JP2009510037A5 - - Google Patents

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Publication number
JP2009510037A5
JP2009510037A5 JP2008532862A JP2008532862A JP2009510037A5 JP 2009510037 A5 JP2009510037 A5 JP 2009510037A5 JP 2008532862 A JP2008532862 A JP 2008532862A JP 2008532862 A JP2008532862 A JP 2008532862A JP 2009510037 A5 JP2009510037 A5 JP 2009510037A5
Authority
JP
Japan
Prior art keywords
formula
compound
pyran
dihydro
piperidinyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2008532862A
Other languages
English (en)
Japanese (ja)
Other versions
JP5209479B2 (ja
JP2009510037A (ja
Filing date
Publication date
Priority claimed from GBGB0519966.6A external-priority patent/GB0519966D0/en
Priority claimed from GB0602853A external-priority patent/GB0602853D0/en
Application filed filed Critical
Priority claimed from PCT/GB2006/003585 external-priority patent/WO2007036711A1/en
Publication of JP2009510037A publication Critical patent/JP2009510037A/ja
Publication of JP2009510037A5 publication Critical patent/JP2009510037A5/ja
Application granted granted Critical
Publication of JP5209479B2 publication Critical patent/JP5209479B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2008532862A 2005-09-30 2006-09-27 Ｍ１受容体にて活性を有するベンゾイミダゾロン類 Expired - Fee Related JP5209479B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0519966.6 2005-09-30
GBGB0519966.6A GB0519966D0 (en) 2005-09-30 2005-09-30 Compounds
GB0602853.4 2006-02-13
GB0602853A GB0602853D0 (en) 2006-02-13 2006-02-13 Compounds
PCT/GB2006/003585 WO2007036711A1 (en) 2005-09-30 2006-09-27 BENZIMIDAZOLONES WHICH HAVE ACTIVITY AT Ml RECEPTOR

Publications (3)

Publication Number Publication Date
JP2009510037A JP2009510037A (ja) 2009-03-12
JP2009510037A5 true JP2009510037A5 (https=) 2009-11-12
JP5209479B2 JP5209479B2 (ja) 2013-06-12

Family

ID=37398768

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008532862A Expired - Fee Related JP5209479B2 (ja) 2005-09-30 2006-09-27 Ｍ１受容体にて活性を有するベンゾイミダゾロン類

Country Status (4)

Country Link
US (1) US8288413B2 (https=)
EP (1) EP1937670A1 (https=)
JP (1) JP5209479B2 (https=)
WO (1) WO2007036711A1 (https=)

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BRPI0616609A2 (pt) 2005-09-30 2011-06-28 Glaxo Group Ltd compostos que têm atividade no receptor m1, composição farmacêutica contendo tais compostos, processo para preparação dos mesmos, bem como seus usos em medicina
WO2007036711A1 (en) 2005-09-30 2007-04-05 Glaxo Group Limited BENZIMIDAZOLONES WHICH HAVE ACTIVITY AT Ml RECEPTOR
EP1960389B1 (en) 2005-09-30 2012-08-15 Glaxo Group Limited Compounds which have activity at m1 receptor and their uses in medicine
GB0605785D0 (en) * 2006-03-22 2006-05-03 Glaxo Group Ltd Compounds
GB0605784D0 (en) * 2006-03-22 2006-05-03 Glaxo Group Ltd Compounds
GB0605786D0 (en) * 2006-03-22 2006-05-03 Glaxo Group Ltd Compounds
GB0706165D0 (en) * 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706170D0 (en) * 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706164D0 (en) * 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706174D0 (en) * 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
US8119661B2 (en) 2007-09-11 2012-02-21 Astrazeneca Ab Piperidine derivatives and their use as muscarinic receptor modulators
PE20091194A1 (es) * 2007-09-20 2009-09-05 Glaxo Group Ltd Derivados de heterociclicos como moduladores del receptor m1
WO2009037294A1 (en) * 2007-09-20 2009-03-26 Glaxo Group Limited Compounds which have activity at m1 receptor and their uses in medicine
GB0718415D0 (en) * 2007-09-20 2007-10-31 Glaxo Group Ltd Compounds
CN103497146B (zh) * 2013-09-27 2016-04-13 山东大学 2-(n-芳甲基哌啶-4-氨基)-4-(取代苯酚)苯环衍生物及其制备方法与应用
CN106045916B (zh) * 2016-05-31 2018-08-31 江苏之江化工有限公司 一种咪唑酮类化合物的合成方法
CN109206323A (zh) * 2017-07-07 2019-01-15 上海现代制药股份有限公司 一种萘胺药物中间体的制备方法

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US4292321A (en) 1979-05-24 1981-09-29 Warner-Lambert Company 1,3,8-Triazaspirodecane-4-ones, pharmaceutical compositions thereof and method of use thereof
DE3124366A1 (de) 1981-06-20 1982-12-30 Hoechst Ag, 6000 Frankfurt N-oxacyclyl-alkylpiperidin-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und deren verwendung
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ATE275141T1 (de) 1999-10-13 2004-09-15 Banyu Pharma Co Ltd Substituierte imidazolin-derivate
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BR0317230A (pt) 2002-12-13 2005-10-25 Smithkline Beecham Corp Composto, composição, métodos de antagonizar uma atividade do receptor de quimiocina ccr-5, e de tratar uma infecção viral em um paciente, e, uso de um composto
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WO2007036711A1 (en) 2005-09-30 2007-04-05 Glaxo Group Limited BENZIMIDAZOLONES WHICH HAVE ACTIVITY AT Ml RECEPTOR
EP1960389B1 (en) 2005-09-30 2012-08-15 Glaxo Group Limited Compounds which have activity at m1 receptor and their uses in medicine
BRPI0616609A2 (pt) 2005-09-30 2011-06-28 Glaxo Group Ltd compostos que têm atividade no receptor m1, composição farmacêutica contendo tais compostos, processo para preparação dos mesmos, bem como seus usos em medicina
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GB0706190D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706170D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706188D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706187D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706168D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706189D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706173D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706164D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706165D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706174D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds
GB0706167D0 (en) 2007-03-29 2007-05-09 Glaxo Group Ltd Compounds

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