JP2009512658A5 - - Google Patents
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- Publication number
- JP2009512658A5 JP2009512658A5 JP2008535989A JP2008535989A JP2009512658A5 JP 2009512658 A5 JP2009512658 A5 JP 2009512658A5 JP 2008535989 A JP2008535989 A JP 2008535989A JP 2008535989 A JP2008535989 A JP 2008535989A JP 2009512658 A5 JP2009512658 A5 JP 2009512658A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutical composition
- composition according
- progestogen
- transdermal patch
- guestden
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 239000008194 pharmaceutical composition Substances 0.000 claims 10
- 239000000583 progesterone congener Substances 0.000 claims 8
- BFPYWIDHMRZLRN-UHFFFAOYSA-N 17alpha-ethynyl estradiol Natural products OC1=CC=C2C3CCC(C)(C(CC4)(O)C#C)C4C3CCC2=C1 BFPYWIDHMRZLRN-UHFFFAOYSA-N 0.000 claims 3
- BFPYWIDHMRZLRN-SLHNCBLASA-N Ethinyl estradiol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 BFPYWIDHMRZLRN-SLHNCBLASA-N 0.000 claims 3
- 229940011871 estrogen Drugs 0.000 claims 3
- 239000000262 estrogen Substances 0.000 claims 3
- 229960002568 ethinylestradiol Drugs 0.000 claims 3
- 239000013543 active substance Substances 0.000 claims 2
- 230000000694 effects Effects 0.000 claims 2
- SIGSPDASOTUPFS-XUDSTZEESA-N gestodene Chemical compound O=C1CC[C@@H]2[C@H]3CC[C@](CC)([C@](C=C4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 SIGSPDASOTUPFS-XUDSTZEESA-N 0.000 claims 2
- 229940095055 progestogen systemic hormonal contraceptives Drugs 0.000 claims 2
- 230000001568 sexual effect Effects 0.000 claims 2
- WWYNJERNGUHSAO-XUDSTZEESA-N (+)-Norgestrel Chemical compound O=C1CC[C@@H]2[C@H]3CC[C@](CC)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 WWYNJERNGUHSAO-XUDSTZEESA-N 0.000 claims 1
- 150000001875 compounds Chemical group 0.000 claims 1
- 229960004976 desogestrel Drugs 0.000 claims 1
- RPLCPCMSCLEKRS-BPIQYHPVSA-N desogestrel Chemical compound C1CC[C@@H]2[C@H]3C(=C)C[C@](CC)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 RPLCPCMSCLEKRS-BPIQYHPVSA-N 0.000 claims 1
- 229960005352 gestodene Drugs 0.000 claims 1
- 229940088597 hormone Drugs 0.000 claims 1
- 239000005556 hormone Substances 0.000 claims 1
- 229960004400 levonorgestrel Drugs 0.000 claims 1
- 239000000203 mixture Substances 0.000 claims 1
- 239000000825 pharmaceutical preparation Substances 0.000 claims 1
- 230000001105 regulatory effect Effects 0.000 claims 1
- JUNDJWOLDSCTFK-MTZCLOFQSA-N trimegestone Chemical compound C1CC2=CC(=O)CCC2=C2[C@@H]1[C@@H]1CC[C@@](C(=O)[C@@H](O)C)(C)[C@@]1(C)CC2 JUNDJWOLDSCTFK-MTZCLOFQSA-N 0.000 claims 1
- 229950008546 trimegestone Drugs 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102005050729A DE102005050729A1 (de) | 2005-10-19 | 2005-10-19 | Verfahren zur präventiven bedarfsweisen hormonalen Kontrazeption |
| PCT/EP2006/010273 WO2007045513A1 (de) | 2005-10-19 | 2006-10-19 | Verfahren zur präventiven bedarsweisen hormonalen kontrazeption |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013197047A Division JP2014001239A (ja) | 2005-10-19 | 2013-09-24 | 予防用要求次第ホルモン避妊方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009512658A JP2009512658A (ja) | 2009-03-26 |
