JP2011507847A5 - - Google Patents
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- Publication number
- JP2011507847A5 JP2011507847A5 JP2010539482A JP2010539482A JP2011507847A5 JP 2011507847 A5 JP2011507847 A5 JP 2011507847A5 JP 2010539482 A JP2010539482 A JP 2010539482A JP 2010539482 A JP2010539482 A JP 2010539482A JP 2011507847 A5 JP2011507847 A5 JP 2011507847A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- alkyl
- dba
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 CC(C)(C)*C(c(cc1*C(c2ccc(C)cc2I)=O)ccc1Oc1c(C)cc(CC(O)=O)c(N)c1)=O Chemical compound CC(C)(C)*C(c(cc1*C(c2ccc(C)cc2I)=O)ccc1Oc1c(C)cc(CC(O)=O)c(N)c1)=O 0.000 description 4
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US843307P | 2007-12-19 | 2007-12-19 | |
| US61/008,433 | 2007-12-19 | ||
| PCT/US2008/013833 WO2009085177A1 (en) | 2007-12-19 | 2008-12-18 | Phenyl acetic acid derivatives as inflammation modulators |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011507847A JP2011507847A (ja) | 2011-03-10 |
| JP2011507847A5 true JP2011507847A5 (OSRAM) | 2011-12-22 |
| JP5437267B2 JP5437267B2 (ja) | 2014-03-12 |
Family
ID=40564868
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010539482A Expired - Fee Related JP5437267B2 (ja) | 2007-12-19 | 2008-12-18 | 炎症モジュレーターとしてのフェニル酢酸誘導体 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US8183293B2 (OSRAM) |
| EP (1) | EP2231595B1 (OSRAM) |
| JP (1) | JP5437267B2 (OSRAM) |
| KR (1) | KR20100102668A (OSRAM) |
| CN (1) | CN101903338A (OSRAM) |
| AR (1) | AR071279A1 (OSRAM) |
| AU (1) | AU2008343924B2 (OSRAM) |
| BR (1) | BRPI0821197A2 (OSRAM) |
| CA (1) | CA2707789A1 (OSRAM) |
| CL (1) | CL2008003832A1 (OSRAM) |
| CO (1) | CO6321234A2 (OSRAM) |
| CR (1) | CR11572A (OSRAM) |
| EA (1) | EA201001029A1 (OSRAM) |
| ES (1) | ES2471919T3 (OSRAM) |
| IL (1) | IL206069A0 (OSRAM) |
| MA (1) | MA32013B1 (OSRAM) |
| PE (1) | PE20091526A1 (OSRAM) |
| TN (1) | TN2010000223A1 (OSRAM) |
| TW (1) | TW200940051A (OSRAM) |
| WO (1) | WO2009085177A1 (OSRAM) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2457900A1 (en) | 2010-11-25 | 2012-05-30 | Almirall, S.A. | New pyrazole derivatives having CRTh2 antagonistic behaviour |
| JP2015500326A (ja) | 2011-12-16 | 2015-01-05 | アトピックス テラピューティクス リミテッド | 好酸球性食道炎の治療のためのｃｒｔｈ２拮抗薬およびプロトンポンプ阻害薬の組み合わせ |
| US9974759B2 (en) * | 2013-05-31 | 2018-05-22 | Indiana University Research And Technology Corporation | Beta 2 adrenoceptor antagonists for treating orthostatic hypotension |
| US20180021302A1 (en) | 2015-02-13 | 2018-01-25 | Institut National De La Sante Et De La Recherche Medicale (Inserm) | Ptgdr-1 and/or ptgdr-2 antagonists for preventing and/or treating systemic lupus erythematosus |
| DK3433234T3 (da) | 2016-03-22 | 2022-01-03 | Merck Sharp & Dohme | Allosteriske modulatorer af nicotinacetylcholinreceptorer |
| ES2733477T3 (es) * | 2017-07-04 | 2019-11-29 | Fis Fabbrica Italiana Sintetici Spa | Procedimiento eficaz para la preparación de sitagliptina a través de una preparación muy eficaz del intermedio ácido 2,4,5-trifluorofenilacético |
Family Cites Families (41)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8704158D0 (en) | 1987-02-23 | 1987-04-01 | Wellcome Found | Substituted hydantoin compounds |
| US5849780A (en) | 1992-01-30 | 1998-12-15 | Sanofi | 1-benzenesulfonyl-1-1,3-dihydroindol-2-one derivatives, their preparation and pharmaceutical compositions in which they are present |
