JP2010511019A5 - - Google Patents
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- Publication number
- JP2010511019A5 JP2010511019A5 JP2009538726A JP2009538726A JP2010511019A5 JP 2010511019 A5 JP2010511019 A5 JP 2010511019A5 JP 2009538726 A JP2009538726 A JP 2009538726A JP 2009538726 A JP2009538726 A JP 2009538726A JP 2010511019 A5 JP2010511019 A5 JP 2010511019A5
- Authority
- JP
- Japan
- Prior art keywords
- substituted
- unsubstituted
- alkyl
- compound
- heteroaryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US86814906P | 2006-12-01 | 2006-12-01 | |
| US99474007P | 2007-09-21 | 2007-09-21 | |
| PCT/EP2007/063108 WO2008065199A1 (en) | 2006-12-01 | 2007-11-30 | Imidazolopyridine compounds useful for the treatment of degenerative and inflammatory diseases |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010511019A JP2010511019A (ja) | 2010-04-08 |
| JP2010511019A5 true JP2010511019A5 (enExample) | 2010-12-09 |
Family
ID=39047973
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009538726A Pending JP2010511019A (ja) | 2006-12-01 | 2007-11-30 | 変性疾患及び炎症性疾患の治療に有用なイミダゾロピリジン化合物 |
Country Status (4)
| Country | Link |
|---|---|
| US (2) | US7951818B2 (enExample) |
| EP (1) | EP2099798A1 (enExample) |
| JP (1) | JP2010511019A (enExample) |
| WO (1) | WO2008065199A1 (enExample) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE602007012133D1 (de) * | 2006-12-01 | 2011-03-03 | Andrew Burritt | Triazolopyridinverbindungen zur behandlung von degenerations- und entzündungskrankheiten |
| JP2010511019A (ja) * | 2006-12-01 | 2010-04-08 | ガラパゴス・ナムローゼ・フェンノートシャップ | 変性疾患及び炎症性疾患の治療に有用なイミダゾロピリジン化合物 |
| CA2739344A1 (en) * | 2008-10-14 | 2010-04-22 | Actelion Pharmaceuticals Ltd | Phenethylamide derivatives and their heterocyclic analogues |
| CA2745871C (en) | 2008-12-08 | 2018-02-20 | Gilead Connecticut, Inc. | Imidazopyrazine syk inhibitors |
| PA8854101A1 (es) * | 2008-12-18 | 2010-07-27 | Ortho Mcneil Janssen Pharm | Derivados de imidazol bicíclicos sustituidos como moduladores de gamma secretasa |
| CN102325765B (zh) | 2009-02-06 | 2014-12-24 | 杨森制药公司 | 作为γ-分泌酶调节剂的取代的双环杂环化合物 |
| TWI461425B (zh) | 2009-02-19 | 2014-11-21 | Janssen Pharmaceuticals Inc | 作為伽瑪分泌酶調節劑之新穎經取代的苯并唑、苯并咪唑、唑并吡啶及咪唑并吡啶衍生物類 |
| MX2011011753A (es) | 2009-05-07 | 2011-11-29 | Janssen Pharmaceuticals Inc | Nuevos derivados sustitutos de indazol y aza-indazol como moduladores de la gamma secretasa. |
| SG177644A1 (en) | 2009-07-15 | 2012-03-29 | Janssen Pharmaceuticals Inc | Substituted triazole and imidazole derivatives as gamma secretase modulators |
| JP2013517246A (ja) | 2010-01-15 | 2013-05-16 | ジヤンセン・フアーマシユーチカルズ・インコーポレーテツド | γセクレターゼ調節物質としての新規置換二環トリアゾール誘導体 |
| EP2545052B1 (en) | 2010-03-11 | 2014-11-12 | Gilead Connecticut, Inc. | Imidazopyridines syk inhibitors |
| KR20140047032A (ko) | 2011-03-24 | 2014-04-21 | 얀센 파마슈티칼즈, 인코포레이티드 | 감마 세크레타제 조정제로서의 신규 치환 트리아졸릴 피페라진 및 트리아졸릴 피페리딘 유도체 |
| EA023045B1 (ru) | 2011-07-15 | 2016-04-29 | Янссен Фармасьютикалз, Инк. | Новые замещенные производные индола в качестве модуляторов гамма-секретазы |
| NZ702611A (en) | 2012-05-16 | 2016-10-28 | Cellzome Ltd | Substituted 3, 4 - dihydro - 2h - pyrido [1, 2 -a] pyrazine - 1, 6 - dione derivatives useful for the treatment of (inter alia) alzheimer’s disease |
| JP6275161B2 (ja) | 2012-12-20 | 2018-02-07 | ヤンセン ファーマシューティカ エヌ．ベー． | γセクレターゼ調節剤としての新規な三環式３，４−ジヒドロ−２Ｈ−ピリド［１，２−ａ］ピラジン−１，６−ジオン誘導体 |
| HK1212346A1 (en) | 2013-01-17 | 2016-06-10 | Janssen Pharmaceutica Nv | Novel substituted pyrido-piperazinone derivatives as gamma secretase modulators |
| US10562897B2 (en) | 2014-01-16 | 2020-02-18 | Janssen Pharmaceutica Nv | Substituted 3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-diones as gamma secretase modulators |
| CN107129496A (zh) * | 2017-06-02 | 2017-09-05 | 贵州大学 | 一种8‑碘‑6‑硝基‑咪唑并[1,2‑a]吡啶的制备工艺 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE9802794D0 (sv) | 1998-08-21 | 1998-08-21 | Astra Ab | New compounds |
| WO2004014908A1 (en) * | 2002-08-13 | 2004-02-19 | Warner-Lambert Company Llc | Heterobicylcic metalloproteinase inhibitors |
| WO2004026867A2 (en) * | 2002-09-19 | 2004-04-01 | Schering Corporation | Imidazopyridines as cyclin dependent kinase inhibitors |
| US20050288502A1 (en) * | 2004-06-25 | 2005-12-29 | Andersen Denise L | Substituted heterocyclic compounds and methods of use |
| US7893058B2 (en) * | 2006-05-15 | 2011-02-22 | Janssen Pharmaceutica Nv | Imidazolopyrazine compounds useful for the treatment of degenerative and inflammatory diseases |
| JP2010511019A (ja) * | 2006-12-01 | 2010-04-08 | ガラパゴス・ナムローゼ・フェンノートシャップ | 変性疾患及び炎症性疾患の治療に有用なイミダゾロピリジン化合物 |
-
2007
- 2007-11-30 JP JP2009538726A patent/JP2010511019A/ja active Pending
- 2007-11-30 EP EP07847622A patent/EP2099798A1/en not_active Withdrawn
- 2007-11-30 US US11/998,818 patent/US7951818B2/en not_active Expired - Fee Related
- 2007-11-30 WO PCT/EP2007/063108 patent/WO2008065199A1/en not_active Ceased
-
2011
- 2011-05-25 US US13/115,977 patent/US20120010206A1/en not_active Abandoned
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