JP2011500596A5 - - Google Patents

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Publication number
JP2011500596A5
JP2011500596A5 JP2010529085A JP2010529085A JP2011500596A5 JP 2011500596 A5 JP2011500596 A5 JP 2011500596A5 JP 2010529085 A JP2010529085 A JP 2010529085A JP 2010529085 A JP2010529085 A JP 2010529085A JP 2011500596 A5 JP2011500596 A5 JP 2011500596A5
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JP
Japan
Prior art keywords
methyl
phenyl
triazin
trifluoromethyl
methylamino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2010529085A
Other languages
English (en)
Japanese (ja)
Other versions
JP5411867B2 (ja
JP2011500596A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2008/079525 external-priority patent/WO2009049165A1/en
Publication of JP2011500596A publication Critical patent/JP2011500596A/ja
Publication of JP2011500596A5 publication Critical patent/JP2011500596A5/ja
Application granted granted Critical
Publication of JP5411867B2 publication Critical patent/JP5411867B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2010529085A 2007-10-11 2008-10-10 新規sEH阻害剤およびそれらの使用 Expired - Fee Related JP5411867B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US97916407P 2007-10-11 2007-10-11
US60/979,164 2007-10-11
PCT/US2008/079525 WO2009049165A1 (en) 2007-10-11 2008-10-10 Novel seh inhibitors and their use

Publications (3)

Publication Number Publication Date
JP2011500596A JP2011500596A (ja) 2011-01-06
JP2011500596A5 true JP2011500596A5 (https=) 2011-11-24
JP5411867B2 JP5411867B2 (ja) 2014-02-12

Family

ID=40549593

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010529085A Expired - Fee Related JP5411867B2 (ja) 2007-10-11 2008-10-10 新規sEH阻害剤およびそれらの使用

Country Status (5)

Country Link
US (1) US8008483B2 (https=)
EP (1) EP2209376B1 (https=)
JP (1) JP5411867B2 (https=)
ES (1) ES2404580T3 (https=)
WO (1) WO2009049165A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7994317B2 (en) 2006-11-03 2011-08-09 GlaxoSmithKline, LLC sEH inhibitors and their use
JP5372943B2 (ja) 2007-10-11 2013-12-18 グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー 新規sEH阻害剤およびそれらの使用
MY152834A (en) 2009-08-18 2014-11-28 Multitest Elektronische Syst An elastic unit for clamping an electronic component and extending below an electronic component receiving volume of an align fixture
EP2567959B1 (en) 2011-09-12 2014-04-16 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2015003355A2 (en) * 2013-07-11 2015-01-15 Agios Pharmaceuticals, Inc. Therapeutically active compounds and their methods of use
SI3397631T1 (sl) * 2015-12-29 2022-01-31 Pfizer Inc. Substituirani 3-azabiciklo(3.1.0)heksani kot zaviralci ketoheksokinaze
EA035363B1 (ru) * 2016-11-17 2020-06-02 Пфайзер Инк. Замещенные 3-азабицикло[3.1.0]гексаны в качестве ингибиторов кетогексокиназы
EP4308555A4 (en) * 2021-03-18 2025-07-30 Sironax Ltd RECEPTOR-INTERACTING PROTEIN-1 INHIBITORS, PREPARATIONS AND USES THEREOF

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1255704B (it) * 1992-09-30 1995-11-10 Boehringer Mannheim Italia Ammine eterocicliche utili nella terapia dell'asma e dell'infiammazione delle vie aeree
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
KR100875362B1 (ko) 2002-02-05 2008-12-22 아스텔라스세이야쿠 가부시키가이샤 2,4,6-트리아미노-1,3,5-트리아진 유도체
US20050197350A1 (en) 2003-03-31 2005-09-08 Taisho Pharmaceutical Co., Ltd. Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof
WO2005028467A1 (en) 2003-09-15 2005-03-31 Anadys Pharmaceuticals, Inc. Antibacterial 3,5-diaminopiperidine-substitute aromatic and heteroaromatic compounds
JP2007126454A (ja) * 2005-10-06 2007-05-24 Taisho Pharmaceut Co Ltd アニリド誘導体
WO2007098352A2 (en) * 2006-02-16 2007-08-30 Boehringer Ingelheim International Gmbh Substituted pyridineamide compounds useful as soluble epoxide hydrolase inhibitors
CA2643859A1 (en) * 2006-03-10 2007-09-20 Boehringer Ingelheim International Gmbh Soluble epoxide hydrolase inhibitors and methods of using same
AR059826A1 (es) * 2006-03-13 2008-04-30 Univ California Inhibidores de urea conformacionalmente restringidos de epoxido hidrolasa soluble
US7994317B2 (en) * 2006-11-03 2011-08-09 GlaxoSmithKline, LLC sEH inhibitors and their use
JP5372943B2 (ja) 2007-10-11 2013-12-18 グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー 新規sEH阻害剤およびそれらの使用
WO2009049154A1 (en) 2007-10-11 2009-04-16 Smithkline Beecham Corporation NOVEL sEH INHIBITORS AND THEIR USE
US20120009151A1 (en) * 2007-12-21 2012-01-12 Progenics Pharmaceuticals, Inc. Triazines And Related Compounds Having Antiviral Activity, Compositions And Methods Thereof

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