤激酶抑制剂
MA40836A (fr) 2014-10-23 2017-08-29 Tetraphase Pharmaceuticals Inc Procédures de semi-synthèse
WO2017097891A1 (en) 2015-12-10 2017-06-15 Sandoz Ag Crystalline eravacycline
US10975029B2 (en) 2016-01-22 2021-04-13 Sandoz Ag Crystalline eravacycline bis-hydrochloride
SG11201809561WA (en) 2016-05-02 2018-11-29 Paratek Pharm Innc 9-aminomethyl minocycline compounds and methods of use thereof in urinary tract infection (uti) treatment
CN107759503A (zh) * 2016-08-16 2018-03-06 四川科伦博泰生物医药股份有限公司 一种四环素衍生物及其用途
US20230031954A1 (en) 2016-08-30 2023-02-02 Tetraphase Phamaceuticals, Inc. Tetracycline compounds and methods of treatment
CN110582486B (zh) 2016-10-19 2024-01-12 四相制药公司 艾若威四环素的结晶形式
AU2017353588B2 (en) 2016-11-01 2022-07-14 Paratek Pharmaceuticals, Inc. 9-aminomethyl minocycline compounds and use thereof in treating Community-Acquired Bacterial Pneumonia (CABP)
WO2020097450A1 (en) 2018-11-09 2020-05-14 Tetraphase Pharmaceuticals, Inc. Polymorphic forms of a compound and uses thereof
EP4531866A1 (en) * 2022-05-29 2025-04-09 B.G. Negev Technologies and Applications Ltd., at Ben-Gurion University Eravacycline for treating cancer

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CN107021887A (zh) 2009-05-08 2017-08-08 四相制药公司 四环素类化合物
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CN108276404A (zh) 2012-08-31 2018-07-13 四相制药公司 四环素化合物

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