JP2009501724A - 抗ウイルス性化合物 - Google Patents
抗ウイルス性化合物 Download PDFInfo
- Publication number
- JP2009501724A JP2009501724A JP2008521690A JP2008521690A JP2009501724A JP 2009501724 A JP2009501724 A JP 2009501724A JP 2008521690 A JP2008521690 A JP 2008521690A JP 2008521690 A JP2008521690 A JP 2008521690A JP 2009501724 A JP2009501724 A JP 2009501724A
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- JP
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- Prior art keywords
- alkyl
- cycloalkyl
- substituted
- alkenyl
- alkynyl
- Prior art date
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- 125000002221 trityl group Chemical group [H]C1=C([H])C([H])=C([H])C([H])=C1C([*])(C1=C(C(=C(C(=C1[H])[H])[H])[H])[H])C1=C([H])C([H])=C([H])C([H])=C1[H] 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/19—Cytokines; Lymphokines; Interferons
- A61K38/21—Interferons [IFN]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/572—Five-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
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- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
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- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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Applications Claiming Priority (3)
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| US69909605P | 2005-07-14 | 2005-07-14 | |
| US70055905P | 2005-07-18 | 2005-07-18 | |
| PCT/US2006/027605 WO2007009109A2 (en) | 2005-07-14 | 2006-07-14 | Antiviral compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009501724A true JP2009501724A (ja) | 2009-01-22 |
| JP2009501724A5 JP2009501724A5 (https=) | 2009-07-09 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008521690A Pending JP2009501724A (ja) | 2005-07-14 | 2006-07-14 | 抗ウイルス性化合物 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20070072809A1 (https=) |
| EP (1) | EP1907403B1 (https=) |
| JP (1) | JP2009501724A (https=) |
| KR (1) | KR101345008B1 (https=) |
| CN (1) | CN101243096B (https=) |
| AR (1) | AR054838A1 (https=) |
| AU (1) | AU2006267066A1 (https=) |
| BR (1) | BRPI0613056A2 (https=) |
| CA (1) | CA2614276A1 (https=) |
| MX (1) | MX2008000609A (https=) |
| NZ (1) | NZ564830A (https=) |
| TW (1) | TWI389908B (https=) |
| WO (1) | WO2007009109A2 (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2010503671A (ja) * | 2006-09-13 | 2010-02-04 | ノバルティス アクチエンゲゼルシャフト | 大環状ｈｃｖ阻害剤およびその使用 |
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| AU2006301966A1 (en) | 2005-10-11 | 2007-04-19 | Array Biopharma, Inc. | Compounds and methods for inhibiting hepatitis C viral replication |
| KR20090024834A (ko) * | 2006-07-05 | 2009-03-09 | 인터뮨, 인크. | Ｃ형 간염 바이러스 복제의 신규 억제제 |
| EP2049474B1 (en) | 2006-07-11 | 2015-11-04 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
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| JP7381190B2 (ja) | 2014-12-26 | 2023-11-15 | エモリー・ユニバーシテイ | Ｎ４－ヒドロキシシチジン及び誘導体並びにそれに関連する抗ウイルス用途 |
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2006
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- 2006-07-14 KR KR1020087003628A patent/KR101345008B1/ko not_active Expired - Fee Related
- 2006-07-14 CA CA002614276A patent/CA2614276A1/en not_active Abandoned
- 2006-07-14 AR ARP060103034A patent/AR054838A1/es not_active Application Discontinuation
- 2006-07-14 AU AU2006267066A patent/AU2006267066A1/en not_active Abandoned
- 2006-07-14 EP EP06787506.2A patent/EP1907403B1/en not_active Not-in-force
- 2006-07-14 WO PCT/US2006/027605 patent/WO2007009109A2/en not_active Ceased
- 2006-07-14 NZ NZ564830A patent/NZ564830A/en not_active IP Right Cessation
- 2006-07-14 US US11/487,542 patent/US20070072809A1/en not_active Abandoned
- 2006-07-14 JP JP2008521690A patent/JP2009501724A/ja active Pending
- 2006-07-14 BR BRPI0613056-9A patent/BRPI0613056A2/pt not_active IP Right Cessation
- 2006-07-14 CN CN2006800298851A patent/CN101243096B/zh not_active Expired - Fee Related
- 2006-07-14 MX MX2008000609A patent/MX2008000609A/es active IP Right Grant
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| WO2004000750A1 (en) * | 2000-09-15 | 2003-12-31 | Halliburton Energy Services, Inc. | Well cementing compositions and methods |
| WO2003099274A1 (en) * | 2002-05-20 | 2003-12-04 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
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| JP2010503671A (ja) * | 2006-09-13 | 2010-02-04 | ノバルティス アクチエンゲゼルシャフト | 大環状ｈｃｖ阻害剤およびその使用 |
Also Published As
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| AU2006267066A1 (en) | 2007-01-18 |
| WO2007009109A2 (en) | 2007-01-18 |
| US20070072809A1 (en) | 2007-03-29 |
| NZ564830A (en) | 2010-12-24 |
| KR20080027947A (ko) | 2008-03-28 |
| TW200738741A (en) | 2007-10-16 |
| EP1907403A2 (en) | 2008-04-09 |
| CA2614276A1 (en) | 2007-01-18 |
| BRPI0613056A2 (pt) | 2010-12-14 |
| CN101243096B (zh) | 2013-02-06 |
| WO2007009109A3 (en) | 2007-06-07 |
| CN101243096A (zh) | 2008-08-13 |
| MX2008000609A (es) | 2008-03-19 |
| EP1907403B1 (en) | 2013-12-25 |
| KR101345008B1 (ko) | 2013-12-31 |
| AR054838A1 (es) | 2007-07-18 |
| TWI389908B (zh) | 2013-03-21 |
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