IL206069A0 - Phenyl acetic acid derivatives as inflammation modulators - Google Patents

Phenyl acetic acid derivatives as inflammation modulators

Info

Publication number
IL206069A0
IL206069A0 IL206069A IL20606910A IL206069A0 IL 206069 A0 IL206069 A0 IL 206069A0 IL 206069 A IL206069 A IL 206069A IL 20606910 A IL20606910 A IL 20606910A IL 206069 A0 IL206069 A0 IL 206069A0
Authority
IL
Israel
Prior art keywords
acetic acid
acid derivatives
phenyl acetic
inflammation modulators
modulators
Prior art date
Application number
IL206069A
Other languages
English (en)
Original Assignee
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc filed Critical Amgen Inc
Publication of IL206069A0 publication Critical patent/IL206069A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/22Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms
    • C07C311/29Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/15Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/21Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/02Systems containing only non-condensed rings with a three-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/04Systems containing only non-condensed rings with a four-membered ring

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Otolaryngology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
IL206069A 2007-12-19 2010-05-30 Phenyl acetic acid derivatives as inflammation modulators IL206069A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US843307P 2007-12-19 2007-12-19
PCT/US2008/013833 WO2009085177A1 (en) 2007-12-19 2008-12-18 Phenyl acetic acid derivatives as inflammation modulators

Publications (1)

Publication Number Publication Date
IL206069A0 true IL206069A0 (en) 2010-11-30

Family

ID=40564868

Family Applications (1)

Application Number Title Priority Date Filing Date
IL206069A IL206069A0 (en) 2007-12-19 2010-05-30 Phenyl acetic acid derivatives as inflammation modulators

Country Status (20)

Country Link
US (1) US8183293B2 (OSRAM)
EP (1) EP2231595B1 (OSRAM)
JP (1) JP5437267B2 (OSRAM)
KR (1) KR20100102668A (OSRAM)
CN (1) CN101903338A (OSRAM)
AR (1) AR071279A1 (OSRAM)
AU (1) AU2008343924B2 (OSRAM)
BR (1) BRPI0821197A2 (OSRAM)
CA (1) CA2707789A1 (OSRAM)
CL (1) CL2008003832A1 (OSRAM)
CO (1) CO6321234A2 (OSRAM)
CR (1) CR11572A (OSRAM)
EA (1) EA201001029A1 (OSRAM)
ES (1) ES2471919T3 (OSRAM)
IL (1) IL206069A0 (OSRAM)
MA (1) MA32013B1 (OSRAM)
PE (1) PE20091526A1 (OSRAM)
TN (1) TN2010000223A1 (OSRAM)
TW (1) TW200940051A (OSRAM)
WO (1) WO2009085177A1 (OSRAM)

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EP2457900A1 (en) 2010-11-25 2012-05-30 Almirall, S.A. New pyrazole derivatives having CRTh2 antagonistic behaviour
MX2014007239A (es) 2011-12-16 2014-08-08 Atopix Therapeutics Ltd Combinacion de un antagonista crth2 y un inhibidor de bomba de proton para el tratamiento de esofagitis eosinofilica.
US9974759B2 (en) * 2013-05-31 2018-05-22 Indiana University Research And Technology Corporation Beta 2 adrenoceptor antagonists for treating orthostatic hypotension
JP6770522B2 (ja) * 2015-02-13 2020-10-14 アンスティチュ ナショナル ドゥ ラ サンテ エ ドゥ ラ ルシェルシュ メディカル 全身性エリテマトーデスを予防し、及び/又は、治療するためのptgdr−1及び/又はptgdr−2アンタゴニスト
MY195948A (en) 2016-03-22 2023-02-27 Merck Sharp & Dohme Allosteric Modulators of Nicotinic Acetylcholine Receptors
EP3424927B1 (en) 2017-07-04 2019-04-17 F.I.S.- Fabbrica Italiana Sintetici S.p.A. Efficient process for the preparation of sitagliptin through a very effective preparation of the intermediate 2,4,5-trifluorophenylacetic acid

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IL110159A0 (en) 1993-06-30 1994-10-07 Wellcome Found Diaryl compounds, their preparation and pharmaceutical compositions containing them
US5545669A (en) 1994-06-02 1996-08-13 Adams; Jerry L. Anti-inflammatory compounds
PT799206E (pt) 1994-12-20 2003-01-31 Hoffmann La Roche Derivados de aril- e heteroaril-sulfonamida processo para a sua preparacao e sua utilizacao como antagonistas da endotelina
US6008234A (en) 1996-09-12 1999-12-28 Berlex Laboratories, Inc. Benzamidine derivatives substituted by cyclic amino acid and cyclic hydroxy acid derivatives and their use as anti-coagulants
CN1234798A (zh) 1996-09-12 1999-11-10 舍林股份公司 环状氨基酸和环状羟基羧酸衍生物取代的苄脒衍生物和它们用作抗凝剂的用途
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JP2013500978A (ja) 2009-07-31 2013-01-10 パンミラ ファーマシューティカルズ,エルエルシー. Dp2受容体アンタゴニストの眼の医薬組成物
SG177736A1 (en) 2009-07-31 2012-02-28 Panmira Pharmaceuticals Llc Dermal formulations of dp2 receptor antagonists

Also Published As

Publication number Publication date
BRPI0821197A2 (pt) 2015-06-16
CR11572A (es) 2010-08-13
JP2011507847A (ja) 2011-03-10
TN2010000223A1 (en) 2011-11-11
MA32013B1 (fr) 2011-01-03
AU2008343924A1 (en) 2009-07-09
US8183293B2 (en) 2012-05-22
JP5437267B2 (ja) 2014-03-12
AU2008343924A2 (en) 2011-02-17
AU2008343924B2 (en) 2013-01-17
EP2231595B1 (en) 2014-04-23
WO2009085177A1 (en) 2009-07-09
KR20100102668A (ko) 2010-09-24
EA201001029A1 (ru) 2011-06-30
EP2231595A1 (en) 2010-09-29
TW200940051A (en) 2009-10-01
US20090275659A1 (en) 2009-11-05
CN101903338A (zh) 2010-12-01
CA2707789A1 (en) 2009-07-09
PE20091526A1 (es) 2009-11-01
AR071279A1 (es) 2010-06-09
CL2008003832A1 (es) 2010-03-26
CO6321234A2 (es) 2011-09-20
ES2471919T3 (es) 2014-06-27

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