JP2010530380A5 - - Google Patents
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- Publication number
- JP2010530380A5 JP2010530380A5 JP2010512555A JP2010512555A JP2010530380A5 JP 2010530380 A5 JP2010530380 A5 JP 2010530380A5 JP 2010512555 A JP2010512555 A JP 2010512555A JP 2010512555 A JP2010512555 A JP 2010512555A JP 2010530380 A5 JP2010530380 A5 JP 2010530380A5
- Authority
- JP
- Japan
- Prior art keywords
- phenyl
- methyl
- pyrrol
- piperazin
- ethane
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 CC(C(B(*c1c(C)c(*)c(*)c(*)c1C)C(*)C1*)*)N1C(C(c1c(*)[n](*)c(**)c1*)=*)=O Chemical compound CC(C(B(*c1c(C)c(*)c(*)c(*)c1C)C(*)C1*)*)N1C(C(c1c(*)[n](*)c(**)c1*)=*)=O 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07290755 | 2007-06-18 | ||
| EP07290755.3 | 2007-06-18 | ||
| PCT/EP2008/004459 WO2008155022A1 (en) | 2007-06-18 | 2008-06-04 | Pyrrole derivatives as p2y12 antagonists |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010530380A JP2010530380A (ja) | 2010-09-09 |
| JP2010530380A5 true JP2010530380A5 (https=) | 2011-07-07 |
| JP5371969B2 JP5371969B2 (ja) | 2013-12-18 |
Family
ID=39092503
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010512555A Expired - Fee Related JP5371969B2 (ja) | 2007-06-18 | 2008-06-04 | Ｐ２ｙ１２拮抗薬としてのピロール誘導体 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US7910576B2 (https=) |
| EP (1) | EP2167487B1 (https=) |
| JP (1) | JP5371969B2 (https=) |
| KR (1) | KR20100020478A (https=) |
| CN (1) | CN101679358B (https=) |
| AU (1) | AU2008266515B2 (https=) |
| BR (1) | BRPI0812912A2 (https=) |
| CA (1) | CA2690243A1 (https=) |
| IL (1) | IL202758A (https=) |
| MX (1) | MX2009013431A (https=) |
| MY (1) | MY148901A (https=) |
| WO (1) | WO2008155022A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008051440A1 (en) | 2006-10-20 | 2008-05-02 | Novartis Ag | Crystal modifications -3- (1h-ind0l-3-yl) -4- [2- (4-methyl-piperazin-1-yl) -quinazolin-4-yl] -pyrrole-2, 5-d ione |
| US9539246B2 (en) | 2011-08-30 | 2017-01-10 | University Of Utah Research Foundation | Methods and compositions for treating nephrogenic diabetes insipidus |
| DE102014108210A1 (de) | 2014-06-11 | 2015-12-17 | Dietrich Gulba | Rodentizid |
| MX2021012105A (es) | 2019-04-03 | 2021-11-03 | Aligos Therapeutics Inc | Compuestos de pirrol. |
| EP4070658A1 (de) | 2021-04-06 | 2022-10-12 | BIORoxx GmbH | Verwendung von blutgerinnungshemmenden verbindungen als rodentizide |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3458515A (en) * | 1966-07-21 | 1969-07-29 | American Home Prod | Piperazine substituted pyrroles |
| US20020061892A1 (en) * | 2000-02-22 | 2002-05-23 | Tao Wang | Antiviral azaindole derivatives |
| US6861424B2 (en) | 2001-06-06 | 2005-03-01 | Schering Aktiengesellschaft | Platelet adenosine diphosphate receptor antagonists |
| US6956040B2 (en) * | 2001-07-16 | 2005-10-18 | Ranbaxy Laboratories Limited | Oxazolidinone piperazinyl derivatives as potential antimicrobials |
| DE60333866D1 (de) | 2002-12-11 | 2010-09-30 | Bayer Schering Pharma Ag | 2-aminocarbonlyl-chinolin-verbindungen als adenosin diphosphat plättchenrezeptor antagonisten |
| WO2005009971A1 (ja) | 2003-07-24 | 2005-02-03 | Astellas Pharma Inc. | キノロン誘導体又はその塩 |
| US7273881B2 (en) * | 2004-01-16 | 2007-09-25 | Bristol-Myers Squibb Company | Modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
| CN1778801A (zh) * | 2004-11-22 | 2006-05-31 | 中国农业科学院兰州畜牧与兽药研究所 | 喹诺酮7－((4－((z)－2－(2－氨基－4－噻唑基)－2－甲氧亚胺乙酰基)－1－哌嗪基)化合物及其制备方法 |
| BRPI0606437A (pt) * | 2005-01-06 | 2008-03-11 | Astrazeneca Ab | composto ou um sal farmaceuticamente aceitável do mesmo, composição farmacêutica, uso de um composto, e, método de tratamento de um distúrbio de agregação de plaqueta |
| JP2008094720A (ja) | 2005-01-20 | 2008-04-24 | Astellas Pharma Inc | キノロン誘導体のプロドラッグ又はその塩 |
| WO2006103544A2 (en) * | 2005-03-28 | 2006-10-05 | Pharmacia & Upjohn Company Llc | 4-piperazinylthieno [2, 3-d] pyrimidine compounds as platelet aggregation inhibitors |
| PT1951254E (pt) * | 2005-11-03 | 2012-04-12 | Portola Pharm Inc | [4-(6-halo-7-substituído-2,4-dioxo-1,4-di-hidro-2hquinazolin- 3-il)-fenil]-5-cloro-tiofen-2-il-sulfonilureias e formas e métodos relacionados com as mesmas |
| US20070259879A1 (en) * | 2006-03-06 | 2007-11-08 | Trimeris, Inc. | Piperazine and piperidine biaryl derivatives |
-
2008
- 2008-06-04 AU AU2008266515A patent/AU2008266515B2/en not_active Ceased
- 2008-06-04 MY MYPI20094985A patent/MY148901A/en unknown
- 2008-06-04 WO PCT/EP2008/004459 patent/WO2008155022A1/en not_active Ceased
- 2008-06-04 BR BRPI0812912-6A2A patent/BRPI0812912A2/pt not_active IP Right Cessation
- 2008-06-04 KR KR1020097026371A patent/KR20100020478A/ko not_active Ceased
- 2008-06-04 EP EP08759015.4A patent/EP2167487B1/en not_active Withdrawn - After Issue
- 2008-06-04 CA CA2690243A patent/CA2690243A1/en not_active Abandoned
- 2008-06-04 MX MX2009013431A patent/MX2009013431A/es active IP Right Grant
- 2008-06-04 CN CN2008800208356A patent/CN101679358B/zh not_active Expired - Fee Related
- 2008-06-04 JP JP2010512555A patent/JP5371969B2/ja not_active Expired - Fee Related
-
2009
- 2009-12-15 IL IL202758A patent/IL202758A/en not_active IP Right Cessation
- 2009-12-16 US US12/639,500 patent/US7910576B2/en not_active Expired - Fee Related
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