JP2011225463A - Blood-sucking flying insect pest-controlling agent and method for protecting animal - Google Patents
Blood-sucking flying insect pest-controlling agent and method for protecting animal Download PDFInfo
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Classifications
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
Description
本発明は、犬や猫などの愛玩動物、牛、豚、鶏などの家畜や家禽に対する飛翔性吸血害虫防除剤およびこれを用いてなる動物の防護方法に関する。 The present invention relates to a flying blood-sucking pest control agent for pets such as dogs and cats, livestock such as cattle, pigs and chickens, and poultry, and a method for protecting animals using the same.
犬や猫などの愛玩動物、牛、豚、鶏などの家畜や家禽類は屋外で飼育されることが多く、また、主として屋内で飼育されている場合であっても屋外に出る機会も多く、特に春から秋にかけての高温時期には蚊に代表される飛翔性吸血害虫による影響を受けることが多い。
かかる飛翔性吸血害虫から動物を守る方法として、従来、蚊取り線香や蒸散性殺虫成分を含有したマットなどを飼育小屋などに配置する方法が知られているが、この方法はその効果の範囲が飼育小屋周辺などの極めて限定された場所に限られていた。
しかし、このような動物は飼育小屋を離れて動き回ることも多く、上記のような方法では効果的に蚊などの飛翔性吸血害虫から動物への接触、吸血を抑制し、動物を防護することは十分ではなかった。
一方で、動物の体表面に寄生するノミやダニなどの駆除を目的とした滴下剤と呼ばれるノミやダニなどの防除剤については、例えば特許文献１に記載されているが、同特許文献１では動物の体表面に寄生することのない蚊などの飛翔性吸血害虫に対する具体的効果についての記載はなく、依然として飛翔性吸血害虫による吸血からこのような動物を防護する方法は未知のままであった。
Pets such as dogs and cats, livestock and poultry such as cattle, pigs, and chickens are often raised outdoors, and even if they are mainly raised indoors, there are many opportunities to go outdoors. In particular, it is often affected by flying blood-sucking pests such as mosquitoes at high temperatures from spring to autumn.
As a method of protecting animals from such flying blood-sucking pests, conventionally, a method of arranging a mosquito-repellent incense stick or a mat containing a transpirationable insecticide component in a breeding shed is known. It was limited to very limited places such as the surroundings.
However, these animals often move away from their sheds, and the above methods can effectively prevent mosquitoes and other flying blood-sucking insects from touching and sucking blood and protecting them. It was not enough.
On the other hand, fleas and mites control agents called dripping agents for the purpose of controlling fleas and ticks that parasitize on the body surface of animals are described in Patent Document 1, for example. There is no description of specific effects on flying blood-sucking pests such as mosquitoes that do not infest the animal's body surface, and how to protect such animals from blood-feeding by flying blood-sucking insects remains unknown .
本発明は、飛翔性吸血害虫による吸血から動物を防護するための飛翔性吸血害虫防除剤およびこれを用いてなる動物の防護方法に関するものである。 The present invention relates to a flying blood-sucking insect control agent for protecting an animal from blood sucking by a flying blood-sucking insect and a method for protecting an animal using the same.
本発明者は、前記したような犬や猫などの愛玩動物、牛、豚、鶏などの家畜や家禽類を飛翔性吸血害虫による吸血から守る効果的な方法の開発を鋭意検討した結果、有機溶剤中に、３−フェノキシベンジル ２，２−ジメチル−３−（２−メチルプロプ−１−エニル）シクロプロパンカルボキシラートおよび／またはジョチュウギクエキスを有効成分として含有してなることを特徴とする飛翔性吸血害虫防除剤を、動物の体表面に部分的に付着処理することにより動物に対する飛翔性吸血害虫による吸血を阻害し、防護することができることを見出し、本発明を完成した。 The present inventor has intensively studied the development of an effective method for protecting domestic animals such as pets such as dogs and cats, domestic animals and poultry such as cattle, pigs and chickens from blood-feeding insects. A flight characterized in that 3-phenoxybenzyl 2,2-dimethyl-3- (2-methylprop-1-enyl) cyclopropanecarboxylate and / or jojoba extract is contained as an active ingredient in a solvent. The present invention has been completed by discovering that a blood-sucking insect pest control agent can be partially adhered to the body surface of the animal to inhibit and protect the animal from sucking blood by a flying blood-sucking insect.
