AU2002255473A1 - Process for preparing intermediates of hiv protease inhibitors - Google Patents

Process for preparing intermediates of hiv protease inhibitors

Info

Publication number
AU2002255473A1
AU2002255473A1 AU2002255473A AU2002255473A AU2002255473A1 AU 2002255473 A1 AU2002255473 A1 AU 2002255473A1 AU 2002255473 A AU2002255473 A AU 2002255473A AU 2002255473 A AU2002255473 A AU 2002255473A AU 2002255473 A1 AU2002255473 A1 AU 2002255473A1
Authority
AU
Australia
Prior art keywords
protease inhibitors
hiv protease
preparing intermediates
intermediates
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2002255473A
Inventor
Roman Davis
Thomas Claiborne Lovelace
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of AU2002255473A1 publication Critical patent/AU2002255473A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2002255473A 2000-10-24 2001-10-22 Process for preparing intermediates of hiv protease inhibitors Abandoned AU2002255473A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24282200P 2000-10-24 2000-10-24
US60/242,822 2000-10-24
PCT/US2001/051428 WO2002067239A2 (en) 2000-10-24 2001-10-22 Process for preparing intermediates of hiv protease inhibitors

Publications (1)

Publication Number Publication Date
AU2002255473A1 true AU2002255473A1 (en) 2002-09-04

Family

ID=22916319

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2002255473A Abandoned AU2002255473A1 (en) 2000-10-24 2001-10-22 Process for preparing intermediates of hiv protease inhibitors

Country Status (4)

Country Link
EP (1) EP1404680A2 (en)
JP (1) JP2004519473A (en)
AU (1) AU2002255473A1 (en)
WO (2) WO2002067239A2 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050261507A1 (en) * 2002-06-27 2005-11-24 Doan Brian D Preparation of stereoisomers of (3alpha/beta, 6alpha/beta)hexahydrofuro[2,3-b]furan-3-ol
KR101429300B1 (en) * 2006-03-29 2014-08-11 길리애드 사이언시즈, 인코포레이티드 Process for preparation of hiv protease inhibitors
PL2089371T3 (en) 2006-11-09 2011-06-30 Janssen Sciences Ireland Uc Methods for the preparation of hexahydrofuro[2,3-b]furan-3-ol
CN103864813B (en) * 2012-12-18 2017-02-22 上海迪赛诺化学制药有限公司 Synthetic methods of hexahydrofuro[2,3-b]furan-3-ol and enantiomer thereof
CN107607635B (en) * 2017-08-15 2020-07-31 东北制药集团股份有限公司 Method for detecting content of propiolic alcohol in levophosphamide salt by adopting headspace gas chromatography
CR20220316A (en) 2019-12-06 2022-10-07 Vertex Pharma Substituted tetrahydrofurans as modulators of sodium channels
CN117794920A (en) 2021-06-04 2024-03-29 沃泰克斯药物股份有限公司 N- (hydroxyalkyl (hetero) aryl) tetrahydrofurancarboxamides as sodium channel modulators

Also Published As

Publication number Publication date
EP1404680A2 (en) 2004-04-07
WO2002067239A3 (en) 2004-01-08
WO2002067239A2 (en) 2002-08-29
WO2002060905A2 (en) 2002-08-08
JP2004519473A (en) 2004-07-02

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase