JP2010520306A - エストロゲン関連受容体−αモジュレーターとしての置換フェノキシチアゾリジンジオン - Google Patents
エストロゲン関連受容体−αモジュレーターとしての置換フェノキシチアゾリジンジオン Download PDFInfo
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- JP2010520306A JP2010520306A JP2009552881A JP2009552881A JP2010520306A JP 2010520306 A JP2010520306 A JP 2010520306A JP 2009552881 A JP2009552881 A JP 2009552881A JP 2009552881 A JP2009552881 A JP 2009552881A JP 2010520306 A JP2010520306 A JP 2010520306A
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/44—Two oxygen atoms
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Applications Claiming Priority (2)
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|---|---|---|---|
| US89345307P | 2007-03-07 | 2007-03-07 | |
| PCT/US2008/056004 WO2008109727A1 (en) | 2007-03-07 | 2008-03-06 | Substituted phenoxy thiazolidinediones as estrogen related receptor-alpha modulators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010520306A true JP2010520306A (ja) | 2010-06-10 |
| JP2010520306A5 JP2010520306A5 (enExample) | 2011-03-24 |
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| Country | Link |
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| EP (1) | EP2129668A1 (enExample) |
| JP (1) | JP2010520306A (enExample) |
| KR (1) | KR20090127410A (enExample) |
| CN (1) | CN101679322A (enExample) |
| AR (1) | AR065655A1 (enExample) |
| AU (1) | AU2008222745A1 (enExample) |
| BR (1) | BRPI0808445A2 (enExample) |
| CA (1) | CA2679944A1 (enExample) |
| CL (1) | CL2008000670A1 (enExample) |
| CO (1) | CO6231008A2 (enExample) |
| EA (1) | EA200970837A1 (enExample) |
| EC (1) | ECSP099614A (enExample) |
| IL (1) | IL200757A0 (enExample) |
| MX (1) | MX2009009517A (enExample) |
| NI (1) | NI200900163A (enExample) |
| NZ (1) | NZ579372A (enExample) |
| SV (1) | SV2009003367A (enExample) |
| TW (1) | TW200902508A (enExample) |
| UA (1) | UA98485C2 (enExample) |
| WO (1) | WO2008109727A1 (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013532682A (ja) * | 2010-07-28 | 2013-08-19 | オーキッド ケミカルズ アンド ファーマシューティカルズ リミテッド | 肝臓、肺の障害、糖尿病合併症および心血管疾患の処置のためのジフェニルエーテル化合物 |
| JP2023501081A (ja) * | 2019-10-18 | 2023-01-18 | リード ファーマ ホールディング ビー．ブイ． | エストロゲン関連受容体アルファ（ＥＲＲα）モジュレーター |
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| CA2698929C (en) | 2007-09-14 | 2016-01-19 | Addex Pharma S.A. | 1,3-disubstituted-4-phenyl-1h-pyridin-2-ones |
| MY152078A (en) | 2007-09-14 | 2014-08-15 | Ortho Mcneil Janssen Pharm | 1',3'-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2h,1'h-[1,4']bipyridinyl-2'-ones |
| ES2637794T3 (es) | 2007-11-14 | 2017-10-17 | Janssen Pharmaceuticals, Inc. | Derivados de imidazo[1,2-A]piridina y su uso como moduladores alostéricos positivos de receptores MGLUR2 |
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| RU2517181C2 (ru) | 2008-10-16 | 2014-05-27 | Орто-Макнейл-Янссен Фармасьютикалз, Инк. | Производные индола и бензоморфолина в качестве модулятора метаботропных глутаматных рецепторов |
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| EP2383263B1 (en) * | 2008-12-30 | 2014-04-16 | Industry-academic Cooperation Foundation, Chosun University | Novel thiazolidinedione derivative and use thereof |
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| WO2015110435A1 (en) | 2014-01-21 | 2015-07-30 | Janssen Pharmaceutica Nv | Combinations comprising positive allosteric modulators or orthosteric agonists of metabotropic glutamatergic receptor subtype 2 and their use |
| HUE045610T2 (hu) | 2014-01-21 | 2020-01-28 | Janssen Pharmaceutica Nv | 2-es altípusú metabotróp glutamáterg receptor pozitív allosztérikus modulátorait vagy ortosztérikus agonistáit tartalmazó kombinációk és alkalmazásuk |
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| US20210393621A1 (en) | 2018-10-26 | 2021-12-23 | The Research Foundation For The State University Of New York | Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia |
| CN114341135B (zh) * | 2019-07-04 | 2025-03-18 | 领先制药控股公司 | 雌激素相关受体α(ERRα)调节剂 |
| CN112538038B (zh) * | 2019-09-20 | 2022-05-20 | 暨南大学 | 2-吲哚酮类ERRα反向激动剂及其药物组合物和应用 |
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| JPH09176162A (ja) * | 1995-12-22 | 1997-07-08 | Toubishi Yakuhin Kogyo Kk | チアゾリジンジオン誘導体及びその製造法並びにそれを含む医薬組成物 |
