JP2010540448A - 非経口投与に適したセフェム誘導体を含む可溶製剤 - Google Patents
非経口投与に適したセフェム誘導体を含む可溶製剤 Download PDFInfo
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- A61K31/546—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
- A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
- A61K47/183—Amino acids, e.g. glycine, EDTA or aspartame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Dermatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US97419407P | 2007-09-21 | 2007-09-21 | |
| PCT/US2008/076920 WO2009039324A1 (en) | 2007-09-21 | 2008-09-19 | Soluble dosage forms containing cephem derivatives suitable for parenteral administration |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010540448A true JP2010540448A (ja) | 2010-12-24 |
| JP2010540448A5 JP2010540448A5 (enExample) | 2011-11-04 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010525983A Pending JP2010540448A (ja) | 2007-09-21 | 2008-09-19 | 非経口投与に適したセフェム誘導体を含む可溶製剤 |
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| Country | Link |
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| US (3) | US20090082326A1 (enExample) |
| EP (2) | EP2200618A4 (enExample) |
| JP (1) | JP2010540448A (enExample) |
| KR (1) | KR101599560B1 (enExample) |
| CN (3) | CN103919720A (enExample) |
| AU (1) | AU2008302201A1 (enExample) |
| BR (1) | BRPI0816412A2 (enExample) |
| CA (1) | CA2700263A1 (enExample) |
| MX (1) | MX2010003112A (enExample) |
| RU (1) | RU2537237C2 (enExample) |
| WO (1) | WO2009039324A1 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PH12012500528A1 (en) * | 2009-09-21 | 2019-06-14 | Astrazeneca Ab | Compositions and methods for treating bacterial infections using caftaroline |
| JO3190B1 (ar) * | 2011-10-19 | 2018-03-08 | Otsuka Pharma Co Ltd | محلول للتناول عن طريق الفم |
| WO2016008393A1 (zh) * | 2014-07-14 | 2016-01-21 | 正大天晴药业集团股份有限公司 | 头孢罗膦氨基酸盐及其结晶 |
| CN104258403B (zh) * | 2014-09-28 | 2017-03-01 | 刘宗侠 | 一种西洛他唑组合物及其制备方法 |
| KR20170038214A (ko) * | 2015-09-30 | 2017-04-07 | (주)아모레퍼시픽 | 당산 및 플라보노이드를 포함하는 항균용 조성물 |
Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH02124823A (ja) * | 1988-11-02 | 1990-05-14 | Eisai Co Ltd | セファロスポリン含有注射用組成物 |
| JPH02124822A (ja) * | 1988-11-02 | 1990-05-14 | Eisai Co Ltd | セファロスポリン含有注射用組成物 |
| JPH03173822A (ja) * | 1989-09-30 | 1991-07-29 | Eisai Co Ltd | セファロスポリン系薬物を含有する注射用組成物 |
| JPH0840907A (ja) * | 1994-08-03 | 1996-02-13 | Meiji Seika Kaisha Ltd | セファロスポリン注射剤 |
| JP2002220395A (ja) * | 2000-08-10 | 2002-08-09 | Takeda Chem Ind Ltd | ホスホノセフェム化合物 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4028355A (en) * | 1974-01-23 | 1977-06-07 | Smithkline Corporation | Cephalosporin purification process |
| GB8729574D0 (en) * | 1987-12-18 | 1988-02-03 | Fujisawa Pharmaceutical Co | Water-soluble antibiotic composition |
| ATE171705T1 (de) * | 1989-03-30 | 1998-10-15 | Pfizer | Cephalosporine und ihre homologen, verfahren zu ihrer herstellung und pharmazeutische präparate |
