JP2010506942A - Ｃｈｋ１阻害剤の組成物 - Google Patents
Ｃｈｋ１阻害剤の組成物 Download PDFInfo
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- JP2010506942A JP2010506942A JP2009533425A JP2009533425A JP2010506942A JP 2010506942 A JP2010506942 A JP 2010506942A JP 2009533425 A JP2009533425 A JP 2009533425A JP 2009533425 A JP2009533425 A JP 2009533425A JP 2010506942 A JP2010506942 A JP 2010506942A
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- alkylene
- cancer
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- alkyl
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Classifications
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- B—PERFORMING OPERATIONS; TRANSPORTING
- B82—NANOTECHNOLOGY
- B82Y—SPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
- B82Y5/00—Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| PCT/US2007/080150 WO2008067027A2 (en) | 2006-10-20 | 2007-10-02 | Compositions of chkl inhibitors and cyclodextrin |
Publications (2)
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| JP2010506942A true JP2010506942A (ja) | 2010-03-04 |
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|---|---|---|---|---|
| JP2014526512A (ja) * | 2011-09-18 | 2014-10-06 | ユーロ−セルティーク エス．エイ． | 医薬組成物 |
| JP2017155023A (ja) * | 2016-03-04 | 2017-09-07 | ジェイファーマ株式会社 | Ｌａｔ１阻害活性を有する芳香族アミノ酸誘導体を含有する注射剤 |
| JP2018203747A (ja) * | 2012-04-13 | 2018-12-27 | エル アンド エフ リサーチ，リミテッド ライアビリティー カンパニー | シクロデキストリンを使用するための方法 |
| JP2023026562A (ja) * | 2017-05-03 | 2023-02-24 | サイデックス・ファーマシューティカルズ・インコーポレイテッド | シクロデキストリン及びブスルファンを含有する組成物 |
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| GB201008005D0 (en) | 2010-05-13 | 2010-06-30 | Sentinel Oncology Ltd | Pharmaceutical compounds |
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| PE20142355A1 (es) | 2011-10-03 | 2015-01-10 | Respivert Ltd | 1-pirazolil-3-(4-((2-anilinopirimidin-4-il)oxi)naftalen-1-il)ureas como inhibidores de proteinas cinasas activadas por mitogeno p38 |
| AR092790A1 (es) | 2012-02-01 | 2015-05-06 | Euro Celtique Sa | Derivados bencimidazolicos del acido hidroxamico |
| AU2014293013A1 (en) | 2013-07-26 | 2016-03-17 | Race Oncology Ltd. | Combinatorial methods to improve the therapeutic benefit of bisantrene |
| PT3357919T (pt) | 2014-02-14 | 2020-02-20 | Respivert Ltd | Compostos heterocíclicos aromáticos como compostos antiinflamatórios |
| GB201409485D0 (en) | 2014-05-28 | 2014-07-09 | Euro Celtique Sa | Pharmaceutical composition |
| GB201409471D0 (en) | 2014-05-28 | 2014-07-09 | Euro Celtique Sa | Pharmaceutical composition |
| GB201409488D0 (en) | 2014-05-28 | 2014-07-09 | Euro Celtique Sa | Pharmaceutical composition |
| US9890564B2 (en) | 2014-10-28 | 2018-02-13 | Sargent Manufacturing Company | Interconnected lock with direct drive for adjustable deadbolt to latchbolt spacing |
| EP3432880A4 (en) * | 2016-03-20 | 2019-12-11 | Asdera LLC | USE OF CYCLODEXTRINS TO REDUCE ENDOCYTOSIS IN MALIGNES AND NEURODEEGENERATIVE DISEASES |
| CA3040155C (en) | 2016-10-11 | 2024-01-16 | Euro-Celtique S.A. | Compound for use in the treatment of hodgkin lymphoma |
| GB201709403D0 (en) | 2017-06-13 | 2017-07-26 | Euro Celtique Sa | Compounds for treating sarcoma |
| GB201709406D0 (en) | 2017-06-13 | 2017-07-26 | Euro-Cletique S A | Compounds for treating TNBC |
| GB201709402D0 (en) | 2017-06-13 | 2017-07-26 | Euro Celtique Sa | Compounds for treating t-pll |
| GB201709405D0 (en) | 2017-06-13 | 2017-07-26 | Euro Celtique Sa | Compounds for treating ovarian cancer |
| JP2020535235A (ja) | 2017-09-28 | 2020-12-03 | アスデラ エルエルシー | リン脂質の調節異常が関与する疾患および障害におけるシクロデキストリンの使用 |
| CN109078005B (zh) * | 2018-08-07 | 2021-11-26 | 江苏领航生物科技有限公司 | 一种白消安组合物及其制备方法和应用 |
| JP2022522928A (ja) | 2018-12-18 | 2022-04-21 | ムンディファーマ・インターナショナル・コーポレーション・リミテッド | 多発性骨髄腫を治療するための化合物 |
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| WO2025034702A1 (en) | 2023-08-07 | 2025-02-13 | Revolution Medicines, Inc. | Rmc-6291 for use in the treatment of ras protein-related disease or disorder |
| WO2025080946A2 (en) | 2023-10-12 | 2025-04-17 | Revolution Medicines, Inc. | Ras inhibitors |