| WO2001025181A1 (en) * | 1999-10-01 | 2001-04-12 | Eisai Co., Ltd. | Carboxylic acid derivatives and drugs containing the same |
| WO2006019741A1 (en) * | 2004-07-14 | 2006-02-23 | Janssen Pharmaceutica N.V. | Arylidenes for the treatment of estrogen related receptor-alpha mediated diseases |
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| EP1398029A1 (en) | 2002-09-10 | 2004-03-17 | LION Bioscience AG | NR3B1 nuclear receptor binding 3-substituted pyrazole derivatives |
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| JP2010520307A (ja) * | 2007-03-07 | 2010-06-10 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | エストロゲン関連受容体−アルファモジュレーターとしての置換フェノキシｎ−アルキル置換チアゾリジンジオン |
-
2008
- 2008-03-06 WO PCT/US2008/056004 patent/WO2008109727A1/en not_active Ceased
- 2008-03-06 AU AU2008222745A patent/AU2008222745A1/en not_active Abandoned
- 2008-03-06 NZ NZ579372A patent/NZ579372A/en not_active IP Right Cessation
- 2008-03-06 TW TW097107941A patent/TW200902508A/zh unknown
- 2008-03-06 CN CN200880015196A patent/CN101679322A/zh active Pending
- 2008-03-06 JP JP2009552881A patent/JP2010520306A/ja active Pending
- 2008-03-06 CA CA002679944A patent/CA2679944A1/en not_active Abandoned
- 2008-03-06 US US12/043,269 patent/US7846953B2/en not_active Expired - Fee Related
- 2008-03-06 MX MX2009009517A patent/MX2009009517A/es active IP Right Grant
- 2008-03-06 BR BRPI0808445-9A patent/BRPI0808445A2/pt not_active IP Right Cessation
- 2008-03-06 EP EP08731504A patent/EP2129668A1/en not_active Ceased
- 2008-03-06 UA UAA200910123A patent/UA98485C2/ru unknown
- 2008-03-06 KR KR1020097020449A patent/KR20090127410A/ko not_active Withdrawn
- 2008-03-06 EA EA200970837A patent/EA200970837A1/ru unknown
- 2008-03-06 CL CL2008000670A patent/CL2008000670A1/es unknown
- 2008-03-07 AR ARP080100962A patent/AR065655A1/es not_active Application Discontinuation
-
2009
- 2009-09-04 NI NI200900163A patent/NI200900163A/es unknown
- 2009-09-06 IL IL200757A patent/IL200757A0/en unknown
- 2009-09-07 EC EC2009009614A patent/ECSP099614A/es unknown
- 2009-09-07 SV SV2009003367A patent/SV2009003367A/es unknown
- 2009-09-11 CO CO09097934A patent/CO6231008A2/es not_active Application Discontinuation
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2010
- 2010-10-07 US US12/899,812 patent/US8344009B2/en not_active Expired - Fee Related
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JPH09176162A (ja) * | 1995-12-22 | 1997-07-08 | Toubishi Yakuhin Kogyo Kk | チアゾリジンジオン誘導体及びその製造法並びにそれを含む医薬組成物 |
| WO2001025181A1 (en) * | 1999-10-01 | 2001-04-12 | Eisai Co., Ltd. | Carboxylic acid derivatives and drugs containing the same |
| WO2006019741A1 (en) * | 2004-07-14 | 2006-02-23 | Janssen Pharmaceutica N.V. | Arylidenes for the treatment of estrogen related receptor-alpha mediated diseases |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013532682A (ja) * | 2010-07-28 | 2013-08-19 | オーキッド ケミカルズ アンド ファーマシューティカルズ リミテッド | 肝臓、肺の障害、糖尿病合併症および心血管疾患の処置のためのジフェニルエーテル化合物 |
| JP2023501081A (ja) * | 2019-10-18 | 2023-01-18 | リード ファーマ ホールディング ビー．ブイ． | エストロゲン関連受容体アルファ（ＥＲＲα）モジュレーター |
| JP7629912B2 (ja) | 2019-10-18 | 2025-02-14 | リード ファーマ ホールディング ビー．ブイ． | エストロゲン関連受容体アルファ（ＥＲＲα）モジュレーター |
Also Published As
| Publication number | Publication date |
|---|---|
| KR20090127410A (ko) | 2009-12-11 |
| WO2008109727A8 (en) | 2009-12-17 |
| AR065655A1 (es) | 2009-06-24 |
| NZ579372A (en) | 2012-02-24 |
| US8344009B2 (en) | 2013-01-01 |
| CN101679322A (zh) | 2010-03-24 |
| EP2129668A1 (en) | 2009-12-09 |
| NI200900163A (es) | 2010-07-22 |
| SV2009003367A (es) | 2010-08-10 |
| TW200902508A (en) | 2009-01-16 |
| US20090111855A1 (en) | 2009-04-30 |
| CA2679944A1 (en) | 2008-09-12 |
| ECSP099614A (es) | 2009-10-30 |
| CO6231008A2 (es) | 2010-12-20 |
| US7846953B2 (en) | 2010-12-07 |
| AU2008222745A1 (en) | 2008-09-12 |
| MX2009009517A (es) | 2009-09-16 |
| UA98485C2 (ru) | 2012-05-25 |
| BRPI0808445A2 (pt) | 2014-08-05 |
| IL200757A0 (en) | 2010-05-17 |
| WO2008109727A1 (en) | 2008-09-12 |
| EA200970837A1 (ru) | 2010-04-30 |
| US20110237625A1 (en) | 2011-09-29 |
| CL2008000670A1 (es) | 2008-11-03 |
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