JP2011509305A - A2arアゴニストによる神経障害性疼痛の髄腔内治療 - Google Patents

A2arアゴニストによる神経障害性疼痛の髄腔内治療 Download PDF

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JP2011509305A
JP2011509305A JP2010542368A JP2010542368A JP2011509305A JP 2011509305 A JP2011509305 A JP 2011509305A JP 2010542368 A JP2010542368 A JP 2010542368A JP 2010542368 A JP2010542368 A JP 2010542368A JP 2011509305 A JP2011509305 A JP 2011509305A
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alkyl
alkylene
aryl
heteroaryl
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JP2011509305A5 (https=
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リンダ ワトキンズ
リサ ローラム
マーク ハッチンソン
ロバート トンプソン
アンソニー ボーグルホウル
フランク シュミットマン
ジェイソン リーガー
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PGxHealth LLC
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PGxHealth LLC
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)
JP2010542368A 2008-01-09 2009-01-09 A2arアゴニストによる神経障害性疼痛の髄腔内治療 Pending JP2011509305A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1991208P 2008-01-09 2008-01-09
PCT/US2009/030565 WO2009089425A1 (en) 2008-01-09 2009-01-09 Intrathecal treatment of neuropathic pain with a2ar agonists

Publications (2)

Publication Number Publication Date
JP2011509305A true JP2011509305A (ja) 2011-03-24
JP2011509305A5 JP2011509305A5 (https=) 2012-02-09

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JP2010542368A Pending JP2011509305A (ja) 2008-01-09 2009-01-09 A2arアゴニストによる神経障害性疼痛の髄腔内治療

Country Status (10)

Country Link
US (1) US20090181920A1 (https=)
EP (1) EP2240020A4 (https=)
JP (1) JP2011509305A (https=)
CN (1) CN101938904A (https=)
AU (1) AU2009204084A1 (https=)
BR (1) BRPI0907248A2 (https=)
CA (1) CA2711495A1 (https=)
EA (1) EA201001135A1 (https=)
IL (1) IL206801A0 (https=)
WO (1) WO2009089425A1 (https=)

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Also Published As

Publication number Publication date
WO2009089425A1 (en) 2009-07-16
US20090181920A1 (en) 2009-07-16
BRPI0907248A2 (pt) 2019-02-26
CA2711495A1 (en) 2009-07-16
CN101938904A (zh) 2011-01-05
EP2240020A1 (en) 2010-10-20
EA201001135A1 (ru) 2011-02-28
IL206801A0 (en) 2010-12-30
AU2009204084A1 (en) 2009-07-16
EP2240020A4 (en) 2011-05-11

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