すなわち、本発明は以下の［１］〜［６］に関する。
［１］ 有機溶剤中に、３−フェノキシベンジル ２，２−ジメチル−３−（２−メチルプロプ−１−エニル）シクロプロパンカルボキシラートおよび／またはジョチュウギクエキスを有効成分として含有してなることを特徴とする飛翔性吸血害虫防除剤。
［２］ ピリプロキシフェンをさらに含有してなる前記１に記載の飛翔性吸血害虫防除剤。
［３］ 有機溶剤がジエチレングリコールモノエチルエーテルであることを特徴とする前記１または２に記載の飛翔性吸血害虫防除剤。
［４］ 有機溶剤がケロシンであることを特徴とする前記１または２に記載の飛翔性吸血害虫防除剤。
［５］ 有機溶剤がカプリル酸トリグリセライドであることを特徴とする前記１または２に記載の飛翔性吸血害虫防除剤。
［６］ 前記１または２に記載の飛翔性吸血害虫防除剤を、動物の体表面に部分的に付着処理し、飛翔性吸血害虫による吸血を阻害してなることを特徴とする動物の防護方法。
That is, the present invention relates to the following [1] to [6].
[1] An organic solvent containing 3-phenoxybenzyl 2,2-dimethyl-3- (2-methylprop-1-enyl) cyclopropanecarboxylate and / or chrysanthemum extract as an active ingredient. Characteristic flying insect-feeding insecticide.
[2] The flying blood-sucking pest control agent according to 1, further comprising pyriproxyfen.
[3] The flying blood-sucking insecticide as described in 1 or 2 above, wherein the organic solvent is diethylene glycol monoethyl ether.
[4] The flying blood-sucking insecticide as described in 1 or 2 above, wherein the organic solvent is kerosene.
[5] The flying blood-sucking insecticide as described in 1 or 2 above, wherein the organic solvent is caprylic acid triglyceride.
[6] A method for protecting an animal comprising the step of adhering the flying blood-sucking pest control agent according to 1 or 2 to the surface of an animal to inhibit blood feeding by the flying blood-sucking insect. .
本発明の飛翔性吸血害虫防除剤を、動物の体表面に部分的に付着処理することにより、長期間にわたって飛翔性吸血害虫による吸血を阻害し、防護することができる。 By applying the flying blood-sucking pest control agent of the present invention to the surface of the animal partly, the blood sucking by the flying blood-sucking insect can be inhibited and protected over a long period of time.
本発明の飛翔性吸血害虫防除剤の適用対象となる動物としては、家畜、家禽、愛玩動物などの各種動物、特に哺乳類、鳥類などの動物が挙げられ、より具体的には、犬、猫、ウサギ、ハムスター、フェレットなどの愛玩動物、牛、馬、豚、羊、山羊、鶏、家鴨、七面鳥などの家畜や家禽が挙げられる。 Examples of animals to which the flying blood-sucking pest control agent of the present invention is applied include various animals such as livestock, poultry and pets, particularly mammals and birds, and more specifically, dogs, cats, Examples include pets such as rabbits, hamsters and ferrets, and livestock and poultry such as cows, horses, pigs, sheep, goats, chickens, domestic duck, and turkeys.
本発明の飛翔性吸血害虫防除剤の適用対象となる飛翔性吸血害虫としては蚊が代表的であり、例えばアカイエカ、コガタアカイエカ、ネッタイイエカ等のイエカ類、ネッタイシマカ、ヒトスジシマカ等のヤブカ類、シナハマダラカ等のハマダラカ類などを挙げることができる。 The flying blood-sucking insect pests to which the flying blood-sucking insect-controlling agent of the present invention is applied are typically mosquitoes. And the like.