| AU7006094A (en) | 1993-06-30 | 1995-01-24 | Wellcome Foundation Limited, The | Anti-atherosclerotic diaryl compounds |
| US5545669A (en) | 1994-06-02 | 1996-08-13 | Adams; Jerry L. | Anti-inflammatory compounds |
| US5962682A (en) | 1994-12-20 | 1999-10-05 | Hoffmann-La Roche Inc. | Aryl- and hetaryl-sulfonamide derivatives, their preparation and their use as endothelin antagonists |
| DK0929547T3 (da) | 1996-09-12 | 2003-03-10 | Schering Ag | Benzamidinderivater substitueret af cykliske aminosyrederivater eller cykliske hydroxysyrederivater og deres anvendelse som antikoagulantia |
| US6008234A (en) | 1996-09-12 | 1999-12-28 | Berlex Laboratories, Inc. | Benzamidine derivatives substituted by cyclic amino acid and cyclic hydroxy acid derivatives and their use as anti-coagulants |
| TW523506B (en) | 1996-12-18 | 2003-03-11 | Ono Pharmaceutical Co | Sulfonamide or carbamide derivatives and drugs containing the same as active ingredients |
| JPH11202458A (ja) | 1998-01-16 | 1999-07-30 | Fuji Photo Film Co Ltd | ハロゲン化銀写真感光材料 |
| US5929250A (en) | 1997-01-23 | 1999-07-27 | Smithkline Beecham Corporation | IL-8 receptor antagonists |
| JP2002512997A (ja) | 1998-04-29 | 2002-05-08 | バーテックス ファーマシューティカルズ インコーポレイテッド | Ｉｍｐｄｈ酵素のインヒビター |
| AR023659A1 (es) | 1998-09-18 | 2002-09-04 | Vertex Pharma | Un compuesto inhibidor de p38, una composicion farmaceutica que lo comprende y el uso de dicha composicion en el tratamiento y prevencion de estados patologicos |
| US6248739B1 (en) | 1999-01-08 | 2001-06-19 | Pharmacia & Upjohn Company | Quinolinecarboxamides as antiviral agents |
| OA11839A (en) | 1999-03-01 | 2005-08-23 | Pfizer Prod Inc | Oxamic acids and derivatives as thyroid receptor ligands. |
| AU2825000A (en) | 1999-03-10 | 2000-09-28 | Shionogi & Co., Ltd. | Medicinal compositions with (2.2.1) and (3.1.1) bicycloskeleton antagonistic to both of pgd2/txa2 receptors |
| JP3486408B2 (ja) | 1999-08-23 | 2004-01-13 | 株式会社ビー・エム・エル | 物質のヒトプロスタグランジンｄ２受容体に対する性質の同定方法 |
| US6531291B1 (en) | 1999-11-10 | 2003-03-11 | The Trustees Of Columbia University In The City Of New York | Antimicrobial activity of gemfibrozil and related compounds and derivatives and metabolites thereof |
| AU2001236605A1 (en) | 2000-02-01 | 2001-08-14 | Cor Therapeutics, Inc. | Indole and benzimidazole inhibitors of factor xa |
| US20010047027A1 (en) | 2000-04-12 | 2001-11-29 | Marc Labelle | Prostaglandin D2 receptor antagonists |
| AU2001260627A1 (en) | 2000-06-02 | 2001-12-17 | Shionogi And Co., Ltd. | Drug composition antagonistic to both pgd2/txa2 receptors |
| US6878522B2 (en) | 2000-07-07 | 2005-04-12 | Baiyong Li | Methods for the identification of compounds useful for the treatment of disease states mediated by prostaglandin D2 |
| AU2002229611A1 (en) | 2000-12-08 | 2002-06-18 | Institut National De La Sante Et De La Recherche Medicale (Inserm) | Use of active compounds capable of modulating the intracellular pathway triggered by the dp receptor in langerhans cells |
| CA2433100A1 (en) | 2000-12-27 | 2002-07-04 | Helmut Haning | Indole derivatives as ligands of thyroid receptors |
| EP1395590B1 (en) | 2001-05-23 | 2006-09-27 | Merck Frosst Canada & Co. | Dihydropyrrolo¬1,2-a|indole and tetrahydropyrido¬1,2-a|indole derivatives as prostaglandin d2 receptor antagonists |
