JP2011521962A5 - - Google Patents

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Publication number
JP2011521962A5
JP2011521962A5 JP2011511814A JP2011511814A JP2011521962A5 JP 2011521962 A5 JP2011521962 A5 JP 2011521962A5 JP 2011511814 A JP2011511814 A JP 2011511814A JP 2011511814 A JP2011511814 A JP 2011511814A JP 2011521962 A5 JP2011521962 A5 JP 2011521962A5
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JP
Japan
Prior art keywords
agent
compound
prodrug
alkyl
pharmaceutically acceptable
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2011511814A
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English (en)
Japanese (ja)
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JP2011521962A (ja
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Publication date
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Priority claimed from PCT/US2009/045452 external-priority patent/WO2009146365A1/en
Publication of JP2011521962A publication Critical patent/JP2011521962A/ja
Publication of JP2011521962A5 publication Critical patent/JP2011521962A5/ja
Withdrawn legal-status Critical Current

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JP2011511814A 2008-05-29 2009-05-28 メラニン凝集ホルモン受容体−1アンタゴニストとしてのヒドロキシ置換チエノピリミジノン Withdrawn JP2011521962A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5694908P 2008-05-29 2008-05-29
US61/056,949 2008-05-29
PCT/US2009/045452 WO2009146365A1 (en) 2008-05-29 2009-05-28 Hydroxy substituted thieno pyrimidinones as melanin concentrating hormone receptor-1 antagonists

Publications (2)

Publication Number Publication Date
JP2011521962A JP2011521962A (ja) 2011-07-28
JP2011521962A5 true JP2011521962A5 (https=) 2011-10-06

Family

ID=41017166

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011511814A Withdrawn JP2011521962A (ja) 2008-05-29 2009-05-28 メラニン凝集ホルモン受容体−1アンタゴニストとしてのヒドロキシ置換チエノピリミジノン

Country Status (17)

Country Link
US (1) US7989433B2 (https=)
EP (1) EP2310394A1 (https=)
JP (1) JP2011521962A (https=)
KR (1) KR20110021988A (https=)
CN (1) CN102099360A (https=)
AR (1) AR075260A1 (https=)
AU (1) AU2009251331A1 (https=)
BR (1) BRPI0913197A2 (https=)
CA (1) CA2726264A1 (https=)
CO (1) CO6280492A2 (https=)
EA (1) EA201001882A1 (https=)
IL (1) IL209354A0 (https=)
MX (1) MX2010012803A (https=)
PE (1) PE20091928A1 (https=)
TW (1) TW201000487A (https=)
WO (1) WO2009146365A1 (https=)
ZA (1) ZA201008451B (https=)

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Publication number Priority date Publication date Assignee Title
JP2010525077A (ja) * 2007-04-25 2010-07-22 ブリストル−マイヤーズ スクイブ カンパニー 非塩基性メラニン凝集ホルモン受容体−1アンタゴニスト
NZ602089A (en) 2010-02-17 2014-05-30 Takeda Pharmaceutical Heterocyclic compounds having cell division cycle 7 inhibitory activity
CA2857231A1 (en) 2011-12-06 2013-06-13 Unilever Plc Skin anti-ageing composition
IL225900A0 (en) * 2013-04-22 2014-03-31 Perrigo Api Ltd A process for the preparation of nicotine that includes the enzymatic reduction of 4-(methylamino)-1-(3-pyridinyl)-1-butanone
EP2921856B1 (en) * 2014-03-18 2016-09-14 Serum Institute Of India Private Limited A quantitative assay for 4-pyrrolidinopyridine (4-ppy) in polysaccharide-protein conjugate vaccines
RU2687160C2 (ru) * 2014-12-30 2019-05-07 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Пиколинамидные соединения с фунгицидной активностью
JP6687625B2 (ja) 2014-12-30 2020-04-22 ダウ アグロサイエンシィズ エルエルシー 殺真菌活性を有するピコリンアミド化合物
AU2021206286A1 (en) * 2020-01-10 2024-08-08 Consynance Therapeutics, Inc. Therapeutic combinations of drugs and methods of using them
HUP2200222A1 (hu) 2022-06-17 2023-12-28 Richter Gedeon Nyrt MCHR1 antagonisták a Prader-Willi szindróma kezelésére

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