JP2011520847A5 - - Google Patents
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- Publication number
- JP2011520847A5 JP2011520847A5 JP2011508945A JP2011508945A JP2011520847A5 JP 2011520847 A5 JP2011520847 A5 JP 2011520847A5 JP 2011508945 A JP2011508945 A JP 2011508945A JP 2011508945 A JP2011508945 A JP 2011508945A JP 2011520847 A5 JP2011520847 A5 JP 2011520847A5
- Authority
- JP
- Japan
- Prior art keywords
- ethoxy
- xaa
- acetyl
- amino
- seq
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 0 *C(CCC(NCCOCC*CCOCCOCC(NCCCC[C@](C(P)=O)N*)O)O)[N+]([O-])=O Chemical compound *C(CCC(NCCOCC*CCOCCOCC(NCCCC[C@](C(P)=O)N*)O)O)[N+]([O-])=O 0.000 description 8
- XJXNZODHKPMSDQ-PLNGDYQASA-N C/C(/C(C)=O)=C/C(N)=C Chemical compound C/C(/C(C)=O)=C/C(N)=C XJXNZODHKPMSDQ-PLNGDYQASA-N 0.000 description 1
- CVMXXJSHVQQZRG-UHFFFAOYSA-N CC1CCC(CNC(CCCCCCCCCCCCCCCCCCC(O)[U])[U])CC1 Chemical compound CC1CCC(CNC(CCCCCCCCCCCCCCCCCCC(O)[U])[U])CC1 CVMXXJSHVQQZRG-UHFFFAOYSA-N 0.000 description 1
- JRMQQXSMFOBGII-UHFFFAOYSA-N O=CCCCCCCCCCCCCCCCCCNCC1CCCCC1 Chemical compound O=CCCCCCCCCCCCCCCCCCNCC1CCCCC1 JRMQQXSMFOBGII-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08156360.3 | 2008-05-16 | ||
| EP08156360 | 2008-05-16 | ||
| EP09154461.9 | 2009-03-05 | ||
| EP09154461 | 2009-03-05 | ||
| PCT/EP2009/055989 WO2009138511A1 (en) | 2008-05-16 | 2009-05-18 | Long-acting y2 and/or y4 receptor agonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2011520847A JP2011520847A (ja) | 2011-07-21 |
| JP2011520847A5 true JP2011520847A5 (cg-RX-API-DMAC7.html) | 2012-07-05 |
Family
ID=40934036
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011508945A Withdrawn JP2011520847A (ja) | 2008-05-16 | 2009-05-18 | 遅効型y2及び/又はy4レセプターアゴニスト |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20110275559A1 (cg-RX-API-DMAC7.html) |
| EP (1) | EP2279204A1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP2011520847A (cg-RX-API-DMAC7.html) |
| KR (1) | KR20110017874A (cg-RX-API-DMAC7.html) |
| CN (1) | CN102027007A (cg-RX-API-DMAC7.html) |
| AU (1) | AU2009248041B2 (cg-RX-API-DMAC7.html) |
| BR (1) | BRPI0912615A2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2723855A1 (cg-RX-API-DMAC7.html) |
| IL (1) | IL208836A0 (cg-RX-API-DMAC7.html) |
| MX (1) | MX2010011845A (cg-RX-API-DMAC7.html) |
| RU (1) | RU2504550C2 (cg-RX-API-DMAC7.html) |
| WO (1) | WO2009138511A1 (cg-RX-API-DMAC7.html) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5767582B2 (ja) | 2009-07-02 | 2015-08-19 | 武田薬品工業株式会社 | ペプチド及びその用途 |
| US20130040877A1 (en) * | 2009-09-18 | 2013-02-14 | Novo Nordisk A/S | Long-acting y2 receptor agonists |
| CN102905722A (zh) * | 2009-11-13 | 2013-01-30 | 诺沃—诺迪斯克有限公司 | 长效y2受体激动剂 |
| GB201001333D0 (en) * | 2010-01-27 | 2010-03-17 | Imp Innovations Ltd | Novel compounds and their effects on feeding behaviour |
| WO2012006566A2 (en) | 2010-07-09 | 2012-01-12 | Amylin Pharmaceuticals, Inc. | Microcrystalline y receptor agonists |
| HUE036066T2 (hu) | 2010-12-16 | 2018-06-28 | Novo Nordisk As | GLP-1 agonistát és N-(8-(2-hidroxibenzoil)amino)kaprilsav sóját tartalmazó szilárd készítmények |
| HRP20181447T1 (hr) | 2012-03-22 | 2018-11-02 | Novo Nordisk A/S | Pripravci glp-1 peptida i njihova priprava |
| MY172578A (en) | 2013-05-02 | 2019-12-03 | Novo Nordisk As | Oral dosing of glp-1 compounds |
| EP2842965A1 (en) | 2013-09-03 | 2015-03-04 | Gubra ApS | Neuromedin U analogs comprising serum albumin binding amino acid residue |