本発明の飛翔性吸血害虫防除剤は、有機溶剤中に、有効成分として３−フェノキシベンジル ２，２−ジメチル−３−（２−メチルプロプ−１−エニル）シクロプロパンカルボキシラートおよび／またはジョチュウギクエキスを含有してなるものである。
ここで、３−フェノキシベンジル ２，２−ジメチル−３−（２−メチルプロプ−１−エニル）シクロプロパンカルボキシラートには種々の立体異性体が存在するが、本発明においては任意の活性な立体異性体またはその混合物が使用され、例えば、３−フェノキシベンジル （１Ｒ）−シス，トランス−２，２−ジメチル−３−（２−メチルプロプ−１−エニル）シクロプロパンカルボキシラート（一般名＝ｄ−フェノトリン）が使用される。
The flying blood-sucking insect pest control agent of the present invention comprises 3-phenoxybenzyl 2,2-dimethyl-3- (2-methylprop-1-enyl) cyclopropanecarboxylate and / or chrysanthemum as an active ingredient in an organic solvent. It contains an extract.
Here, various stereoisomers exist in 3-phenoxybenzyl 2,2-dimethyl-3- (2-methylprop-1-enyl) cyclopropanecarboxylate. In the present invention, any active stereoisomer is present. Or a mixture thereof, such as 3-phenoxybenzyl (1R) -cis, trans-2,2-dimethyl-3- (2-methylprop-1-enyl) cyclopropanecarboxylate (generic name = d-phenothrin). ) Is used.
かかる飛翔性吸血害虫防除剤において、その有効成分である３−フェノキシベンジル ２，２−ジメチル−３−（２−メチルプロプ−１−エニル）シクロプロパンカルボキシラートおよび／またはジョチュウギクエキスの含有量は、通常１〜８０質量％、好ましくは３〜６０質量％、更に好ましくは５〜４０質量％の範囲である。
尚、ジョチュウギクエキスはピレトリンＩ、ピレトリンII、ジャスモリンＩ、ジャスモリンII、シネリンＩ、シネリンIIなどの殺虫成分（まとめて総ピレトリンという）を通常３０〜７０質量％含有する混合物であるため、ジョチュウギクエキスを単独または併用して使用する場合には、総ピレトリンの量を基準として上記範囲内にあることが好ましい。
尚、有効成分としてジョチュウギクエキスを単独で使用する場合には、その有効成分量は、上記範囲内であっても総ピレトリンの量として１〜４０質量％、好ましくは１〜３０質量％、更に好ましくは２〜２５質量％程度の少ない量でも十分であり、３−フェノキシベンジル ２，２−ジメチル−３−（２−メチルプロプ−１−エニル）シクロプロパンカルボキシラートと併用する場合においても、ジョチュウギクエキスの使用量としては３０質量％以下の少量で併用することができる。
In the flying blood-sucking pest control agent, the content of 3-phenoxybenzyl 2,2-dimethyl-3- (2-methylprop-1-enyl) cyclopropanecarboxylate and / or chrysanthemum extract as the active ingredient is The range is usually 1 to 80% by mass, preferably 3 to 60% by mass, and more preferably 5 to 40% by mass.
In addition, Jochugi extract is a mixture containing usually 30 to 70% by mass of insecticidal components (collectively referred to as total pyrethrin) such as pyrethrin I, pyrethrin II, jasmolin I, jasmolin II, cinerin I, and cineline II. When a chrysanthemum extract is used alone or in combination, it is preferably within the above range based on the total amount of pyrethrin.
