JP2010506942A - Ｃｈｋ１阻害剤の組成物 - Google Patents
Ｃｈｋ１阻害剤の組成物 Download PDFInfo
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- JP2010506942A JP2010506942A JP2009533425A JP2009533425A JP2010506942A JP 2010506942 A JP2010506942 A JP 2010506942A JP 2009533425 A JP2009533425 A JP 2009533425A JP 2009533425 A JP2009533425 A JP 2009533425A JP 2010506942 A JP2010506942 A JP 2010506942A
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- alkylene
- cancer
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- alkyl
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Classifications
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- B—PERFORMING OPERATIONS; TRANSPORTING
- B82—NANOTECHNOLOGY
- B82Y—SPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
- B82Y5/00—Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
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| PCT/US2007/080150 WO2008067027A2 (en) | 2006-10-20 | 2007-10-02 | Compositions of chkl inhibitors and cyclodextrin |
Publications (2)
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| JP2010506942A true JP2010506942A (ja) | 2010-03-04 |
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| WO (1) | WO2008067027A2 (https=) |
| ZA (1) | ZA200902670B (https=) |
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| JP2014526512A (ja) * | 2011-09-18 | 2014-10-06 | ユーロ−セルティーク エス．エイ． | 医薬組成物 |
| JP2017155023A (ja) * | 2016-03-04 | 2017-09-07 | ジェイファーマ株式会社 | Ｌａｔ１阻害活性を有する芳香族アミノ酸誘導体を含有する注射剤 |
| JP2018203747A (ja) * | 2012-04-13 | 2018-12-27 | エル アンド エフ リサーチ，リミテッド ライアビリティー カンパニー | シクロデキストリンを使用するための方法 |
| JP2023026562A (ja) * | 2017-05-03 | 2023-02-24 | サイデックス・ファーマシューティカルズ・インコーポレイテッド | シクロデキストリン及びブスルファンを含有する組成物 |
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| US11020363B2 (en) | 2009-05-29 | 2021-06-01 | Cydex Pharmaceuticals, Inc. | Injectable nitrogen mustard compositions comprising a cyclodextrin derivative and methods of making and using the same |
| GB201008005D0 (en) | 2010-05-13 | 2010-06-30 | Sentinel Oncology Ltd | Pharmaceutical compounds |
| KR101995274B1 (ko) | 2011-10-03 | 2019-07-02 | 레스피버트 리미티드 | P38 map 키나제 저해제인 1-피라졸릴-3-(4-((2-아닐리노피리미딘-4-일)옥시)나프탈렌-1-일) 우레아 |
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| TWI573792B (zh) | 2012-02-01 | 2017-03-11 | 歐陸斯迪公司 | 新穎治療劑 |
| CN112472699A (zh) | 2013-07-26 | 2021-03-12 | 种族肿瘤学公司 | 改善比生群及衍生物的治疗益处的组合方法 |
| PT3357919T (pt) | 2014-02-14 | 2020-02-20 | Respivert Ltd | Compostos heterocíclicos aromáticos como compostos antiinflamatórios |
| GB201409471D0 (en) | 2014-05-28 | 2014-07-09 | Euro Celtique Sa | Pharmaceutical composition |
| GB201409488D0 (en) | 2014-05-28 | 2014-07-09 | Euro Celtique Sa | Pharmaceutical composition |
| GB201409485D0 (en) | 2014-05-28 | 2014-07-09 | Euro Celtique Sa | Pharmaceutical composition |
| US9890564B2 (en) | 2014-10-28 | 2018-02-13 | Sargent Manufacturing Company | Interconnected lock with direct drive for adjustable deadbolt to latchbolt spacing |
| US20200000840A1 (en) * | 2016-03-20 | 2020-01-02 | Asdera Llc | Use of cyclodextrins to reduce endocytosis in malignant and neurodegenerative disorders |
| AU2016426574B2 (en) | 2016-10-11 | 2023-07-13 | Euro-Celtique S.A. | Hodgkin lymphoma therapy |
| GB201709405D0 (en) | 2017-06-13 | 2017-07-26 | Euro Celtique Sa | Compounds for treating ovarian cancer |
| GB201709402D0 (en) | 2017-06-13 | 2017-07-26 | Euro Celtique Sa | Compounds for treating t-pll |
| GB201709406D0 (en) | 2017-06-13 | 2017-07-26 | Euro-Cletique S A | Compounds for treating TNBC |
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2007
- 2007-10-02 WO PCT/US2007/080150 patent/WO2008067027A2/en not_active Ceased
- 2007-10-02 MY MYPI20091558 patent/MY150649A/en unknown
