JP2010528009A5 - - Google Patents

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JP2010528009A5
JP2010528009A5 JP2010509367A JP2010509367A JP2010528009A5 JP 2010528009 A5 JP2010528009 A5 JP 2010528009A5 JP 2010509367 A JP2010509367 A JP 2010509367A JP 2010509367 A JP2010509367 A JP 2010509367A JP 2010528009 A5 JP2010528009 A5 JP 2010528009A5
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substituted
aryl
heteroaryl
heterocyclic
alkyl
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JP2010509367A
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Japanese (ja)
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JP5378362B2 (ja
JP2010528009A (ja
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Priority claimed from PCT/US2008/006475 external-priority patent/WO2008144062A1/en
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Publication of JP2010528009A5 publication Critical patent/JP2010528009A5/ja
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JP2010509367A 2007-05-21 2008-05-20 Ｃｓｆ−１ｒ阻害剤、組成物および使用方法 Expired - Fee Related JP5378362B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US93930307P 2007-05-21 2007-05-21
US60/939,303 2007-05-21
PCT/US2008/006475 WO2008144062A1 (en) 2007-05-21 2008-05-20 Csf-1r inhibitors, compositions, and methods of use

Publications (3)

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JP2010528009A JP2010528009A (ja) 2010-08-19
JP2010528009A5 true JP2010528009A5 (https=) 2011-07-07
JP5378362B2 JP5378362B2 (ja) 2013-12-25

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JP2010509367A Expired - Fee Related JP5378362B2 (ja) 2007-05-21 2008-05-20 Ｃｓｆ−１ｒ阻害剤、組成物および使用方法

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US (1) US8293769B2 (https=)
EP (1) EP2152700B1 (https=)
JP (1) JP5378362B2 (https=)
KR (1) KR20100017866A (https=)
CN (1) CN101754965B (https=)
AU (1) AU2008254425A1 (https=)
BR (1) BRPI0812159A2 (https=)
CA (1) CA2685967A1 (https=)
EA (1) EA200901548A1 (https=)
ES (1) ES2452349T3 (https=)
MX (1) MX2009012679A (https=)
WO (1) WO2008144062A1 (https=)

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KR101938431B1 (ko) 2011-05-05 2019-01-14 노파르티스 아게 뇌 종양의 치료를 위한 csf-1r 억제제
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JP2016506921A (ja) 2013-01-30 2016-03-07 バイエル ファーマ アクチエンゲゼルシャフト アミノ置換イソチアゾール
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US20230382871A1 (en) * 2020-09-23 2023-11-30 Shanghai Institute Of Materia Medica, Chinese Academy Of Sciences Csf1r kinase inhibitor and use thereof
US12043632B2 (en) 2020-12-23 2024-07-23 Ajax Therapeutics, Inc. 6-heteroaryloxy benzimidazoles and azabenzimidazoles as JAK2 inhibitors
WO2023009712A1 (en) * 2021-07-29 2023-02-02 Ajax Therapeutics, Inc. Heteroaryloxy thiazolo azines as jak2 inhibitors
US12162881B2 (en) 2021-11-09 2024-12-10 Ajax Therapeutics, Inc. Forms and compositions of inhibitors of JAK2
WO2023086319A1 (en) 2021-11-09 2023-05-19 Ajax Therapeutics, Inc. 6-he tero aryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors
CN115201383B (zh) * 2022-09-15 2022-12-20 常州合全药业有限公司 一种同时测定5-氯-2-硝基吡啶及其同分异构体的方法

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JP2007518823A (ja) * 2004-01-23 2007-07-12 アムゲン インコーポレイテッド キノリン、キナゾリン、ピリジン、及びピリミジン化合物と炎症、血管新生、及び癌に対する治療におけるそれら化合物の用途
EP1674466A1 (en) * 2004-12-27 2006-06-28 4Sc Ag 2,5- and 2,6-disubstituted benzazole analogues useful as protein kinase inhibitors
CA2649288C (en) 2006-04-19 2015-11-24 Novartis Ag 6-o-substituted benzoxazole and benzothiazole compounds and methods of inhibiting csf-1r signaling

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