In addition, when using the licorice extract alone as an active ingredient, the amount of the active ingredient is 1 to 40% by mass, preferably 1 to 30% by mass as the total pyrethrin even within the above range. More preferably, a small amount of about 2 to 25% by mass is sufficient, and even when used in combination with 3-phenoxybenzyl 2,2-dimethyl-3- (2-methylprop-1-enyl) cyclopropanecarboxylate, As a usage-amount of a chrysanthemum extract, it can use together in a small amount of 30 mass% or less.
飛翔性吸血害虫防除剤は、前記した有効成分を有機溶剤に溶解してなるものである。
かかる目的で使用される有機溶剤としては、当該有効成分を溶解し、かつ動物に悪影響を与えないものであれば特に限定されることなく使用できる。
このような有機溶剤としては、例えばエタノール、イソプロパノール、ベンジルアルコールなどのアルコール類、プロピレングリコールなどのグリコール類、ジエチレングリコールモノメチルエーテル、ジエチレングリコールモノエチルエーテル、ジエチレングリコールモノブチルエーテルなどのグリコールエステル類、カプリル酸モノグリセライド、ジグリセライド、またはトリグリセライド、カプロン酸モノグリセライド、ジグリセライド、またはトリグリセライドなどの脂肪族カルボン酸のグリセライド類、ケロシン、炭酸プロピレンなどが代表的であり、また、大豆油、ヤシ油、パーム油、アマニ油、綿実油、ナタネ油、キリ油、ヒマシ油、オリーブ油、米糠油などの植物油が挙げられ、好ましくは、ジエチレングリコールモノエチルエーテル、ケロシン、カプリル酸トリグリセライドが用いられる。また、これらの有機溶剤の２種以上を混合して使用することもできる。
The flying blood-sucking pest control agent is obtained by dissolving the above-mentioned active ingredient in an organic solvent.
The organic solvent used for this purpose is not particularly limited as long as it dissolves the active ingredient and does not adversely affect animals.
Examples of such organic solvents include alcohols such as ethanol, isopropanol, and benzyl alcohol, glycols such as propylene glycol, glycol esters such as diethylene glycol monomethyl ether, diethylene glycol monoethyl ether, and diethylene glycol monobutyl ether, caprylic acid monoglyceride, and diglyceride. Or glycerides of aliphatic carboxylic acids such as triglyceride, caproic acid monoglyceride, diglyceride, or triglyceride, kerosene, propylene carbonate, etc., and soybean oil, coconut oil, palm oil, linseed oil, cottonseed oil, rapeseed And vegetable oils such as oil, tung oil, castor oil, olive oil and rice bran oil, preferably diethylene glycol monoethyl Ether, kerosene, caprylic acid triglyceride used. Also, two or more of these organic solvents can be mixed and used.
本発明の飛翔性吸血害虫防除剤は、基本的には前記したような有効成分が有機溶剤中に溶解されてなるものであるが、共力剤、安定剤、香料、他の生理活性物質が適宜含有されていてもよい。 The flying blood-sucking pest control agent of the present invention is basically one in which the active ingredient as described above is dissolved in an organic solvent, but a synergist, a stabilizer, a fragrance, and other physiologically active substances. It may be contained as appropriate.
共力剤としては、例えば、Ｎ−（２−エチルヘキシル）−１−イソプロピル−４−メチルビシクロ［２，２，２］オクト−５−エン−２，３−ジカルボキシイミド、Ｎ−（２−エチルヘキシル）ビシクロ［２，２，１］ヘプト−５−エン−２，３−ジカルボキシイミド（ＭＧＫ−２６４）、チオシアノ酢酸イソボルニル（ＩＢＴＡ）、ピペロニルブトキサイドなどが挙げられる。 Examples of the synergist include N- (2-ethylhexyl) -1-isopropyl-4-methylbicyclo [2,2,2] oct-5-ene-2,3-dicarboximide, N- (2- And ethylhexyl) bicyclo [2,2,1] hept-5-ene-2,3-dicarboximide (MGK-264), isobornyl thiocyanoacetate (IBTA), piperonyl butoxide, and the like.
