JP2011509305A5 - - Google Patents

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Publication number
JP2011509305A5
JP2011509305A5 JP2010542368A JP2010542368A JP2011509305A5 JP 2011509305 A5 JP2011509305 A5 JP 2011509305A5 JP 2010542368 A JP2010542368 A JP 2010542368A JP 2010542368 A JP2010542368 A JP 2010542368A JP 2011509305 A5 JP2011509305 A5 JP 2011509305A5
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JP
Japan
Prior art keywords
alkylene
alkyl
aryl
heteroaryl
cycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010542368A
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English (en)
Japanese (ja)
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JP2011509305A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2009/030565 external-priority patent/WO2009089425A1/en
Publication of JP2011509305A publication Critical patent/JP2011509305A/ja
Publication of JP2011509305A5 publication Critical patent/JP2011509305A5/ja
Pending legal-status Critical Current

Links

JP2010542368A 2008-01-09 2009-01-09 Ａ２ａｒアゴニストによる神経障害性疼痛の髄腔内治療 Pending JP2011509305A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1991208P 2008-01-09 2008-01-09
PCT/US2009/030565 WO2009089425A1 (en) 2008-01-09 2009-01-09 Intrathecal treatment of neuropathic pain with a2ar agonists

Publications (2)

Publication Number Publication Date
JP2011509305A JP2011509305A (ja) 2011-03-24
JP2011509305A5 true JP2011509305A5 (https=) 2012-02-09

Family

ID=40851205

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010542368A Pending JP2011509305A (ja) 2008-01-09 2009-01-09 Ａ２ａｒアゴニストによる神経障害性疼痛の髄腔内治療

Country Status (10)

Country Link
US (1) US20090181920A1 (https=)
EP (1) EP2240020A4 (https=)
JP (1) JP2011509305A (https=)
CN (1) CN101938904A (https=)
AU (1) AU2009204084A1 (https=)
BR (1) BRPI0907248A2 (https=)
CA (1) CA2711495A1 (https=)
EA (1) EA201001135A1 (https=)
IL (1) IL206801A0 (https=)
WO (1) WO2009089425A1 (https=)

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US20130123208A1 (en) * 2010-05-12 2013-05-16 The Regents of the University of Colorado, a body corporation Method of treating multiple sclerosis with adenosine receptor agonists
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EP2646454B1 (en) 2010-12-03 2015-07-08 Epizyme, Inc. 7-deazapurine modulators of histone methyltransferase, and methods of use thereof
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TWI674262B (zh) 2011-01-10 2019-10-11 美商英菲尼提製藥股份有限公司 製備異喹啉酮之方法及異喹啉酮之固體形式
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