- 2007-10-02 UA UAA200903745A patent/UA95310C2/ru unknown
- 2007-10-02 JP JP2009533425A patent/JP2010506942A/ja active Pending
- 2007-10-02 BR BRPI0717460-8A2A patent/BRPI0717460A2/pt not_active IP Right Cessation
- 2007-10-02 CN CN2007800390301A patent/CN101528215B/zh not_active Expired - Fee Related
- 2007-10-02 MX MX2009004214A patent/MX2009004214A/es active IP Right Grant
- 2007-10-02 EP EP07871106A patent/EP2063879A2/en not_active Withdrawn
- 2007-10-02 EA EA200900571A patent/EA200900571A1/ru unknown
- 2007-10-02 NZ NZ575394A patent/NZ575394A/en not_active IP Right Cessation
- 2007-10-02 AU AU2007325576A patent/AU2007325576B2/en not_active Ceased
- 2007-10-02 US US12/442,529 patent/US8455471B2/en not_active Expired - Fee Related
- 2007-10-02 CA CA2673483A patent/CA2673483C/en not_active Expired - Fee Related
- 2007-10-02 KR KR1020097007975A patent/KR20090065537A/ko not_active Ceased
- 2007-10-02 KR KR1020117017995A patent/KR20110098009A/ko not_active Ceased
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2009
- 2009-03-20 CR CR10680A patent/CR10680A/es unknown
- 2009-03-26 IL IL197869A patent/IL197869A/en not_active IP Right Cessation
- 2009-04-17 CO CO09039148A patent/CO6180503A2/es not_active Application Discontinuation
- 2009-04-17 ZA ZA200902670A patent/ZA200902670B/xx unknown
- 2009-04-17 TN TNP2009000146A patent/TN2009000146A1/fr unknown
- 2009-04-20 SV SV2009003227A patent/SV2009003227A/es unknown
- 2009-04-20 NO NO20091544A patent/NO20091544L/no not_active Application Discontinuation
- 2009-05-07 MA MA31850A patent/MA30872B1/fr unknown
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| WO2006105262A1 (en) * | 2005-03-29 | 2006-10-05 | Icos Corporation | HETEROARYL UREA DERIVATIVES USEFUL FOR INHIBITING CHKl |
| JP2008535830A (ja) * | 2005-03-29 | 2008-09-04 | イコス・コーポレイション | Ｃｈｋ１阻害に有用なヘテロアリール尿素誘導体 |
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| JP2014526512A (ja) * | 2011-09-18 | 2014-10-06 | ユーロ−セルティーク エス．エイ． | 医薬組成物 |
| JP2018039848A (ja) * | 2011-09-18 | 2018-03-15 | ユーロ−セルティーク エス．エイ． | 医薬組成物 |
| JP2018203747A (ja) * | 2012-04-13 | 2018-12-27 | エル アンド エフ リサーチ，リミテッド ライアビリティー カンパニー | シクロデキストリンを使用するための方法 |
| US10980828B2 (en) | 2012-04-13 | 2021-04-20 | L & F Research LLC | Method of using cyclodextrin |
| JP2017155023A (ja) * | 2016-03-04 | 2017-09-07 | ジェイファーマ株式会社 | Ｌａｔ１阻害活性を有する芳香族アミノ酸誘導体を含有する注射剤 |
| JP2023026562A (ja) * | 2017-05-03 | 2023-02-24 | サイデックス・ファーマシューティカルズ・インコーポレイテッド | シクロデキストリン及びブスルファンを含有する組成物 |
| JP7597778B2 (ja) | 2017-05-03 | 2024-12-10 | サイデックス・ファーマシューティカルズ・インコーポレイテッド | シクロデキストリン及びブスルファンを含有する組成物 |
Also Published As
| Publication number | Publication date |
|---|---|
| US8455471B2 (en) | 2013-06-04 |
| WO2008067027A3 (en) | 2009-04-16 |
| WO2008067027A2 (en) | 2008-06-05 |
| CA2673483C (en) | 2014-04-08 |
| KR20090065537A (ko) | 2009-06-22 |
| CN101528215B (zh) | 2011-10-19 |
| EP2063879A2 (en) | 2009-06-03 |
| BRPI0717460A2 (pt) | 2013-12-24 |
| MX2009004214A (es) | 2009-05-11 |
| CA2673483A1 (en) | 2008-06-05 |
| MA30872B1 (fr) | 2009-11-02 |
| CR10680A (es) | 2009-10-13 |
| UA95310C2 (ru) | 2011-07-25 |
| TN2009000146A1 (en) | 2010-10-18 |
| US20100022512A1 (en) | 2010-01-28 |
| AU2007325576B2 (en) | 2013-01-10 |
| IL197869A0 (en) | 2009-12-24 |
| CO6180503A2 (es) | 2010-07-19 |
| SV2009003227A (es) | 2010-02-04 |
| NO20091544L (no) | 2009-06-10 |
| NZ575394A (en) | 2012-01-12 |
| ZA200902670B (en) | 2010-06-30 |
| KR20110098009A (ko) | 2011-08-31 |
| IL197869A (en) | 2013-11-28 |
| MY150649A (en) | 2014-02-14 |
| CN101528215A (zh) | 2009-09-09 |
| AU2007325576A1 (en) | 2008-06-05 |
| EA200900571A1 (ru) | 2009-12-30 |
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