| WO2025171296A1 (en) | 2024-02-09 | 2025-08-14 | Revolution Medicines, Inc. | Ras inhibitors |
| WO2025217307A1 (en) | 2024-04-09 | 2025-10-16 | Revolution Medicines, Inc. | Methods for predicting response to a ras(on) inhibitor and combination therapies |
| WO2025240847A1 (en) | 2024-05-17 | 2025-11-20 | Revolution Medicines, Inc. | Ras inhibitors |
| WO2025255438A1 (en) | 2024-06-07 | 2025-12-11 | Revolution Medicines, Inc. | Methods of treating a ras protein-related disease or disorder |
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2007
- 2007-10-02 CA CA2673483A patent/CA2673483C/en not_active Expired - Fee Related
- 2007-10-02 AU AU2007325576A patent/AU2007325576B2/en not_active Ceased
- 2007-10-02 BR BRPI0717460-8A2A patent/BRPI0717460A2/pt not_active IP Right Cessation
- 2007-10-02 EA EA200900571A patent/EA200900571A1/ru unknown
- 2007-10-02 NZ NZ575394A patent/NZ575394A/en not_active IP Right Cessation
- 2007-10-02 US US12/442,529 patent/US8455471B2/en not_active Expired - Fee Related
- 2007-10-02 KR KR1020117017995A patent/KR20110098009A/ko not_active Ceased
- 2007-10-02 EP EP07871106A patent/EP2063879A2/en not_active Withdrawn
- 2007-10-02 WO PCT/US2007/080150 patent/WO2008067027A2/en not_active Ceased
- 2007-10-02 MX MX2009004214A patent/MX2009004214A/es active IP Right Grant
- 2007-10-02 MY MYPI20091558 patent/MY150649A/en unknown
- 2007-10-02 JP JP2009533425A patent/JP2010506942A/ja active Pending
- 2007-10-02 CN CN2007800390301A patent/CN101528215B/zh not_active Expired - Fee Related
- 2007-10-02 UA UAA200903745A patent/UA95310C2/ru unknown
- 2007-10-02 KR KR1020097007975A patent/KR20090065537A/ko not_active Ceased
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2009
- 2009-03-20 CR CR10680A patent/CR10680A/es unknown
- 2009-03-26 IL IL197869A patent/IL197869A/en not_active IP Right Cessation
- 2009-04-17 ZA ZA200902670A patent/ZA200902670B/xx unknown
- 2009-04-17 TN TNP2009000146A patent/TN2009000146A1/fr unknown
- 2009-04-17 CO CO09039148A patent/CO6180503A2/es not_active Application Discontinuation
- 2009-04-20 NO NO20091544A patent/NO20091544L/no not_active Application Discontinuation
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Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2014526512A (ja) * | 2011-09-18 | 2014-10-06 | ユーロ−セルティーク エス．エイ． | 医薬組成物 |
| JP2018039848A (ja) * | 2011-09-18 | 2018-03-15 | ユーロ−セルティーク エス．エイ． | 医薬組成物 |
| JP2018203747A (ja) * | 2012-04-13 | 2018-12-27 | エル アンド エフ リサーチ，リミテッド ライアビリティー カンパニー | シクロデキストリンを使用するための方法 |
| US10980828B2 (en) | 2012-04-13 | 2021-04-20 | L & F Research LLC | Method of using cyclodextrin |
| JP2017155023A (ja) * | 2016-03-04 | 2017-09-07 | ジェイファーマ株式会社 | Ｌａｔ１阻害活性を有する芳香族アミノ酸誘導体を含有する注射剤 |
| JP2023026562A (ja) * | 2017-05-03 | 2023-02-24 | サイデックス・ファーマシューティカルズ・インコーポレイテッド | シクロデキストリン及びブスルファンを含有する組成物 |
| JP7597778B2 (ja) | 2017-05-03 | 2024-12-10 | サイデックス・ファーマシューティカルズ・インコーポレイテッド | シクロデキストリン及びブスルファンを含有する組成物 |
Also Published As
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|---|---|
| CN101528215B (zh) | 2011-10-19 |
| WO2008067027A2 (en) | 2008-06-05 |
| WO2008067027A3 (en) | 2009-04-16 |
| US20100022512A1 (en) | 2010-01-28 |
| AU2007325576A1 (en) | 2008-06-05 |
| IL197869A (en) | 2013-11-28 |
| SV2009003227A (es) | 2010-02-04 |
| BRPI0717460A2 (pt) | 2013-12-24 |
| MA30872B1 (fr) | 2009-11-02 |
| CA2673483C (en) | 2014-04-08 |
| CN101528215A (zh) | 2009-09-09 |
| EP2063879A2 (en) | 2009-06-03 |
| TN2009000146A1 (en) | 2010-10-18 |
| NO20091544L (no) | 2009-06-10 |
| UA95310C2 (ru) | 2011-07-25 |
| KR20110098009A (ko) | 2011-08-31 |
| MY150649A (en) | 2014-02-14 |
| US8455471B2 (en) | 2013-06-04 |
| KR20090065537A (ko) | 2009-06-22 |
| CO6180503A2 (es) | 2010-07-19 |
| CR10680A (es) | 2009-10-13 |
| MX2009004214A (es) | 2009-05-11 |
| NZ575394A (en) | 2012-01-12 |
| CA2673483A1 (en) | 2008-06-05 |
| EA200900571A1 (ru) | 2009-12-30 |
| ZA200902670B (en) | 2010-06-30 |
| AU2007325576B2 (en) | 2013-01-10 |
| IL197869A0 (en) | 2009-12-24 |
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