| TW473479B (en) * | 1997-12-19 | 2002-01-21 | Takeda Chemical Industries Ltd | Phosphonocephem derivatives, their production and use |
| US7527807B2 (en) * | 2000-06-21 | 2009-05-05 | Cubist Pharmaceuticals, Inc. | Compositions and methods for increasing the oral absorption of antimicrobials |
| CA2418614C (en) * | 2000-08-10 | 2008-06-10 | Takeda Chemical Industries, Ltd. | Phosphonocephem compound |
| TWI344847B (en) * | 2003-04-28 | 2011-07-11 | Takeda Chemical Industries Ltd | Composition for injection |
-
2008
- 2008-09-19 AU AU2008302201A patent/AU2008302201A1/en not_active Abandoned
- 2008-09-19 EP EP20080832124 patent/EP2200618A4/en not_active Withdrawn
- 2008-09-19 CA CA2700263A patent/CA2700263A1/en not_active Abandoned
- 2008-09-19 US US12/233,662 patent/US20090082326A1/en not_active Abandoned
- 2008-09-19 MX MX2010003112A patent/MX2010003112A/es active IP Right Grant
- 2008-09-19 CN CN201410162742.4A patent/CN103919720A/zh active Pending
- 2008-09-19 RU RU2010115268/15A patent/RU2537237C2/ru not_active Application Discontinuation
- 2008-09-19 KR KR1020107008731A patent/KR101599560B1/ko not_active Expired - Fee Related
- 2008-09-19 EP EP15166135.2A patent/EP2952195A1/en not_active Withdrawn
- 2008-09-19 JP JP2010525983A patent/JP2010540448A/ja active Pending
- 2008-09-19 CN CN200880117449A patent/CN101868240A/zh active Pending
- 2008-09-19 BR BRPI0816412A patent/BRPI0816412A2/pt not_active IP Right Cessation
- 2008-09-19 WO PCT/US2008/076920 patent/WO2009039324A1/en not_active Ceased
- 2008-09-19 CN CN2012104792814A patent/CN102935065A/zh active Pending
-
2011
- 2011-09-19 US US13/235,874 patent/US20120010180A1/en not_active Abandoned
-
2015
- 2015-03-04 US US14/638,449 patent/US20150196572A1/en not_active Abandoned
Patent Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH02124823A (ja) * | 1988-11-02 | 1990-05-14 | Eisai Co Ltd | セファロスポリン含有注射用組成物 |
| JPH02124822A (ja) * | 1988-11-02 | 1990-05-14 | Eisai Co Ltd | セファロスポリン含有注射用組成物 |
| JPH03173822A (ja) * | 1989-09-30 | 1991-07-29 | Eisai Co Ltd | セファロスポリン系薬物を含有する注射用組成物 |
| JPH0840907A (ja) * | 1994-08-03 | 1996-02-13 | Meiji Seika Kaisha Ltd | セファロスポリン注射剤 |
| JP2002220395A (ja) * | 2000-08-10 | 2002-08-09 | Takeda Chem Ind Ltd | ホスホノセフェム化合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| CN101868240A (zh) | 2010-10-20 |
| KR20100075942A (ko) | 2010-07-05 |
| US20090082326A1 (en) | 2009-03-26 |
| RU2010115268A (ru) | 2011-10-27 |
| MX2010003112A (es) | 2010-08-11 |
| EP2200618A4 (en) | 2010-11-03 |
| CA2700263A1 (en) | 2009-03-26 |
| WO2009039324A1 (en) | 2009-03-26 |
| BRPI0816412A2 (pt) | 2017-05-16 |
| CN102935065A (zh) | 2013-02-20 |
| EP2952195A1 (en) | 2015-12-09 |
| CN103919720A (zh) | 2014-07-16 |
| KR101599560B1 (ko) | 2016-03-03 |
| US20150196572A1 (en) | 2015-07-16 |
| AU2008302201A1 (en) | 2009-03-26 |
| US20120010180A1 (en) | 2012-01-12 |
| RU2537237C2 (ru) | 2014-12-27 |
| EP2200618A1 (en) | 2010-06-30 |
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