| WO2015073878A1 (en) * | 2013-11-15 | 2015-05-21 | Ur Diet, Llc | Real-time satiety biofeedback |
| PT3068421T (pt) * | 2013-11-15 | 2019-07-11 | Novo Nordisk As | Compostos de pyy eletivo e usos dos mesmos |
| EP3068795B1 (en) | 2013-11-15 | 2019-03-06 | Novo Nordisk A/S | Hpyy(1-36) having a beta-homoarginine substitution at position 35 |
| RS59026B1 (sr) | 2013-11-15 | 2019-08-30 | Novo Nordisk As | Selektivna pyy jedinjenja i njihova upotreba |
| US20240100450A9 (en) * | 2014-01-17 | 2024-03-28 | Repligen Corporation | Sterilizing chromatography columns |
| KR102393642B1 (ko) | 2014-01-17 | 2022-05-03 | 리플리겐 코포레이션 | 크로마토그래피 컬럼 살균 |
| EP3145523A4 (en) * | 2014-05-21 | 2018-02-21 | President and Fellows of Harvard College | Ras inhibitory peptides and uses thereof |
| CA2988500A1 (en) * | 2015-06-12 | 2016-12-15 | Novo Nordisk A/S | Selective pyy compounds and uses thereof |
| RS64643B1 (sr) | 2018-02-02 | 2023-10-31 | Novo Nordisk As | Čvrste kompozicije koje sadrže glp-1 agonist i so n-(8-(2-hidroksibenzoil)amino)kaprilne kiseline i lubrikant |
| TW202535916A (zh) | 2018-11-01 | 2025-09-16 | 美商美國禮來大藥廠 | 蛋白質酪胺酸-酪胺酸類似物及其使用方法 |
| GB201908426D0 (en) * | 2019-06-12 | 2019-07-24 | Imp College Innovations Ltd | Appetite suppressing compounds |
| MX2022013024A (es) * | 2020-04-17 | 2023-03-15 | I2O Therapeutics Inc | Analogos del peptido tirosina tirosina (pyy) de accion prolongada y metodos de uso de los mismos. |
| EP4329812A1 (en) | 2021-04-27 | 2024-03-06 | Aardvark Therapeutics Inc. | Combination of bitter receptor agonist and gut-signaling compound |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2275207C2 (ru) * | 2000-12-14 | 2006-04-27 | Амилин Фармасьютикалз, Инк. | Способ снижения доступности питательного вещества, способ подавления аппетита |
| AU2004273573B2 (en) * | 2003-09-19 | 2010-04-22 | Novo Nordisk A/S | Albumin-binding derivatives of therapeutic peptides |
| JP5638177B2 (ja) * | 2004-02-11 | 2014-12-10 | アミリン・ファーマシューティカルズ, リミテッド・ライアビリティ・カンパニーAmylin Pharmaceuticals, Llc | 膵臓ポリペプチドファミリーモチーフおよびそのモチーフを含むポリペプチド |
| MXPA06010345A (es) * | 2004-03-17 | 2007-06-19 | 7Tm Pharma As | Agonistas de receptor selectivo de y4 para intervenciones terapeuticas. |
| AU2005261740A1 (en) * | 2004-07-08 | 2006-01-19 | Novo Nordisk A/S | Polypeptide protracting tags comprising a tetrazole moiety |
| CN101222942A (zh) * | 2005-07-18 | 2008-07-16 | 诺沃-诺迪斯克有限公司 | 用于治疗肥胖的肽 |
-
2009
- 2009-05-18 AU AU2009248041A patent/AU2009248041B2/en not_active Ceased
- 2009-05-18 KR KR1020107027495A patent/KR20110017874A/ko not_active Withdrawn
- 2009-05-18 WO PCT/EP2009/055989 patent/WO2009138511A1/en not_active Ceased
- 2009-05-18 RU RU2010149474/04A patent/RU2504550C2/ru not_active IP Right Cessation
- 2009-05-18 BR BRPI0912615A patent/BRPI0912615A2/pt not_active Application Discontinuation
- 2009-05-18 CA CA2723855A patent/CA2723855A1/en not_active Withdrawn
- 2009-05-18 MX MX2010011845A patent/MX2010011845A/es not_active Application Discontinuation
- 2009-05-18 JP JP2011508945A patent/JP2011520847A/ja not_active Withdrawn
- 2009-05-18 CN CN2009801173043A patent/CN102027007A/zh not_active Withdrawn
- 2009-05-18 US US12/993,015 patent/US20110275559A1/en not_active Abandoned
- 2009-05-18 EP EP09745843A patent/EP2279204A1/en not_active Withdrawn
-
2010
- 2010-10-20 IL IL208836A patent/IL208836A0/en unknown