JP2010502767A5 - - Google Patents

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Publication number
JP2010502767A5
JP2010502767A5 JP2009538434A JP2009538434A JP2010502767A5 JP 2010502767 A5 JP2010502767 A5 JP 2010502767A5 JP 2009538434 A JP2009538434 A JP 2009538434A JP 2009538434 A JP2009538434 A JP 2009538434A JP 2010502767 A5 JP2010502767 A5 JP 2010502767A5
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JP
Japan
Prior art keywords
salt
compound
medicament
compound according
treating
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JP2009538434A
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English (en)
Japanese (ja)
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JP2010502767A (ja
JP5161237B2 (ja
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Priority claimed from PCT/US2007/078103 external-priority patent/WO2008033798A2/en
Publication of JP2010502767A publication Critical patent/JP2010502767A/ja
Publication of JP2010502767A5 publication Critical patent/JP2010502767A5/ja
Application granted granted Critical
Publication of JP5161237B2 publication Critical patent/JP5161237B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009538434A 2006-09-11 2007-09-11 Ｓｙｋキナーゼ阻害剤としてのピロロピラジン Expired - Fee Related JP5161237B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US82516806P 2006-09-11 2006-09-11
US60/825,168 2006-09-11
PCT/US2007/078103 WO2008033798A2 (en) 2006-09-11 2007-09-11 A pyrrolopyrazin as syk-kinase inhibitor

Publications (3)

Publication Number Publication Date
JP2010502767A JP2010502767A (ja) 2010-01-28
JP2010502767A5 true JP2010502767A5 (enExample) 2010-10-07
JP5161237B2 JP5161237B2 (ja) 2013-03-13

Family

ID=39032357

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009538434A Expired - Fee Related JP5161237B2 (ja) 2006-09-11 2007-09-11 Ｓｙｋキナーゼ阻害剤としてのピロロピラジン

Country Status (32)

Country Link
US (2) US8658649B2 (enExample)
EP (1) EP2094708B1 (enExample)
JP (1) JP5161237B2 (enExample)
KR (1) KR101443056B1 (enExample)
CN (2) CN101511838A (enExample)
AR (1) AR062745A1 (enExample)
AU (1) AU2007296592B8 (enExample)
BR (1) BRPI0716781A2 (enExample)
CA (1) CA2663175C (enExample)
CL (1) CL2007002617A1 (enExample)
CO (1) CO6160236A2 (enExample)
CR (1) CR10636A (enExample)
DK (1) DK2094708T3 (enExample)
ES (1) ES2437318T3 (enExample)
GT (1) GT200900055A (enExample)
HN (1) HN2009000455A (enExample)
IL (1) IL197381A (enExample)
MA (1) MA30781B1 (enExample)
MX (1) MX2009002616A (enExample)
MY (1) MY148107A (enExample)
NI (1) NI200900021A (enExample)
NO (1) NO20091265L (enExample)
NZ (1) NZ575496A (enExample)
PE (1) PE20081372A1 (enExample)
PT (1) PT2094708E (enExample)
RU (1) RU2440352C2 (enExample)
TN (2) TN2009000050A1 (enExample)
TW (1) TWI399379B (enExample)
UA (1) UA94622C2 (enExample)
UY (1) UY30584A1 (enExample)
WO (1) WO2008033798A2 (enExample)
ZA (1) ZA200901073B (enExample)

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KR101261514B1 (ko) 2008-02-25 2013-05-07 에프. 호프만-라 로슈 아게 피롤로피라진 키나아제 저해제
CN101952295B (zh) 2008-02-25 2013-11-20 霍夫曼-拉罗奇有限公司 吡咯并吡嗪激酶抑制剂
CA2716223A1 (en) 2008-02-25 2009-09-03 F. Hoffmann-La Roche Ag Pyrrolopyrazine kinase inhibitors
EP2247593B1 (en) 2008-02-25 2011-08-10 F. Hoffmann-La Roche AG Pyrrolopyrazine kinase inhibitors
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AU2009322409A1 (en) 2008-12-04 2011-06-23 Sanofi Crystalline forms
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RU2012152354A (ru) 2010-05-20 2014-06-27 Ф. Хоффманн-Ля Рош Аг Производные пирролопиразина в качестве ингибиторов syk и jak
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EP2489663A1 (en) 2011-02-16 2012-08-22 Almirall, S.A. Compounds as syk kinase inhibitors
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JP6159028B2 (ja) 2013-07-31 2017-07-05 ギリアード サイエンシーズ， インコーポレイテッド Ｓｙｋ阻害剤
EP3942045A1 (en) 2019-03-21 2022-01-26 Onxeo A dbait molecule in combination with kinase inhibitor for the treatment of cancer
EP4054579A1 (en) 2019-11-08 2022-09-14 Institut National de la Santé et de la Recherche Médicale (INSERM) Methods for the treatment of cancers that have acquired resistance to kinase inhibitors
WO2021148581A1 (en) 2020-01-22 2021-07-29 Onxeo Novel dbait molecule and its use
CN116969927B (zh) * 2023-06-07 2024-03-19 中南民族大学 一种从荜茇中提取分离的化合物及该化合物在制备抗炎药物中的应用

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