JP2010502767A5 - - Google Patents

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Publication number
JP2010502767A5
JP2010502767A5 JP2009538434A JP2009538434A JP2010502767A5 JP 2010502767 A5 JP2010502767 A5 JP 2010502767A5 JP 2009538434 A JP2009538434 A JP 2009538434A JP 2009538434 A JP2009538434 A JP 2009538434A JP 2010502767 A5 JP2010502767 A5 JP 2010502767A5
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JP
Japan
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salt
compound
medicament
compound according
treating
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JP2009538434A
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English (en)
Japanese (ja)
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JP2010502767A (ja
JP5161237B2 (ja
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Priority claimed from PCT/US2007/078103 external-priority patent/WO2008033798A2/en
Publication of JP2010502767A publication Critical patent/JP2010502767A/ja
Publication of JP2010502767A5 publication Critical patent/JP2010502767A5/ja
Application granted granted Critical
Publication of JP5161237B2 publication Critical patent/JP5161237B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009538434A 2006-09-11 2007-09-11 Ｓｙｋキナーゼ阻害剤としてのピロロピラジン Expired - Fee Related JP5161237B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US82516806P 2006-09-11 2006-09-11
US60/825,168 2006-09-11
PCT/US2007/078103 WO2008033798A2 (en) 2006-09-11 2007-09-11 A pyrrolopyrazin as syk-kinase inhibitor

Publications (3)

Publication Number Publication Date
JP2010502767A JP2010502767A (ja) 2010-01-28
JP2010502767A5 true JP2010502767A5 (enExample) 2010-10-07
JP5161237B2 JP5161237B2 (ja) 2013-03-13

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ID=39032357

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009538434A Expired - Fee Related JP5161237B2 (ja) 2006-09-11 2007-09-11 Ｓｙｋキナーゼ阻害剤としてのピロロピラジン

Country Status (32)

Country Link
US (2) US8658649B2 (enExample)
EP (1) EP2094708B1 (enExample)
JP (1) JP5161237B2 (enExample)
KR (1) KR101443056B1 (enExample)
CN (2) CN103804383A (enExample)
AR (1) AR062745A1 (enExample)
AU (1) AU2007296592B8 (enExample)
BR (1) BRPI0716781A2 (enExample)
CA (1) CA2663175C (enExample)
CL (1) CL2007002617A1 (enExample)
CO (1) CO6160236A2 (enExample)
CR (1) CR10636A (enExample)
DK (1) DK2094708T3 (enExample)
ES (1) ES2437318T3 (enExample)
GT (1) GT200900055A (enExample)
HN (1) HN2009000455A (enExample)
IL (1) IL197381A (enExample)
MA (1) MA30781B1 (enExample)
MX (1) MX2009002616A (enExample)
MY (1) MY148107A (enExample)
NI (1) NI200900021A (enExample)
NO (1) NO20091265L (enExample)
NZ (1) NZ575496A (enExample)
PE (1) PE20081372A1 (enExample)
PT (1) PT2094708E (enExample)
RU (1) RU2440352C2 (enExample)
TN (2) TN2009000049A1 (enExample)
TW (1) TWI399379B (enExample)
UA (1) UA94622C2 (enExample)
UY (1) UY30584A1 (enExample)
WO (1) WO2008033798A2 (enExample)
ZA (1) ZA200901073B (enExample)

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EP2247595B1 (en) 2008-02-25 2011-07-20 F. Hoffmann-La Roche AG Pyrrolopyrazine kinase inhibitors
RU2503676C2 (ru) 2008-02-25 2014-01-10 Ф.Хоффманн-Ля Рош Аг Пирролопиразиновые ингибиторы киназы
DK2250172T3 (da) 2008-02-25 2012-01-16 Hoffmann La Roche Pyrrolopyrazinkinaseinhibitorer
ATE519763T1 (de) 2008-02-25 2011-08-15 Hoffmann La Roche Pyrrolopyrazin-kinasehemmer
ES2372908T3 (es) * 2008-02-25 2012-01-27 F. Hoffmann-La Roche Ag Inhibidores de la pirrolopirazina quinasa.
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PA8851701A1 (es) 2008-12-03 2010-07-27 Sanofi Aventis Tratamiento para la glomerulonefritis
TW201033211A (en) 2008-12-04 2010-09-16 Sanofi Aventis Crystalline forms
AR074776A1 (es) * 2008-12-18 2011-02-09 Sanofi Aventis Metodo para tratar la degeneracion macular; modulando el sistema inmunitario del paciente
US20110112101A1 (en) * 2009-03-05 2011-05-12 Sanofi-Aventis Treatment for ocular-related disorders
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SG181857A1 (en) 2009-12-23 2012-07-30 Takeda Pharmaceutical Fused heteroaromatic pyrrolidinones as syk inhibitors
US8481541B2 (en) 2010-03-22 2013-07-09 Hoffmann-La Roche Inc. Pyrrolopyrazine kinase inhibitors
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AU2020242287A1 (en) 2019-03-21 2021-09-02 INSERM (Institut National de la Santé et de la Recherche Médicale) A Dbait molecule in combination with kinase inhibitor for the treatment of cancer
KR20220098759A (ko) 2019-11-08 2022-07-12 인쎄름 (엥스띠뛰 나씨오날 드 라 쌍떼 에 드 라 흐쉐르슈 메디깔) 키나제 억제제에 대해 내성을 획득한 암의 치료 방법
WO2021148581A1 (en) 2020-01-22 2021-07-29 Onxeo Novel dbait molecule and its use
CN116969927B (zh) * 2023-06-07 2024-03-19 中南民族大学 一种从荜茇中提取分离的化合物及该化合物在制备抗炎药物中的应用

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