安定剤としては、例えば、ブチルヒドロキシトルエン（ＢＨＴ）、ブチルヒドロキシアニソール（ＢＨＡ）、４，４’−チオビス（３−メチル−６−ｔ−ブチルフェノール）（ＴＢＭＢＰ）などが挙げられる。 Examples of the stabilizer include butylhydroxytoluene (BHT), butylhydroxyanisole (BHA), 4,4′-thiobis (3-methyl-6-tert-butylphenol) (TBMBP), and the like.
香料としては、シトロネラール、シトロネロール、リモネン等のテルペンまたはテルペン誘導体が挙げられる。 Examples of the fragrances include terpenes or terpene derivatives such as citronellal, citronellol, and limonene.
他の生理活性物質としては、例えば、ピリプロキシフェン、メトプレン等の昆虫成長調節剤が挙げられる。 Examples of other physiologically active substances include insect growth regulators such as pyriproxyfen and metoprene.
本発明の飛翔性吸血害虫防除剤を用いて飛翔性吸血害虫から動物を防護する方法としては、通常、動物の体表の一部に当該防除剤を滴下、塗布、噴霧などの方法により、動物の体表面に付着処理することにより行われる。
かかる付着処理方法は、対象とする動物の大きさによっても変わり、犬や猫などの小動物の場合には単に動物の体表に１〜数箇所に滴下するだけでも十分である。
施用量は、本発明の飛翔性吸血害虫防除剤中の有効成分含有量に依存するが、一般的には有効成分量として、動物の体重１ｋｇ当り、３〜５００ｍｇ、好ましくは１０〜４００ｍｇ、さらに好ましくは１５〜３５０ｍｇである。
As a method for protecting an animal from a flying blood-sucking pest using the flying blood-sucking pest control agent of the present invention, the animal is usually applied to a part of the body surface of the animal by dropping, coating, spraying, etc. This is done by attaching to the body surface.
Such an adhesion treatment method varies depending on the size of the target animal, and in the case of a small animal such as a dog or a cat, it is sufficient to simply drop it on the body surface of the animal at one to several places.
The application amount depends on the content of the active ingredient in the flying blood-sucking pest control agent of the present invention. Generally, the amount of the active ingredient is 3 to 500 mg, preferably 10 to 400 mg, preferably 1 to 400 mg per kg of the animal body weight. Preferably it is 15-350 mg.
以下、実施例にて本発明をより詳細に説明する。 Hereinafter, the present invention will be described in more detail with reference to examples.
実施例１：
ｄ−フェノトリン３０ｇ、ピリプロキシフェン０．６ｇ、ＢＨＴ０．０１ｇをジエチレングリコールモノエチルエーテル６９．９ｇに加え、本発明の防除剤１を作製した。
Example 1:
30 g of d-phenothrin, 0.6 g of pyriproxyfen and 0.01 g of BHT were added to 69.9 g of diethylene glycol monoethyl ether to prepare the control agent 1 of the present invention.
実施例２：
ｄ−フェノトリン１５ｇ、ピリプロキシフェン０．３ｇ、ＢＨＴ０．０１ｇをジエチレングリコールモノエチルエーテル８４．７ｇに加え、本発明の防除剤２を作製した。
Example 2:
15 g of d-phenothrin, 0.3 g of pyriproxyfen and 0.01 g of BHT were added to 84.7 g of diethylene glycol monoethyl ether to prepare the control agent 2 of the present invention.
実施例３：
ｄ−フェノトリン２０ｇ、ジョチュウギクエキス（総ピレトリン含量５０％）１０ｇ、ピリプロキシフェン０．５ｇ、ＢＨＴ０．０４ｇをケロシン６９．５ｇに加え、本発明の防除剤３を作製した。
Example 3:
20 g of d-phenothrin, 10 g of chrysanthemum extract (total pyrethrin content 50%), 0.5 g of pyriproxyfen and 0.04 g of BHT were added to 69.5 g of kerosene to prepare the control agent 3 of the present invention.