| JP2009512658A5 true JP2009512658A5 (enExample) | 2009-12-10 |
Family
ID=37762565
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008535989A Withdrawn JP2009512658A (ja) | 2005-10-19 | 2006-10-19 | 予防用要求次第ホルモン避妊方法 |
| JP2013197047A Withdrawn JP2014001239A (ja) | 2005-10-19 | 2013-09-24 | 予防用要求次第ホルモン避妊方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013197047A Withdrawn JP2014001239A (ja) | 2005-10-19 | 2013-09-24 | 予防用要求次第ホルモン避妊方法 |
Country Status (13)
| Country | Link |
|---|---|
| US (3) | US20080311180A1 (enExample) |
| EP (1) | EP1937275A1 (enExample) |
| JP (2) | JP2009512658A (enExample) |
| KR (1) | KR20080056774A (enExample) |
| CN (1) | CN101340915A (enExample) |
| BR (1) | BRPI0617683A2 (enExample) |
| CA (1) | CA2626567C (enExample) |
| CR (1) | CR9908A (enExample) |
| DE (1) | DE102005050729A1 (enExample) |
| EC (1) | ECSP088390A (enExample) |
| GT (1) | GT200800038A (enExample) |
| HN (1) | HN2008000621A (enExample) |
| WO (1) | WO2007045513A1 (enExample) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090170823A1 (en) * | 2007-12-20 | 2009-07-02 | Duramed Pharmaceuticals, Inc. | Dosage Regimens and Pharmaceutical Compositions and Packages for Emergency Contraception |
| WO2010119029A1 (en) * | 2009-04-14 | 2010-10-21 | Laboratoire Hra-Pharma | Method for on-demand contraception |
| US20120129825A1 (en) * | 2009-04-14 | 2012-05-24 | Andre Ulmann | Method for on-demand contraception using levonorgestrel or norgestrel |
| DE102010040299A1 (de) | 2010-09-06 | 2012-03-08 | Bayer Schering Pharma Aktiengesellschaft | Transdermale therapeutische Systeme mit kristallisationsinhibierender Schutzfolie (Release Liner) |
| EP2782584B1 (en) | 2011-11-23 | 2021-06-09 | TherapeuticsMD, Inc. | Natural combination hormone replacement formulations and therapies |
| US9301920B2 (en) | 2012-06-18 | 2016-04-05 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
| US10806697B2 (en) | 2012-12-21 | 2020-10-20 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| US20150196640A1 (en) | 2012-06-18 | 2015-07-16 | Therapeuticsmd, Inc. | Progesterone formulations having a desirable pk profile |
| US10806740B2 (en) | 2012-06-18 | 2020-10-20 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
| US20130338122A1 (en) | 2012-06-18 | 2013-12-19 | Therapeuticsmd, Inc. | Transdermal hormone replacement therapies |
| SG11201503275RA (en) | 2012-11-22 | 2015-06-29 | Bayer Pharma AG | Use and application regimen of a pharmaceutical composition containing levonorgestrel and a cox inhibitor for on-demand contraception |
| US10471072B2 (en) | 2012-12-21 | 2019-11-12 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| US10568891B2 (en) | 2012-12-21 | 2020-02-25 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| US10537581B2 (en) | 2012-12-21 | 2020-01-21 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| US9180091B2 (en) | 2012-12-21 | 2015-11-10 | Therapeuticsmd, Inc. | Soluble estradiol capsule for vaginal insertion |
