JP2009531441A5 - - Google Patents
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- Publication number
- JP2009531441A5 JP2009531441A5 JP2009502946A JP2009502946A JP2009531441A5 JP 2009531441 A5 JP2009531441 A5 JP 2009531441A5 JP 2009502946 A JP2009502946 A JP 2009502946A JP 2009502946 A JP2009502946 A JP 2009502946A JP 2009531441 A5 JP2009531441 A5 JP 2009531441A5
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- JP
- Japan
- Prior art keywords
- formula
- compound
- salt
- composition
- patient
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 CC(C)CN(C[C@]([C@](Cc(cc1)ccc1C#N)NC(*)=O)O)S(c(cc1)ccc1OC)(=O)=O Chemical compound CC(C)CN(C[C@]([C@](Cc(cc1)ccc1C#N)NC(*)=O)O)S(c(cc1)ccc1OC)(=O)=O 0.000 description 3
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US78712606P | 2006-03-29 | 2006-03-29 | |
| US60/787,126 | 2006-03-29 | ||
| PCT/US2007/007564 WO2007126812A2 (en) | 2006-03-29 | 2007-03-29 | Process for preparation of hiv protease inhibitors |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012271186A Division JP2013082717A (ja) | 2006-03-29 | 2012-12-12 | Ｈｉｖプロテアーゼインヒビターの調製方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2009531441A JP2009531441A (ja) | 2009-09-03 |
| JP2009531441A5 true JP2009531441A5 (https=) | 2010-05-20 |
| JP5430395B2 JP5430395B2 (ja) | 2014-02-26 |
Family
ID=38323963
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009502946A Active JP5430395B2 (ja) | 2006-03-29 | 2007-03-29 | Ｈｉｖプロテアーゼインヒビターの調製方法 |
| JP2012271186A Withdrawn JP2013082717A (ja) | 2006-03-29 | 2012-12-12 | Ｈｉｖプロテアーゼインヒビターの調製方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012271186A Withdrawn JP2013082717A (ja) | 2006-03-29 | 2012-12-12 | Ｈｉｖプロテアーゼインヒビターの調製方法 |
Country Status (24)
| Country | Link |
|---|---|
| US (4) | US8173623B2 (https=) |
| EP (2) | EP1999133B1 (https=) |
| JP (2) | JP5430395B2 (https=) |
| KR (2) | KR101395377B1 (https=) |
| CN (2) | CN101448838B (https=) |
| AP (2) | AP2757A (https=) |
| AU (1) | AU2007245194B2 (https=) |
| BR (1) | BRPI0710199A2 (https=) |
| CA (1) | CA2647316C (https=) |
| DK (1) | DK1999133T3 (https=) |
| EA (2) | EA016140B1 (https=) |
| ES (2) | ES2430557T3 (https=) |
| HR (2) | HRP20080554B1 (https=) |
| IL (2) | IL194122A (https=) |
| MX (1) | MX2008012398A (https=) |
| NO (2) | NO342102B1 (https=) |
| NZ (2) | NZ596074A (https=) |
| PL (1) | PL1999133T3 (https=) |
| PT (1) | PT1999133E (https=) |
| SG (1) | SG170794A1 (https=) |
| SI (1) | SI1999133T1 (https=) |
| UA (1) | UA97241C2 (https=) |
| WO (1) | WO2007126812A2 (https=) |
| ZA (1) | ZA200808046B (https=) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8921415B2 (en) | 2009-01-29 | 2014-12-30 | Mapi Pharma Ltd. | Polymorphs of darunavir |
| PL2528923T3 (pl) | 2010-01-28 | 2015-01-30 | Mapi Pharma Ltd | Sposób wytwarzania darunawiru i pochodnych darunawiru |
| CN102190638A (zh) * | 2010-03-16 | 2011-09-21 | 中国科学院上海药物研究所 | 联芳基醇二胺类化合物、其药物组合物、制备方法及应用 |
| CN102584748B (zh) * | 2011-01-13 | 2015-02-11 | 浙江九洲药业股份有限公司 | 夫沙那韦中间体的制备方法 |
| EP2702045B1 (en) * | 2011-04-26 | 2017-10-18 | Mylan Laboratories Ltd. | Novel process for the preparation of etravirine |
| EP2634180A1 (en) | 2012-03-01 | 2013-09-04 | Lonza Ltd. | Enzymatic process for the preparation of butyrolactones |
| SI3333173T1 (sl) | 2012-10-03 | 2019-08-30 | Gilead Sciences, Inc. | Postopki za pripravo analogov protivirusnega nukleotida |
| CN103664976B (zh) * | 2013-12-12 | 2015-11-04 | 惠州市莱佛士制药技术有限公司 | 一种顺式六氢呋喃并[2,3-b]呋喃-3-醇的制备方法 |
| EP3104712B1 (en) * | 2014-02-12 | 2020-05-06 | Firmenich Incorporated | Improved process for the synthesis of substituted 1-benzyl-3-(1-(isoxazol-4-ylmethyl)-1h-pyrazol-4-yl)imidazolidine-2,4-diones |
| DK3236972T3 (en) | 2014-12-26 | 2021-10-04 | Univ Emory | Antivirale N4-hydroxycytidin-derivativer |
| JP6435907B2 (ja) * | 2015-02-16 | 2018-12-12 | 住友化学株式会社 | ヘキサヒドロフロフラノール誘導体の製造方法 |
| CN108610227B (zh) * | 2016-12-10 | 2021-02-09 | 中国科学院大连化学物理研究所 | 一种制备双环芳香化合物的方法 |
| JP6804790B1 (ja) | 2017-12-07 | 2020-12-23 | エモリー ユニバーシティー | Ｎ４−ヒドロキシシチジンおよび誘導体ならびにそれらに関連する抗ウイルス用途 |
| SG11202107145SA (en) | 2019-01-25 | 2021-08-30 | Univ Brown | Compositions and methods for treating, preventing or reversing age-associated inflammation and disorders |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU6828894A (en) * | 1993-05-14 | 1994-12-12 | Merck & Co., Inc. | Hiv protease inhibitors |
| AU1369001A (en) * | 1995-12-13 | 2001-03-22 | Abbott Laboratories | Retroviral protease inhibiting compounds |
| EP2314563A3 (en) | 1999-12-23 | 2012-04-04 | Ampac Fine Chemicals LLC | Improved preparation of 2S,3S-N-isobutyl-N-(2-hydroxy-3-amino-4-phenylbutyl)-p-nitrobenzenesulfonylamide hydrochloride and other derivatives of 2-hydroxy-1,3-diamines |
| AU2002255473A1 (en) * | 2000-10-24 | 2002-09-04 | Glaxo Group Limited | Process for preparing intermediates of hiv protease inhibitors |
| CN1561570A (zh) | 2001-07-20 | 2005-01-05 | 皇家菲利浦电子有限公司 | 振荡电路、具有这种振荡电路的变换器以及具有这种变换器的预调节器 |
| AU2003231765B9 (en) * | 2002-04-26 | 2010-01-28 | Gilead Sciences, Inc. | Cellular accumulation of phosphonate analogs of HIV protease inhibitor compounds and the compounds as such |
| US20050239054A1 (en) * | 2002-04-26 | 2005-10-27 | Arimilli Murty N | Method and compositions for identifying anti-HIV therapeutic compounds |
| US7273716B2 (en) * | 2003-04-25 | 2007-09-25 | Gilead Sciences, Inc. | Methods and compositions for identifying therapeutic compounds with GS-7340 ester hydrolase |
-
2007
- 2007-03-29 WO PCT/US2007/007564 patent/WO2007126812A2/en not_active Ceased
- 2007-03-29 NZ NZ596074A patent/NZ596074A/xx not_active IP Right Cessation
- 2007-03-29 CN CN2007800178888A patent/CN101448838B/zh active Active
- 2007-03-29 AU AU2007245194A patent/AU2007245194B2/en active Active
- 2007-03-29 NZ NZ571302A patent/NZ571302A/en not_active IP Right Cessation
- 2007-03-29 EP EP07754134.0A patent/EP1999133B1/en active Active
- 2007-03-29 HR HRP20080554AA patent/HRP20080554B1/hr not_active IP Right Cessation
- 2007-03-29 UA UAA200811574A patent/UA97241C2/uk unknown
- 2007-03-29 SI SI200731323T patent/SI1999133T1/sl unknown
- 2007-03-29 ES ES07754134T patent/ES2430557T3/es active Active
- 2007-03-29 AP AP2008004641A patent/AP2757A/xx active
- 2007-03-29 KR KR1020137034899A patent/KR101395377B1/ko active Active
- 2007-03-29 PT PT77541340T patent/PT1999133E/pt unknown
- 2007-03-29 BR BRPI0710199-6A patent/BRPI0710199A2/pt not_active IP Right Cessation
- 2007-03-29 US US11/729,522 patent/US8173623B2/en active Active
- 2007-03-29 EP EP12192910.3A patent/EP2570416B1/en active Active
- 2007-03-29 JP JP2009502946A patent/JP5430395B2/ja active Active
- 2007-03-29 CN CN201110315578.2A patent/CN102516259B/zh active Active
- 2007-03-29 KR KR1020087026569A patent/KR101429300B1/ko active Active
- 2007-03-29 PL PL07754134T patent/PL1999133T3/pl unknown
- 2007-03-29 EA EA200802074A patent/EA016140B1/ru not_active IP Right Cessation
- 2007-03-29 AP AP2013006690A patent/AP2013006690A0/xx unknown
- 2007-03-29 DK DK07754134.0T patent/DK1999133T3/da active
- 2007-03-29 CA CA2647316A patent/CA2647316C/en active Active
- 2007-03-29 US US12/293,450 patent/US20110065631A1/en not_active Abandoned
- 2007-03-29 MX MX2008012398A patent/MX2008012398A/es active IP Right Grant
- 2007-03-29 ES ES12192910T patent/ES2572001T3/es active Active
- 2007-03-29 SG SG201102217-5A patent/SG170794A1/en unknown
- 2007-03-29 EA EA201100994A patent/EA020088B1/ru not_active IP Right Cessation
- 2007-03-29 HR HRP20140626AA patent/HRP20140626A2/hr not_active Application Discontinuation
-
2008
- 2008-09-16 IL IL194122A patent/IL194122A/en not_active IP Right Cessation
- 2008-09-19 ZA ZA200808046A patent/ZA200808046B/xx unknown
- 2008-10-28 NO NO20084547A patent/NO342102B1/no unknown
-
2012
- 2012-02-21 US US13/401,659 patent/US8431745B2/en active Active
- 2012-12-12 JP JP2012271186A patent/JP2013082717A/ja not_active Withdrawn
-
2013
- 2013-02-27 US US13/779,188 patent/US20130172295A1/en not_active Abandoned
- 2013-03-12 IL IL225167A patent/IL225167A/en not_active IP Right Cessation
-
2018
- 2018-01-17 NO NO20180086A patent/NO342965B1/no unknown
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