実施例４：
ｄ−フェノトリン２０ｇ、ピリプロキシフェン０．４ｇ、ＢＨＴ０．０１ｇをカプリル酸トリグリセライド７９．６ｇに加え、本発明の防除剤４を作製した。
Example 4:
20 g of d-phenothrin, 0.4 g of pyriproxyfen and 0.01 g of BHT were added to 79.6 g of caprylic acid triglyceride to prepare the control agent 4 of the present invention.
前記実施例にて作製した各防除剤を用いて蚊の動物への吸血試験を実施した。 A blood-sucking test on mosquito animals was carried out using each of the control agents prepared in the above Examples.
試験例１：
３０ｃｍ角のステンレス製金網籠の中にアカイエカ雌成虫約５０匹を放ち、砂糖水を与えて１昼夜飼育した。翌日、実験用マウスの背面中央部に所定量の本発明の防除剤を滴下し、４時間飼育した。その後、マウスを２０メッシュの金網で動き回らないように固定し、上記金網内に入れた。１日後、アカイエカ雌成虫を回収し、吸血虫数を調査した。
また、薬剤を滴下しない区を設け、無処理区とした。処理区と無処理区での吸血虫数から、以下のとおり吸血率および補正吸血阻害率を計算した。
About 50 adult mosquitoes were released in a 30 cm square stainless steel wire mesh cage and fed with sugar water and raised overnight. On the next day, a predetermined amount of the control agent of the present invention was dropped onto the center of the back of the experimental mouse and reared for 4 hours. Thereafter, the mouse was fixed so as not to move around with a 20-mesh wire mesh and placed in the wire mesh. One day later, female mosquito mosquitoes were collected, and the number of blood-sucking insects was investigated.
In addition, a section where no drug was dropped was provided, and it was set as an untreated section. From the number of blood sucking insects in the treated group and the untreated group, the blood sucking rate and the corrected blood sucking inhibition rate were calculated as follows.
試験例１の結果を表１に示す。
表１に示すとおり、防除剤１〜４の滴下により高い吸血阻害効果が確認できた。 As shown in Table 1, the high blood-sucking inhibitory effect was confirmed by dripping of the control agents 1-4.
試験例２：
猫（アメリカンショートヘア種、体重：３ｋｇ）の背部の前部、中央部、後部の３ヶ所に実施例３で得た防除剤３をシリンジを用いて０．３ｍＬずつ滴下した。滴下後１週間目と４週間目に防虫ネットで覆った５０×４０×７０ｃｍのケージに猫を入れ、このケージにヒトスジシマカ雌成虫３０〜５０匹を放ち、２７℃で猫とヒトスジシマカ雌成虫を同居させた。
８時間同居させ、その後ヒトスジシマカ雌成虫を回収して、吸血虫数を調査した。また、薬剤を滴下していない区を無処理区として設け、処理区と無処理区での吸血虫数から、試験例１と同様に吸血率および補正吸血阻害率を計算した。
Test example 2:
0.3 mL of the control agent 3 obtained in Example 3 was dropped at three locations on the front, center, and rear of the back of a cat (American shorthair, weight: 3 kg) using a syringe. Cats are placed in a 50 x 40 x 70 cm cage covered with an insect repellent net 1 week and 4 weeks after dropping, and 30 to 50 adults of female white striped mosquitoes are released into this cage. I let you.
The animals were allowed to live for 8 hours, and then the female adult female Aedes albopictus was collected and the number of sucking insects was investigated. In addition, a section where no drug was dropped was provided as an untreated section, and the blood sucking rate and the corrected blood sucking inhibition ratio were calculated in the same manner as in Test Example 1 from the number of blood sucking insects in the treated group and the untreated section.
試験例２の結果を表２に示す。
表２に示すとおり、防除剤３の滴下により、約１ヶ月後において高い吸血阻害が確認できた。 As shown in Table 2, high blood-sucking inhibition was confirmed after about 1 month by dripping the control agent 3.
Claims (6)
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