| US11266661B2 (en) | 2012-12-21 | 2022-03-08 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| US11246875B2 (en) | 2012-12-21 | 2022-02-15 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| CN105451737B (zh) | 2013-05-23 | 2018-04-10 | 拜耳医药股份有限公司 | 药物组合物及其用途以及所述药物组合物用于按需避孕的施用方法 |
| AR100562A1 (es) | 2014-05-22 | 2016-10-12 | Therapeuticsmd Inc | Composición farmacéutica de estradiol y progesterona para terapia de reemplazo hormonal |
| US10328087B2 (en) | 2015-07-23 | 2019-06-25 | Therapeuticsmd, Inc. | Formulations for solubilizing hormones |
| WO2017173044A1 (en) | 2016-04-01 | 2017-10-05 | Therapeuticsmd Inc. | Steroid hormone compositions in medium chain oils |
| KR20180126582A (ko) | 2016-04-01 | 2018-11-27 | 쎄러퓨틱스엠디, 인코퍼레이티드 | 스테로이드 호르몬 약제학적 조성물 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5512292A (en) * | 1990-10-29 | 1996-04-30 | Alza Corporation | Transdermal contraceptive formulations methods and devices |
| DE4229820C2 (de) * | 1992-09-07 | 1998-12-03 | Jenapharm Gmbh | Pharmazeutische Zubereitung auf Gestagen-Basis |
| DE4405898A1 (de) * | 1994-02-18 | 1995-08-24 | Schering Ag | Transdermale therapeutische Systeme enthaltend Sexualsteroide |
| NZ295365A (en) * | 1994-10-24 | 1999-07-29 | Schering Ag | Competitive progesterone antagonists for regulating female fertility as required |
| EP1605949A2 (en) * | 1999-08-31 | 2005-12-21 | Schering Aktiengesellschaft | Mesoprogestins (progesterone receptor modulators) as a component of female contraceptives |
| US7384650B2 (en) * | 1999-11-24 | 2008-06-10 | Agile Therapeutics, Inc. | Skin permeation enhancement composition for transdermal hormone delivery system |
| AU2003245252A1 (en) * | 2002-04-30 | 2003-11-17 | Fmc Corporation | Carrageenan based antimicrobial compositions |
| UA89766C2 (en) * | 2003-12-12 | 2010-03-10 | Байер Шеринг Фарма Акциенгезельшафт | Transdermal delivery system of gestodene |
| CN1913878B (zh) * | 2003-12-12 | 2010-05-26 | 拜耳先灵医药股份有限公司 | 无需渗透促进剂的激素透皮传递 |
-
2005
- 2005-10-19 DE DE102005050729A patent/DE102005050729A1/de not_active Withdrawn
-
2006
- 2006-10-19 CN CNA2006800480426A patent/CN101340915A/zh active Pending
- 2006-10-19 KR KR1020087011824A patent/KR20080056774A/ko not_active Ceased
- 2006-10-19 BR BRPI0617683-6A patent/BRPI0617683A2/pt not_active IP Right Cessation
- 2006-10-19 JP JP2008535989A patent/JP2009512658A/ja not_active Withdrawn
- 2006-10-19 EP EP06828860A patent/EP1937275A1/de not_active Withdrawn
- 2006-10-19 CA CA2626567A patent/CA2626567C/en not_active Expired - Fee Related
- 2006-10-19 WO PCT/EP2006/010273 patent/WO2007045513A1/de not_active Ceased
- 2006-10-19 US US12/090,719 patent/US20080311180A1/en not_active Abandoned
- 2006-10-19 US US11/583,143 patent/US20070111976A1/en not_active Abandoned
-
2008
- 2008-04-18 GT GT200800038A patent/GT200800038A/es unknown
- 2008-04-21 CR CR9908A patent/CR9908A/es not_active Application Discontinuation
- 2008-04-21 HN HN2008000621A patent/HN2008000621A/es unknown
- 2008-04-21 EC EC2008008390A patent/ECSP088390A/es unknown
-
2012
- 2012-05-29 US US13/482,023 patent/US20130089574A1/en not_active Abandoned
-
2013
- 2013-09-24 JP JP2013197047A patent/JP2014001239A/ja not_active Withdrawn
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