| EP1431267A4 (en) | 2001-08-09 | 2004-12-22 | Ono Pharmaceutical Co | COMPOUNDS DERIVED FROM CARBOXYLIC ACID AND MEDICAMENTS COMPRISING SUCH COMPOUNDS AS ACTIVE INGREDIENT |
| SE0200411D0 (sv) | 2002-02-05 | 2002-02-05 | Astrazeneca Ab | Novel use |
| SE0200356D0 (sv) | 2002-02-05 | 2002-02-05 | Astrazeneca Ab | Novel use |
| CA2479352A1 (en) | 2002-03-19 | 2003-09-25 | Ono Pharmaceutical Co., Ltd. | Carboxylic acid compound and a pharmaceutical agent comprising the compound as an active ingredient |
| WO2003097042A1 (en) | 2002-05-16 | 2003-11-27 | Shionogi & Co., Ltd. | Pgd2 receptor antagonist |
| US7534897B2 (en) | 2002-05-16 | 2009-05-19 | Shionogi & Co., Ltd. | Indole arylsulfonaimide compounds exhibiting PGD 2 receptor antagonism |
| GB2388540A (en) | 2002-05-17 | 2003-11-19 | Bayer Ag | New use of Ramatroban |
| SE0201635D0 (sv) | 2002-05-30 | 2002-05-30 | Astrazeneca Ab | Novel compounds |
| TW200307542A (en) | 2002-05-30 | 2003-12-16 | Astrazeneca Ab | Novel compounds |
| GB0224557D0 (en) | 2002-10-22 | 2002-11-27 | Glaxo Group Ltd | Novel compounds |
| EP1585511B1 (en) | 2002-12-20 | 2013-01-23 | Amgen Inc. | Asthma and allergic inflammation modulators |
| WO2005054176A1 (en) | 2003-11-25 | 2005-06-16 | Eli Lilly And Company | Peroxisome proliferator activated receptor modulators |
| EP1937632A1 (en) * | 2005-10-06 | 2008-07-02 | Astra Zeneca AB | Novel compounds |
| JP5069752B2 (ja) * | 2006-12-15 | 2012-11-07 | グラクソ グループ リミテッド | Ｅｐ４受容体アゴニストとしてのベンズアミド誘導体 |
| US7960567B2 (en) | 2007-05-02 | 2011-06-14 | Amgen Inc. | Compounds and methods useful for treating asthma and allergic inflammation |
| KR20120038544A (ko) | 2009-07-31 | 2012-04-23 | 판미라 파마슈티칼스, 엘엘씨 | Ｄｐ2 수용체 길항제의 안과용 약학 조성물 |
| CN102596193A (zh) | 2009-07-31 | 2012-07-18 | 潘米拉制药公司 | Dp2受体拮抗的皮肤调配物 |
-
2008
- 2008-12-18 EA EA201001029A patent/EA201001029A1/ru unknown
- 2008-12-18 KR KR1020107015813A patent/KR20100102668A/ko not_active Withdrawn
- 2008-12-18 BR BRPI0821197-3A patent/BRPI0821197A2/pt not_active IP Right Cessation
- 2008-12-18 US US12/317,066 patent/US8183293B2/en active Active
- 2008-12-18 EP EP08867490.8A patent/EP2231595B1/en active Active
- 2008-12-18 AU AU2008343924A patent/AU2008343924B2/en not_active Ceased
- 2008-12-18 JP JP2010539482A patent/JP5437267B2/ja not_active Expired - Fee Related
- 2008-12-18 ES ES08867490.8T patent/ES2471919T3/es active Active
- 2008-12-18 CN CN2008801215268A patent/CN101903338A/zh active Pending
- 2008-12-18 CA CA2707789A patent/CA2707789A1/en not_active Abandoned
- 2008-12-18 WO PCT/US2008/013833 patent/WO2009085177A1/en not_active Ceased
- 2008-12-19 PE PE2008002152A patent/PE20091526A1/es not_active Application Discontinuation
- 2008-12-19 AR ARP080105608A patent/AR071279A1/es not_active Application Discontinuation
- 2008-12-19 CL CL2008003832A patent/CL2008003832A1/es unknown
- 2008-12-19 TW TW097149926A patent/TW200940051A/zh unknown
-
2010
- 2010-05-20 TN TN2010000223A patent/TN2010000223A1/fr unknown
- 2010-05-30 IL IL206069A patent/IL206069A0/en unknown
- 2010-07-14 MA MA33012A patent/MA32013B1/fr unknown
- 2010-07-19 CR CR11572A patent/CR11572A/es not_active Application Discontinuation
- 2010-07-19 CO CO10087808A patent/CO6321234A2/es not_active Application Discontinuation
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